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￥ 0.00 “MK 1775”的搜索结果
27 个项目
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LY 344864 hydrochloride
Catalog No. A21748 5-HT1F agonistLY 344864 hydrochloride is a selective 5-HT1F agonist with a Ki of 6 nM. 了解更多 -
Taranabant ((1R,2R)stereoisomer)
Catalog No. A21705 CB1 receptor inverse agonistTaranabant (1R,2R)stereoisomer is the R-enantiomer of Taranabant. Taranabant is a highly potent and selective cannabinoid 1 (CB1) receptor inverse agonist. 了解更多 -
Taranabant racemate
Catalog No. A21699 CB1 antagonist/inverse agonistTaranabant racemate is an antagonist and/or inverse agonist of the Cannabinoid-1 (CB1) receptor extracted from patent WO 2004048317 A1. 了解更多 -
Ubrogepant
Catalog No. A21670 CGRP antagonistUbrogepant (MK-1602) is a novel oral calcitonin gene-related peptide receptor (CGRP) antagonist in development for acute treatment of migraine. 了解更多 -
Serlopitant
Catalog No. A21582 Neurokinin-1 (NK-1) receptor antagonistSerlopitant is a selective Neurokinin-1 (NK-1) receptor antagonist. 了解更多 -
Taranabant
Catalog No. A11578 CB1 receptor inverse agonistTaranabant is a highly potent and selective cannabinoid 1 (CB1) receptor inverse agonist that inhibits the binding and functional activity of various agonists, with a binding Ki of 0.13 nM for the human CB1R in vitro. 了解更多 -
MK-2894 sodium salt
Catalog No. A11498 EP4 antagonistMK-2894 sodium salt is a highly potent and selective second generation EP4 antagonist. 了解更多 -
Midodrine hydrochloride
Catalog No. A17757 Adrenergic alpha-1 agonistMidodrine hydrochloride is an ethanolamine derivative that is an adrenergic alpha-1 agonist. It is used as a vasoconstrictor agent in the treatment of hypotension. It improves clinical outcome of chronic hypotension. 了解更多 -
Tafluprost
Catalog No. A17442 prostaglandin analogueTafluprost, also known as MK2452 and AFP-168, is a prostaglandin analogue used topically (as eye drops) to control the progression of glaucoma and in the management of ocular hypertension. 了解更多 -
Bevenopran
Catalog No. A17110 opioid receptor antagonisBevenopran，也称为CB-5945，ADL-5945，MK-2402，OpRA III，是一种外周选择性μ-和δ-阿片样物质受体拮抗剂。 了解更多 -
MK-6096 (Filorexant)
Catalog No. A13168 Orexin receptor 拮抗剂MK-6096 (Filorexant)是目前正处于失眠临床开发中的口服生物利用型有效且选择性可逆的OX（1）R和OX（2）R拮抗剂。MK-6096表现出对人OX（1）R和OX（2）R的有效结合和拮抗作用（结合时<3 nM，FLIPR中为11 nM），对超过170个受体和 酶。 了解更多 -
MK-1064
Catalog No. A16360 -
MK-3697
Catalog No. A12633 -
Fosaprepitant dimeglumine
Catalog No. A11069 -
Vorapaxar (SCH 530348)
Catalog No. A12832 PAR-1 拮抗剂Vorapaxar (SCH 530348)是一种有效的口服活性凝血酶受体（PAR-1）拮抗剂，Ki为8.1 nM。 了解更多 -
MK-4305 (Suvorexant)
Catalog No. A11500 OX receptor 拮抗剂Suvorexant (MK-4305)是OX1R和OX2R的有效，选择性和口服可生物利用的拮抗剂，目前正在临床研究中作为失眠的新疗法。 了解更多 -
MK-0517 (Fosaprepitant)
Catalog No. A11756 neurokinin-1 receptor 拮抗剂MK-0517 (Fosaprepitant,L-758,298)是Aprepitant的水溶性磷酰基前药，它是NK1拮抗剂。 了解更多 -
Laropiprant (MK0524)
Catalog No. A11483 DP1 抑制剂Laropiprant (MK0524)与烟酸合用可降低血液胆固醇。是一种有效的，选择性的 DP receptor 拮抗剂，Ki 值为 0.57 nM，对 TP 受体的 Ki 值为 2.95 nM。 了解更多 -
MK-0974 (Telcagepant)
Catalog No. A11255 -
MK 3207 HCl
Catalog No. A10598 CGRP Receptor 拮抗剂MK 3207 hydrochloride是一种有效的CGRP受体拮抗剂，IC50为0.12 nM。 了解更多 -
Aprepitant (MK-0869)
Catalog No. A10083 neurokinin-1 receptor 拮抗剂Aprepitant (MK-0869)被归类为NK1拮抗剂。已经显示，阿瑞匹坦通过阻止P物质降落在大脑神经元受体上，从而抑制细胞毒性化疗药物引起的急性呕吐和延迟呕吐。还显示出它能增加5-HT3受体拮抗剂恩丹西酮和皮质类固醇地塞米松的活性，它们也可用于预防化学疗法引起的恶心和呕吐。 了解更多
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- 5-HT Receptors (1)
- Adrenergic Receptors (2)
- Opioid Receptors (1)
- G Protein (2)
- Prostanoid Receptors (4)
- Cannabinoid Receptors (3)
- Orexin Receptors (4)
- Neurokinin Receptors (4)
- Protease-Activated Receptors (PAR) (1)
- CGRP Receptor (4)
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- Inhibitor (抑制剂) (2)
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