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￥ 0.00 “263”的搜索结果
40 个项目
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ABT-263 (Navitoclax)
Catalog No. A10022 Bcl-2 抑制剂ABT-263 (Navitoclax)是一种有效的Bcl-2家族抑制剂 (Bcl-2，Bcl-xL和Bcl-w的Ki <1 nmol/L)。ABT-263对Bcl- xL，Bcl-2和Bcl-w，( Ki≤1nmol/ L) 维持高亲和力，但与Mcl-1和A1的结合更弱。 了解更多 -
Centrinone
Catalog No. A20858 PLK4 inhibitorCentrinone (LCR-263) is a selective and reversible inhibitor of polo-like kinase 4 (PLK4) with a Ki of 0.16 nM. 了解更多 -
HG-9-91-01
Catalog No. A21004 SIK inhibitorHG-9-91-01 is a potent and highly selective salt-inducible kinase (SIK) inhibitor with IC50s of 0.92 nM, 6.6 nM and 9.6 nM for SIK1, SIK2 and SIK3 respectively. 了解更多 -
CK-666
Catalog No. A20973 Arp2/3 complex inhibitorCK-666 is a cell-permeable inhibitor of actin-related protein Arp2/3 complex, and binds to Arp2/3 complex, stabilizes the inactive state of the complex, blocking movement of the Arp2 and Arp3 subunits into the activated filament-like (short pitch) conformation. 了解更多 -
Galidesivir hydrochloride
Catalog No. A20930 RdRp inhibitorGalidesivir hydrochloride (BCX 4430 hydrochloride) is a viral RNA-dependent RNA polymerase (RdRp) inhibitor; demonstrated broad-spectrum activity in multiple viruses and a favorable preliminary preclinical safety profile. 了解更多 -
Petesicatib
Catalog No. A13394 cathepsin S inhibitorPetesicatib is a cathepsin S inhibitor, used in research of immune diseases. 了解更多 -
PF-06263276
Catalog No. A12572 pan-JAK inhibitorPF-06263276 (PF 6263276) is a potent and selective pan-JAK inhibitor, with IC50s of 2.2 nM, 23.1 nM, 59.9 nM and 29.7 nM for JAK1, JAK2, JAK3 and TYK2, respectively. 了解更多 -
CNT2 inhibitor-1
Catalog No. A12632 CNT2 InhibitorCNT2 inhibitor-1 is a potent concentrative nucleoside transporter 2 Inhibitor (CNT2), with an IC50 of 640 nM for hCNT2. 了解更多 -
Mutated EGFR-IN-2
Catalog No. A18565 EGFR 抑制剂Mutated EGFR-IN-2 (compound 91) is a mutant-selective EGFR inhibitor extracted from patent WO2017036263A1, which potently inhibits single-mutant EGFR (T790M) and double-mutant EGFR (including L858R/T790M (IC50=??1nM) and ex19del/T790M), and can suppress activity of single gain-of-function mutant EGFR (including L858R and ex19del) as well. Mutated EGFR-IN-2 shows anti-tumor antivity. 了解更多 -
PF-06726304
Catalog No. A16937 -
ARRY-380 (Irbinitinib)
Catalog No. A16413 -
Sildenafil
Catalog No. A12631 PDE5 抑制剂Sildenafil是选择性磷酸二酯酶5（PDE5）抑制剂之一（IC50 = 5.22 nM），被认为是治疗勃起功能障碍的最佳方法。 了解更多 -
PD 198306
Catalog No. A16032 -
Z-VDVAD-FMK
Catalog No. A12637 -
L-685458
Catalog No. A15899 -
AZD3759
Catalog No. A15551 -
Eliglustat tartrate
Catalog No. A15466 Glucocerebroside synthase 抑制剂Eliglustat tartrate通常用作酒石酸盐，据信Eliglustat通过抑制葡萄糖基神经酰胺合酶起作用。 了解更多 -
CDK9 inhibitor 2
Catalog No. A15039 -
Pepstatin A
Catalog No. A14262 -
CK-636
Catalog No. A13827 -
GSK2636771
Catalog No. A11784 -
PX-866 (Sonolisib)
Catalog No. A11261 -
Atazanavir
Catalog No. A10097 HIV Protease 抑制剂Atazanavir是一种氮杂肽及HIV-蛋白酶抑制剂，常与其他抗HIV药物结合，用于治疗HIV感染以及获得性免疫缺乏综合征。 了解更多 -
Atazanavir sulfate (BMS-232632-05)
Catalog No. A10096 HIV Protease 抑制剂Atazanavir sulfate (BMS-232632-05)是蛋白酶抑制剂（PI）类的抗逆转录病毒药物。是一种高选择性的 HIV-1蛋白酶抑制剂。 了解更多 -
BMS-690514
Catalog No. A11263 -
BMS-806 (BMS 378806)
Catalog No. A11201 HIV Entry 抑制剂BMS-806，也称为BMS-378806，选择性抑制HIV-1 gp120与CD4受体结合，EC50为0.85-26.5 nM。通过阻止HIV进入人体细胞而发挥作用。可阻断宿主细胞CD4与病毒gp120蛋白的结合，因此可抑制HIV-1感染的第一步。 了解更多 -
Cyt387 (Momelotinib)
Catalog No. A10263 JAK 抑制剂Cyt387 (Momelotinib)是Janus激酶JAK1和JAK2的抑制剂，可作为ATP竞争者，IC50值分别为11和18 nM。 了解更多 -
PD184352 (CI-1040)
Catalog No. A10212 MEK1/2 抑制剂PD184352 (CI-1040)是一种ATP非竞争性MEK1/2抑制剂，在基于细胞的测定中，IC50为17 nM，对MEK1/2的选择性是对MEK5的100倍。 了解更多 -
Temsirolimus (Torisel)
Catalog No. A10906
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