“glucagon receptor”的搜索结果

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  1. Glucagon (19-29), human

    Catalog No. A14875
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    Ca 2+ /Mg 2+ -ATPase 抑制剂
    Glucagon (19-29), human是有效的Ca2+/Mg2+ -ATPase抑制剂。 了解更多
  2. Vildagliptin dihydrate

    Catalog No. A21898
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    DPP4 inhibitor
    Vildagliptin (LAF237 dihydrate;NVP-LAF 237 dihydrate) is a dipeptidyl peptidase 4 (DPP4) inhibitor that delays the degradation of glucagon-like peptide-1 (GLP-1). 了解更多
  3. ITI214 free base

    Catalog No. A21947
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    picomolar PDE1 inhibitor
    ITI-214 (free base) is a picomolar PDE1 inhibitor with excellent selectivity against other PDE family members and against a panel of enzymes, receptors, transporters, and ion channels, exhibits potent PDE1 inhibitory activity (Ki = 58 pM). 了解更多
  4. ITI214

    Catalog No. A21422
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    PDE1 inhibitor
    ITI-214 is a picomolar PDE1 inhibitor with excellent selectivity against other PDE family members and against a panel of enzymes, receptors, transporters, and ion channels, exhibits potent PDE1 inhibitory activity (Ki = 58 pM). 了解更多
  5. NOD-IN-1

    Catalog No. A13171
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    NOD-like receptors inhibitor
    NOD-IN-1 is a potent mixed inhibitor of nucleotide-binding oligomerization domain (NOD)-like receptors, NOD1 and NOD2, with IC50 of 5.74 μM and 6.45 μM, respectively. 了解更多
  6. MHP 133

    Catalog No. A20058
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    AChE /M1/M2/5HT4/I2 inhibitor
    MHP 133 is a drug with multiple CNS targets, and inhibits acetylcholinesterase (AChE) with Ki of 69 μM; also active against muscarinic M1 and M2 receptors, serotonin 5HT4 receptors, and imidazole I2 receptors. 了解更多
  7. PF-06250112

    Catalog No. A18612
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    BTK 抑制剂
    PF-06250112 is a potent, highly selective, orally bioavailable BTK inhibitor with an IC50 of 0.5 nM, shows inhibitory effect toward BMX nonreceptor tyrosine kinase and TEC with IC50s of 0.9 nM and 1.2 nM, respectively. 了解更多
  8. Anisodamine

    Catalog No. A18215
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    alpha-1 adrenergic receptors / mAChRs inhibitor
    Anisodamine is an inhibitor of alpha-1 adrenergic receptors and mAChRs isolated from Chinese solanacea plant. 了解更多
  9. Cangrelor Tetrasodium

    Catalog No. A17919
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    P2Y12 receptors inhibitor
    Cangrelor Tetrasodium is a high-affinity, reversible inhibitor of P2Y12 receptors that causes almost complete inhibition of ADP-induced platelet aggregate. It is a modified ATP derivative stable to enzymatic degradation. Unlike clopidogrel (Plavix), which is a prodrug, cangrelor is an active drug not requiring metabolic conversion. 了解更多
  10. Nefazodone hydrochloride

    Catalog No. A17622
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    5-HT2 receptors inhibitor
    Nefazodone HCl is an inhibitor of 5-HT2 receptors, SERT, NET, and hERG K+ channels used to treat mood disorders. It decreases immobility time in the forced swim test. 了解更多
  11. Cenicriviroc Mesylate

    Catalog No. A17028
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    CCR2/5 receptors 抑制剂
    Cenicriviroc(TAK-652,TBR-652)是CCR2和CCR5受体的抑制剂,可使其充当防止病毒进入人细胞的进入抑制剂 了解更多
  12. Imidafenacin

    Catalog No. A15490
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    M3 receptors 抑制剂
    Imidafenacin是一种有效的选择性M3受体抑制剂,Kb为0.317 nM。对M2受体的效力较低(IC50 = 4.13 nM)。 了解更多
  13. SB-505124 HCl

    Catalog No. A15232
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    TGF-β Receptors 抑制剂
    SB-505124 Hydrochloride是激活素受体样激酶(ALKS)的抑制剂。 了解更多
  14. Asenapine

    Catalog No. A18010
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    adrenergic receptor inhibitor
    Asenapine(Org 5222) inhibits adrenergic receptor (α1, α2A, α2B, α2C) with Ki of 0.25-1.2 nM and also inhibits 5-HT receptor (1A, 1B, 2A, 2B, 2C, 5A, 6, 7) with Ki of 0.03-4.0 nM. 了解更多
  15. LY223982

    Catalog No. A19436
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    LTB4 receptor inhibitor
    LY223982 is a potent and specific inhibitor of leukotriene B4 receptor, with an IC50 of 13.2 nM against [3H]LTB4 binding to LTB4 receptor. 了解更多
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    BUN60856

    Catalog No. A17233
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    cFMS Receptor Inhibitor
    BUN60856, also known as cFMS Receptor Inhibitor II, is a cFMS inhibitor. 了解更多
  16. Carotegrast

    Catalog No. A21997
    α4 integrin receptor inhibitor
    Carotegrast is an orally available α4 integrin receptor inhibitor with anti-inflammatories activities. 了解更多
  17. Eplivanserin mixture

    Catalog No. A21987
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    serotonin reuptake inhibitor/5-HT2A receptor antagonist
    Eplivanserin mixture is a selective serotonin reuptake inhibitor and a 5-HT2A receptor antagonist, extracted from patent WO 2005/002578 A1. 了解更多
  18. LDN193189 Tetrahydrochloride

    Catalog No. A21881
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    BMP type I receptor inhibitor
    LDN193189 Tetrahydrochloride is a selective BMP type I receptor inhibitor, which efficiently inhibits ALK2 and ALK3 (IC50=5 nM and 30 nM, respectively), with weaker effects on ALK4, ALK5 and ALK7 (IC50??500 nM). 了解更多
  19. Vilazodone D8

    Catalog No. A21876
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    SSR inhibitor / 5-HT1A receptor partial agonist
    Vilazodone D8 is the a deuterium labeled vilazodone, which is a combined serotonin specific reuptake inhibitor (SSRI) and 5-HT1A receptor partial agonist. 了解更多
  20. DDR1-IN-1 dihydrochloride

    Catalog No. A21813
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    DDR1 receptor tyrosine kinase inhibitor
    DDR1-IN-1 dihydrochloride is a potent and selective DDR1 receptor tyrosine kinase inhibitor with an IC50 of 105 nM; 4-fold less potent for DDR2 (IC50 = 413 nM). 了解更多
  21. Vortioxetine

    Catalog No. A21266
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    5-HT1A/5-HT1B/5-HT3A/5-HT7 receptor/SERT inhibitor
    Vortioxetine is a inhibitor of 5-HT1A, 5-HT1B, 5-HT3A, 5-HT7 receptor and SERT, with Ki values of 15 nM, 33 nM, 3.7 nM, 19 nM and 1.6 nM, respectively. 了解更多
  22. Clopidogrel thiolactone

    Catalog No. A20862
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    P2Y12 receptor inhibitor
    Clopidogrel thiolactone is a P2Y12 receptor inhibitor, is a potent antiplatelet agent. 了解更多
  23. Sunitinib

    Catalog No. A17858
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    multi-targeted receptor tyrosine kinase inhibitor
    Sunitinib (SU 11248) is a multi-targeted receptor tyrosine kinase inhibitor with IC50s of 80 nM and 2 nM for VEGFR2 and PDGFRβ, respectively. 了解更多
  24. SU14813 maleate

    Catalog No. A11556
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    multi-targeted receptor tyrosine kinases inhibitor
    SU14813 maleate is a multi-targeted receptor tyrosine kinases inhibitor with IC50s of 50, 2, 4, 15 nM for VEGFR2, VEGFR1, PDGFRβ and KIT. 了解更多
  25. IRAK inhibitor 2

    Catalog No. A11456
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    interleukin-1 receptor associated kinase inhibitor
    IRAK inhibitor 2 is interleukin-1 receptor associated kinase inhibitor . 了解更多
  26. Cabozantinib S-malate

    Catalog No. A11349
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    multiple receptor tyrosine kinases inhibitor
    Cabozantinib S-malate (XL184 S-malate) is a potent multiple receptor tyrosine kinases inhibitor that inhibits VEGFR2, c-Met, Kit, Axl and Flt3 with IC50s of 0.035, 1.3, 4.6, 7 and 11.3 nM, respectively. 了解更多
  27. Edicotinib

    Catalog No. A13008
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    CSF-1 receptor inhibitor
    Edicotinib is a selective and orally available colony-stimulating factor-1 (CSF-1) receptor inhibitor, and has entered phase IIA clinical trial to study rheumatoid arthritis (RA) despite disease. 了解更多
  28. LED209

    Catalog No. A12219
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    bacterial receptor QseC inhibitor
    LED209 is a potent small molecule inhibitor of bacterial receptor QseC, is a potent prodrug that is highly selective for QseC. 了解更多
  29. Sarcosine

    Catalog No. A16692
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    GlyT inhibitor/NMDA receptor
    Sarcosine is a glycine transporter type 1 (GlyT) inhibitor and an N-methyl-D-aspartate (NMDA) receptor co-agonist at the glycine binding site. 了解更多
  30. Darenzepine

    Catalog No. A12333
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    muscarinic receptor inhibitor
    Darenzepine is a muscarinic receptor inhibitor extracted from patent US 20170095465 A1. 了解更多
  31. S18-000003

    Catalog No. A19105
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    RORγt 抑制剂
    S18-000003 is a potent orally bioavailable retinoic acid receptor-related orphan receptor-gamma-t (RORγt) inhibitor with an IC50 of 29 nM. S18-000003 inhibits IL-17 production. 了解更多
  32. RU-301

    Catalog No. A19156
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    pan-TAM receptor inhibitor
    RU-301 is a pan-TAM receptor inhibitor, exerts pan-TAM inhibitory activity by binding at the interface between Gas6 and the Ig1 domain of the respective TAMs with Kd and IC50 values of 12 μM and 10 μM, respectively. 了解更多
  33. JTE-952

    Catalog No. A18391
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    CSF-1R 抑制剂
    TE-952 is a potent, oral active and selective Type II inhibitor of colony stimulating factor-1 receptor (CSF-1R or cFMS, type III receptor tyrosine kinase), with IC50 values of 13 nM and 261 nM for CSF1R and TrkA , respectively. Effective against a mouse collagen-induced model of arthritis. 了解更多
  34. FGFR1/DDR2 inhibitor 1

    Catalog No. A18716
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    FGFR1/DDR2 inhibitor
    FGFR1/DDR2 inhibitor 1 is an inhibitor of fibroblast growth factor receptor 1 (FGFR1) and discoindin domain receptor 2 (DDR2), with IC50 values of 31.1 nM, 108.4 nM and 3.2 nM for FGFR1, KG-1, and DDR2, respectively. 了解更多
  35. ALW-II-41-27

    Catalog No. A12493
    Eph receptor 抑制剂
    ALW-II-41-27是新型的Eph受体酪氨酸激酶抑制剂。 了解更多
  36. Asenapine HCl

    Catalog No. A15002
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    adrenergic receptor/5-HT receptor 抑制剂
    Asenapine hydrochloride抑制肾上腺素能受体(α1,α2A,α2B,α2C)的Ki为0.25-1.2 nM,还抑制5-HT受体(1A,1B,2A,2B,2C,5A,6、7),Ki为0.03- 4.0 nM。 了解更多
  37. Reversine

    Catalog No. A13250
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    human A3 adenosine receptor 拮抗剂 /Aurora 抑制剂
    Reversine是一种有效的人A3腺苷受体拮抗剂,Ki为0.66μM,是一种泛光A/B/C激酶抑制剂,IC50分别为12 nM/13 nM/20 nM。也用于干细胞去分化。 了解更多
  38. Fexofenadine HCl

    Catalog No. A11859
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    COX 抑制剂/histamine H1 receptor 激动剂
    Fexofenadine Hydrochloride是一种抗组胺药,可抑制Cox-1,Cox-2,并且是组胺H1受体激动剂,IC50为246 nM。 了解更多
  39. BBT594

    Catalog No. A21039
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    RET inhibitor
    BBT594 is a potent receptor tyrosine kinase RET inhibitor, used for cancer treatment. 了解更多
  40. Nec-4

    Catalog No. A21033
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    RIP1 inhibitor
    Nec-4, a tricyclic derivative, is a potent receptor interacting protein 1 (RIP1) inhibitor, with an IC50 of 2.6 μM, Ki of 0.46 μM. 了解更多
  41. RIPK1-IN-4

    Catalog No. A21029
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    RIP1 kinase inhibitor
    RIPK1-IN-4 (compound 8) is a potent and selective type II kinase inhibitor of receptor interacting protein 1 (RIP1) kinase and binds to a DLG-out inactive form of RIP1 with an IC50s of 16 nM and 10 nM for RIP1 and ADP-Glo kinase. 了解更多
  42. AN-3485

    Catalog No. A20989
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    TLR inhibitor
    AN-3485 is a benzoxaborole analog, Toll-Like Receptor(TLR) inhibitor with IC50 values ranging from 18 to 580 nM. 了解更多
  43. Leptomycin B

    Catalog No. A20985
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    nuclear export receptor CRM1 inhibitor
    Leptomycin B (CI 940; LMB) is a potent inhibitor of the nuclear export of proteins. Leptomycin B inactivates CRM1/exportin 1 by covalent modification at a cysteine residue. Leptomycin B is a potent antifungal antibiotic blocking the eukaryotic cell cycle. 了解更多
  44. AFP464

    Catalog No. A20978
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    HIF-1?? inhibitor
    AFP464, is an active HIF-1α inhibitor with an IC50 of 0.25 μM, also is a potent aryl hydrocarbon receptor (AhR) activator. 了解更多
  45. Clopidogrel

    Catalog No. A21206
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    platelet inhibitor
    Clopidogrel is a well-known and orally active platelet inhibitor that targets P2Y12 receptor. Clopidogrel is used to inhibit blood clots in coronary artery disease, peripheral vascular disease, and cerebrovascular disease. 了解更多
  46. Dovitinib lactate

    Catalog No. A21851
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    FGFR3 inhibitor
    Dovitinib(CHIR-258; TKI258) lactate is a potent inhibitor of fibroblast growth factor receptor 3 (FGFR3) with an IC50 of 5 nM. 了解更多
  47. HS-10296 hydrochloride

    Catalog No. A21661
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    EGFR/T790M inhibitor
    HS-10296 hydrochloride is an orally available and third-Generation inhibitor of epidermal growth factor receptor (EGFR)-activating mutations and T790M-resistant mutation with limited activity against wild-type EGFR. 了解更多
  48. TAS-115

    Catalog No. A21533
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    VEGFR/c-Met/HGFR inhibitor
    TAS-115 is a potent VEGFR and hepatocyte growth factor receptor (c-Met/HGFR)-targeted kinase inhibitor with IC50s of 30 and 32 nM for rVEGFR2 and rMET, respectively. 了解更多
  49. TAS-115 mesylate

    Catalog No. A21389
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    c-Met/HGFR inhibitor
    TAS-115 mesylate is a potent VEGFRand hepatocyte growth factor receptor (c-Met/HGFR)-targeted kinase inhibitor, with IC50s of 30 and 32 nM for rVEGFR2 and rMET, respectively. 了解更多

产品 1 到 50 共 111个

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