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GPCR / G Protein

产品 151 到 200 共 229个

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  1. Kynurenic acid
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    Kynurenic acid

    Catalog No. A16581
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    GPR35/CXCR8 拮抗剂
    Kynurenic acid, an endogenous tryptophan metabolite, is a broad-spectrum antagonist targeting NMDA, glutamate, α7 nicotinic acetylcholine receptor. Kynurenic acid is also an agonist of GPR35/CXCR8. 了解更多
  2. PS372424
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    PS372424

    Catalog No. A19421
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    Human CXCR3 拮抗剂
    PS372424, a three amino-acid fragment of CXCL10, is a specific human CXCR3 agonist with anti-inflammatory activity, which inhibits the binding of CXCR3 ligand CXCL10 to CXCR3 receptor with IC50 of 42 nM. 了解更多
  3. DJ-V-159
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    DJ-V-159

    Catalog No. A18853
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    GPRC6A agonist
    DJ-V-159 is an agonist for G protein-coupled receptor family C group 6 member A (GPRC6A). 了解更多
  4. LY2922470
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    LY2922470

    Catalog No. A12181
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    GPR40 agonist
    LY2922470 is a potent, selective and orally available agonist of the G protein-coupled receptor 40 (GPR40), with EC50s of 7 nM, 1 nM and 3 nM for human GPR40, mouse GPR40 and rat GPR40, respectively. 了解更多
  5. PSN632408
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    PSN632408

    Catalog No. A20902
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    GPR119 receptors agonist
    PSN632408 is an optimized agonist of GPR119 receptors that shows similar potency to OEA at both recombinant mouse and human GPR119 receptors, exhibiting EC50 values of 5.6 and 7.9 uM, respectively. 了解更多
  6. AM-1638
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    AM-1638

    Catalog No. A21505
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    GPR40/FFA1 full agonist
    AM-1638 is a potent and orally bioavailable GPR40/FFA1 full agonist with an EC50 of 0.16 μM. 了解更多
  7. AF64394
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    AF64394

    Catalog No. A21574
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    GPR3 inverse agonist
    AF64394 is a GPR3 inverse agonist, with a pIC50 of 7.3. 了解更多
  8. (1R,2R)-2-PCCA(hydrochloride)
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    (1R,2R)-2-PCCA(hydrochloride)

    Catalog No. A21655
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    GPR88 receptor agonist
    (1R,2R)-2-PCCA hydrochloride is a diastereomer of 2-PCCA, and acts as a potent GPR88 receptor agonist, with an EC50 of 3 nM in cell-free assay, and 603 nM in cell assay. 了解更多
  9. AM-4668
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    AM-4668

    Catalog No. A21778
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    GPR40 agonist
    AM-4668 is a GPR40 agonist for type 2 diabetes. EC50s of 3.6 nM and 36 nM for GPR40 in A9 cells (GPR40 IP3 assay) and CHO cells (GPR40 aequorin assay), respectively. 了解更多
  10. AMG 837 sodium salt
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    AMG 837 sodium salt

    Catalog No. A21793
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    GPR40 agonist
    AMG 837 sodium salt is a potent GPR40 agonist(EC50=13 nM) with a superior pharmacokinetic profile and robust glucose-dependent stimulation of insulin secretion in rodents. 了解更多
  11. MK-0354
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    MK-0354

    Catalog No. A22008
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    GPR109a receptor agonist
    MK-0354 is a partial agonist of GPR109a receptor, for hGPR109a/ mGPR109a with EC50 of 1.65/1.08 μM, showed no activation of GPR109b. 了解更多
  12. AMG 837
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    AMG 837

    Catalog No. A21160
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    GPR40 agonist
    AMG 837 is a potent GPR40 agonist(EC50=13 nM) with a superior pharmacokinetic profile and robust glucose-dependent stimulation of insulin secretion in rodents. 了解更多
  13. MK-6892
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    MK-6892

    Catalog No. A12982
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    GPR109A 激动剂
    MK-6892是高亲和力烟酸（NA）受体GPR109A的有效，选择性和完全激动剂。人GPR109A的MK-6892的Ki和GTPγSEC 50分别为4 nM和16 nM。 了解更多
  14. TM N1324
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    TM N1324

    Catalog No. A17038
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    GPR39 激动剂
    TM N1324是G蛋白偶联受体39（GPR39）的激动剂，在Zn2+存在下的EC50为9 nM/5 nM，而对于人/鼠GPR39，则在Zn2+不存在时的EC50为280 nM/180 nM。 了解更多
  15. RO462005
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    RO462005

    Catalog No. A13216
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    endothelin receptor 激动剂
    RO462005是内皮素受体选择性激动剂。 了解更多
  16. Radioprotectin-1
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    Radioprotectin-1

    Catalog No. A18628
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    LPA2 agonist
    Radioprotectin-1 is a potent and specific nonlipid agonist of lysophosphatidic acid receptor 2 (LPA2), with an EC50 value of 25 nM for murine LPA2 subtype. 了解更多
  17. GRI 977143
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    GRI 977143

    Catalog No. A15343
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    LPA2 激动剂
    GRI 977143是选择性溶血磷脂酸2（LPA2）受体非脂质激动剂（EC50 = 3.3 uM）。 了解更多
  18. GSK726701A
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    GSK726701A

    Catalog No. A20101
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    EP4 partial agonist
    GSK726701A is a novel prostaglandin E2 receptor 4 (EP4) partial agonist with a pEC50 of 7.4. 了解更多
  19. AGN 210676
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    AGN 210676

    Catalog No. A21281
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    prostaglandin EP2 agonist
    AGN 210676 is a selective prostaglandin EP2 agonist extracted from patent US20070203222A1, Compound example 23, has an EC50 of 5 nM. 了解更多
  20. Treprostinil sodium
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    Treprostinil sodium

    Catalog No. A21046
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    DP1/EP2 agonist
    Treprostinil sodium is a potent DP1 and EP2 agonist with EC50 values of 0.6??0.1 and 6.2??1.2 nM, respectively. 了解更多
  21. NS-304 (Selexipag)
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    NS-304 (Selexipag)

    Catalog No. A13880
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    prostacyclin receptor 激动剂
    NS-304 (Selexipag)是一种选择性的前列环素IP1受体激动剂（人和大鼠IP受体的Ki值为260和2100 nM，EP1-4，DP，FP和TP受体的Ki值为> 10μM）。 了解更多
  22. CP544326 (Taprenepag)
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    CP544326 (Taprenepag)

    Catalog No. A15853
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    EP2 激动剂?
    CP544326 (Taprenepag)是一种有效的选择性前列腺素E2受体激动剂，EC50值为2.8 nM。 了解更多
  23. KAG-308
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    KAG-308

    Catalog No. A18389
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    EP4 激动剂
    KAG-308, a newly-identified EP4-selective agonist shows efficacy for treating ulcerative colitis and can bring about lower risk of colorectal carcinogenesis by oral administration. 了解更多
  24. AB-MECA
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    AB-MECA

    Catalog No. A12189
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    A3 adenosine receptor agonist
    AB-MECA is a high affinity A3 adenosine receptor agonist, has high affinity for recombinant A1 and A3 receptors. 了解更多
  25. CGS 21680
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    CGS 21680

    Catalog No. A11354
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    adenosine A2A receptor agonist
    CGS 21680 is a selective adenosine A2A receptor agonist, with a Ki of 27 nM. 了解更多
  26. APNEA
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    APNEA

    Catalog No. A20845
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    A3 adenosine receptor agonist
    APNEA (N6-[2-(4-Aminophenyl)ethyl]adenosine) is a potent, non-selective A3 adenosine receptor agonist. 了解更多
  27. N6-Cyclohexyladenosine
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    N6-Cyclohexyladenosine

    Catalog No. A21008
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    A1 receptor agonist
    N6-Cyclohexyladenosine is a selective A1 receptor agonist (EC50 = 8.2 nM). 了解更多
  28. CGS 21680 HCl Hydrate
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    CGS 21680 HCl Hydrate

    Catalog No. A11619
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    Adenosine A2A Receptor 激动剂
    CGS 21680 HCl是一种特定的腺苷A2A亚型受体激动剂。 了解更多
  29. Capadenoson
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    Capadenoson

    Catalog No. A14159
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    Adenosine Receptor 激动剂
    Capadenoson是腺苷A1受体的选择性激动剂。 了解更多
  30. IB-MECA
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    IB-MECA

    Catalog No. A14345
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    Adenosine A3-R 激动剂
    IB-MECA已被证明是一种有效的选择性腺苷A3-R激动剂，腺苷A3-R，腺苷A1-R和腺苷A2A-R的Ki值分别为1.1、54和56 nM。 了解更多
  31. 2-Chloroadenosine (CADO)
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    2-Chloroadenosine (CADO)

    Catalog No. A16105
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    Adenosine A Receptor 激动剂
    2-Chloroadenosine (CADO)是腺苷的代谢稳定的类似物，其表现为腺苷A受体激动剂（腺苷A1-R，腺苷A2A-R和腺苷A3-R的Ki值分别为300、80和1900 nM）。 了解更多
  32. CGS 21680 HCl
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    CGS 21680 HCl

    Catalog No. A16441
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    Adenosine A2 receptor 激动剂
    CGS 21680 HCl是腺苷A2受体激动剂，IC50为22 nM，比A1受体高140倍。 了解更多
  33. Regadenoson
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    Regadenoson

    Catalog No. A12541
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    A2A adenosine 激动剂
    Regadenoson是A2A腺苷受体相对于A1，A2B和A3受体的选择性激动剂。还发现Regadenoson是引起冠状动脉血管扩张的完全而有效的激动剂，这种反应具有非常大的A2A受体储备。 了解更多
  34. NECA
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    NECA

    Catalog No. A16962
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    adenosine receptor 激动剂
    NECA是一种高亲和力的腺苷受体激动剂（human A3，A1和A2A受体的Ki值分别为6.2、14和20 nM；human A2B的EC50 = 2.4 μM）。 了解更多
  35. MRS1706
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    MRS1706

    Catalog No. A16868
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    adenosine A2B receptor 反向激动剂
    MRS1706是一种选择性腺苷A2B受体反向激动剂，对人A2B，A1，A2A和A3受体的Ki值分别为1.39、157、112和230 nM。 了解更多
  36. Tecadenoson
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    Tecadenoson

    Catalog No. A13302
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    A1 adenosine receptor agonist
    Tecadenoson (CVT-510) is a selective A1 adenosine receptor agonist. 了解更多
  37. SR 144528
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    SR 144528

    Catalog No. A12376
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    CB2 inverse 激动剂
    SR 144528是一种选择性的外周大麻素受体反向激动剂，对大鼠脾脏和人重组CB2受体的Ki值为0.6 nM，对大鼠脑和人重组CB1受体的Ki值为400 nM。 了解更多
  38. VCE-004.8
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    VCE-004.8

    Catalog No. A18549
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    PPARγ and CB2 receptor dual agonist
    VCE-004.8, a semi-synthetic multitarget cannabinoquinoid, is a specific PPARγ and CB2 receptor dual agonist with potent anti-inflammatory activity. 了解更多
  39. CB2R-IN-1
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    CB2R-IN-1

    Catalog No. A12306
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    cannabinoid CB2 receptor inverse agonist
    CB2R-IN-1 is a potent cannabinoid CB2 receptor inverse agonist with a Ki of 0.9 nM. 了解更多
  40. Taranabant
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    Taranabant

    Catalog No. A11578
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    CB1 receptor inverse agonist
    Taranabant is a highly potent and selective cannabinoid 1 (CB1) receptor inverse agonist that inhibits the binding and functional activity of various agonists, with a binding Ki of 0.13 nM for the human CB1R in vitro. 了解更多
  41. Taranabant ((1R,2R)stereoisomer)
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    Taranabant ((1R,2R)stereoisomer)

    Catalog No. A21705
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    CB1 receptor inverse agonist
    Taranabant (1R,2R)stereoisomer is the R-enantiomer of Taranabant. Taranabant is a highly potent and selective cannabinoid 1 (CB1) receptor inverse agonist. 了解更多
  42. WIN 55,212-2 mesylate
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    WIN 55,212-2 mesylate

    Catalog No. A11932
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    CB receptor 激动剂
    WIN 55,212-2 mesylate是一种有效的cannabinoid receptor激动剂，在神经性疼痛的大鼠模型中具有有效的镇痛作用。它通过受体介导的信号激活p42和p44 MAP激酶。 了解更多
  43. MDA 19
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    MDA 19

    Catalog No. A11939
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    CB2 激动剂
    MDA 19是CB2的有效选择性激动剂，对精神活性CB1受体具有合理的选择性。 了解更多
  44. GW842166X
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    GW842166X

    Catalog No. A11253
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    CB2 receptor 激动剂
    GW842166X是一种选择性的非大麻类CB2受体激动剂，EC50为63 nM，对CB1受体没有显著的活性。 了解更多
  45. Tedalinab
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    Tedalinab

    Catalog No. A14189
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    CB2 receptor 激动剂
    Tedalinab (GRC-10693)是开发用于治疗骨关节炎和神经性疼痛的药物，它可作为有效的选择性大麻素CB2受体激动剂。与相关的CB1受体相比，它对CB2的选择性为4700x，具有很高的口服生物利用度，并在早期临床试验中显示出令人鼓舞的安全性结果以及有效的镇痛和抗炎作用。 了解更多
  46. Bay 59-3074
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    Bay 59-3074

    Catalog No. A16328
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    CB1/CB2 receptor 激动剂
    Bay 59-3074是一种新型的选择性CB1/CB2受体部分激动剂，对人CB1和CB2受体的Ki值分别为48.3和45.5 nM。 了解更多
  47. AM1241
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    AM1241

    Catalog No. A16397
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    CB2 receptor 激动剂
    AM1241是选择性的大麻素CB2受体激动剂，Ki为3.4 nM，相对于CB1受体具有82倍的选择性。 了解更多
  48. Rimonabant hydrochloride
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    Rimonabant hydrochloride

    Catalog No. A11548
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    CB1 receptor inverse 激动剂
    Rimonabant hydrochloride是CB1受体反向激动剂。 了解更多
  49. ML314
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    ML314

    Catalog No. A13570
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    NTR1 激动剂
    ML-314是神经降压素NTR1受体的脑渗透性非肽β-arrestin偏向性激动剂，在主要试验中对NTR1（EC50 = 2.0μM）表现出完全的激动剂行为，对NTR2具有选择性。 了解更多
  50. Orexin 2 Receptor Agonist
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    Orexin 2 Receptor Agonist

    Catalog No. A15982
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    Orexin 2 receptor 激动剂
    Orexin 2 Receptor Agonist一种有效的选择性Orexin2受体激动剂。 了解更多

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