微信关注
China
Total item
Cart Subtotal
￥ 0.00 “Tutalthromycin second gen”的搜索结果
42 个项目
每页
-
MK-2894 sodium salt
Catalog No. A11498 EP4 antagonistMK-2894 sodium salt is a highly potent and selective second generation EP4 antagonist. 了解更多 -
Becampanel
Catalog No. A21194 AMPA antagonistBecampanel (AMP397) is the first competitive AMPA antagonist and an antiepileptic agent. 了解更多 -
Olcegepant hydrochloride
Catalog No. A21900 CGRP1 receptor antagonistOlcegepant hydrochloride is the first potent and selective non-peptide antagonist of the calcitonin gene-related peptide 1 (CGRP1) receptor with IC50 of 0.03 nM and with a Ki of 14.4 pM for human CGRP. 了解更多 -
Enclomiphene citrate
Catalog No. A21830 oestrogen receptor antagonistEnclomiphene citrate is a potent and orally active oestrogen receptor antagonist, with antioestrogenic property. 了解更多 -
AZD9496 maleate
Catalog No. A21726 estrogen receptor (ERα) antagonistAZD9496 maleate is a potent and selective estrogen receptor (ERα) antagonist with IC50 of 0.28 nM. AZD9496 maleate is an orally bioavailable selective oestrogen receptor degrader (SERD). 了解更多 -
Ubrogepant
Catalog No. A21670 CGRP antagonistUbrogepant (MK-1602) is a novel oral calcitonin gene-related peptide receptor (CGRP) antagonist in development for acute treatment of migraine. 了解更多 -
H3B-6545 Hydrochloride
Catalog No. A21629 estrogen receptor covalent antagonistH3B-6545 Hydrochloride is an oral, selective estrogen receptor covalent antagonist (SERCA). 了解更多 -
Fulvestrant R enantiomer
Catalog No. A21545 estrogen receptor antagonistFulvestrant R enantiomer (ICI 182780 R enantiomer; ZD 9238 R enantiomer; ZM 182780 R enantiomer) is the less active R enantiomer of Fulvestrant. Fulvestrant is a potent estrogen receptor antagonist with an IC50 of 9.4 nM. 了解更多 -
ATN-161 trifluoroacetate salt
Catalog No. A21412 integrin α5β1 antagonistATN-161 trifluoroacetate salt is a novel integrin α5β1 antagonist, which inhibits angiogenesis and growth of liver metastases in a murine model. 了解更多 -
Tipelukast
Catalog No. A21249 leukotriene receptor antagonistTipelukast (KCA 757) is a sulfidopeptide leukotriene receptor antagonist, an orally bioavailable anti-inflammatory agent and used for the treatment of asthma. 了解更多 -
Radiprodil
Catalog No. A21193 NMDA NR2B antagonistRadiprodil (RGH-896) is an orally active and selective NMDA NR2B antagonist. A potential therapeutic agent in treatment of neuropathic pain and possibly other chronic pain conditions. 了解更多 -
Integrin Antagonists 27
Catalog No. A20895 integrin αvβ3 antagonistIntegrin Antagonists 27 is a small molecule integrin αvβ3 antagonist with binding affinity of 18 nM, as s novel anticancer agent. 了解更多 -
Sarpogrelate hydrochloride
Catalog No. A17295 5-HT2 antagonistSarpogrelate hydrochloride (MCI-9042), a selective 5-HT2 antagonist, has been widely used as an anti-platelet agent for the treatment of PAD. 了解更多 -
NPS-2143 hydrochloride
Catalog No. A11505 CaSR antagonistNPS-2143 hydrochloride (SB-262470A hydrochloride), an orally active calcilytic agent, is a selective and potent calcium ion-sensing receptor (CaSR) antagonist. 了解更多 -
Tripelennamine hydrochloride
Catalog No. A16767 H1-receptor antagonistTripelennamine hydrochloride, a H1-receptor antagonist, is a psychoactive drug and member of the pyridine andethylenediamine classes that is used as an antipruritic and first-generation antihistamine. 了解更多 -
ORM-15341
Catalog No. A12312 full antagonist for human AR (hAR)ORM-15341 is a potent and full antagonist for human AR (hAR) with IC50 values of 38 nM as shown by transactivation assays in AR-HEK293 cells stably expressing full-length hAR and an androgen-responsive luciferase reporter gene construct. 了解更多 -
Anisotropine Methylbromide (CB-154)
Catalog No. A17354 muscarinic antagonistAnisotropine methylbromide is a muscarinic antagonist and antispasmodic. Anisotropine methylbromide is a quaternary ammonium compound. Its use as treatment adjunct in peptic ulcer has been replaced by the use of more effective agents. 了解更多 -
Spironolactone
Catalog No. A17345 Androgen receptor antagonistSpironolactone is a potent antagonist of the androgen receptor. 了解更多 -
Lifitegrast
Catalog No. A17299 LFA-1 antagonistLifitegrast (SAR 1118) is an integrin lymphocyte function-associated antigen-1 (LFA-1) antagonist; inhibits Jurkat T cell attachment to ICAM-1 with an IC50 of 2.98 nM. 了解更多 -
(E/Z)-4-hydroxy Tamoxifen
Catalog No. A12532 Estrogen receptor 拮抗剂(E/Z)-4-hydroxy Tamoxifen是他莫昔芬的活性代谢产物，是一种选择性雌激素受体（ER）调节剂，广泛用于乳腺癌的治疗和化学预防治疗。 了解更多 -
AZD9496
Catalog No. A15822 -
ODM-201
Catalog No. A15797 -
(+)-MK 801 Maleate
Catalog No. A12761 -
N-desMethyl EnzalutaMide
Catalog No. A13964 -
StemRegenin 1 (SR1)
Catalog No. A12945 AhR 拮抗剂StemRegenin 1 (SR1)是一种细胞可渗透的嘌呤衍生物，作为芳香烃受体的拮抗剂，促进造血干细胞(HSC)的自我更新。 了解更多 -
17 alpha-propionate
Catalog No. A10009 -
Tamoxifen Citrate
Catalog No. A10885 Estrogen receptor 拮抗剂Tamoxifen Citrate是哺乳动物甾醇异构酶的选择性和有效抑制剂。 了解更多 -
Cyproterone acetate
Catalog No. A11409 Androgen Receptor 拮抗剂Cyproterone acetate是17-羟孕酮的合成衍生物，可作为雄激素受体拮抗剂以及具有弱孕激素和糖皮质激素活性的弱孕激素受体激动剂。 了解更多 -
Bicalutamide (Casodex)
Catalog No. A10142 Androgen Receptor 拮抗剂Bicalutamide (Casodex)是一种口服非甾体抗雄激素，用于治疗前列腺癌和多毛症。 了解更多 -
(R)-Bicalutamide
Catalog No. A10008 Androgen Receptor 拮抗剂(R)-Bicalutamide是一种活性的竞争性非甾体雄激素受体拮抗剂，对MDA 453细胞的IC50为0.17μM。 了解更多
42 个项目
每页
联系我们
United StatesAdooq Bioscience
Toll Free: (866) 930-6790
Fax: +1-323-606-8156
Email: sales@adooq.com
Not your Region? View all Distributors
FILTER BY:
Filtering:
- 作用机制: Antagonist (拮抗剂) 删除该内容
购物选项
- 分类
-
- Cytoskeleton (3)
- Cell Metabolism (2)
- GPCR / G Protein (7)
- Neuronal Signaling (2)
- Membrane Transporters/Ion Channels (1)
- Endocrinology / Hormones (19)
- Ready to Use Solution (4)
- Products On Sale (10)
ADOOQ 产品质量保证
We promise all products to perform as described.