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CGS-15943
Catalog No. A14327 -
Preladenant
Catalog No. A13504 -
DPCPX
Catalog No. A16104 -
2-Chloroadenosine (CADO)
Catalog No. A16105 Adenosine A Receptor 激动剂2-Chloroadenosine (CADO)是腺苷的代谢稳定的类似物，其表现为腺苷A受体激动剂（腺苷A1-R，腺苷A2A-R和腺苷A3-R的Ki值分别为300、80和1900 nM）。 了解更多 -
CGS 21680 HCl
Catalog No. A16441 -
Regadenoson
Catalog No. A12541 A2A adenosine 激动剂Regadenoson是A2A腺苷受体相对于A1，A2B和A3受体的选择性激动剂。还发现Regadenoson是引起冠状动脉血管扩张的完全而有效的激动剂，这种反应具有非常大的A2A受体储备。 了解更多 -
Vipadenant (BIIB-014)
Catalog No. A13963 A2A receptor 拮抗剂Vipadenant，也称为BIIB014，CEB-4520，是针对帕金森氏症的有效，选择性和口服腺苷A2A受体拮抗剂。Vipadenant在帕金森氏病的常用模型中显示出强大的口服活性。 了解更多 -
Theophylline-7-acetic acid
Catalog No. A16822 -
Proxyphylline
Catalog No. A16821 A1 adenosine receptors 拮抗剂Proxyphylline是茶碱的衍生物，由于其心血管特性而被用作支气管扩张剂。它与A2腺苷受体（对于血小板，Ki = 850μM）选择性拮抗A1腺苷受体（对于牛脑，Ki = 82 nM）。 了解更多 -
AZD-4635 (HTL1071)
Catalog No. A16820 -
MRS1177
Catalog No. A16871 -
MRS1186
Catalog No. A16870 -
Tecadenoson
Catalog No. A13302 A1 adenosine receptor agonistTecadenoson (CVT-510) is a selective A1 adenosine receptor agonist. 了解更多 -
MT-DADMe-ImmA
Catalog No. A13651 human 5'-methylthioadenosine phosphorylase inhibitorMT-DADMe-ImmA is an inhibitor of human 5'-methylthioadenosine phosphorylase (MTAP) with a Ki of 90 pM. 了解更多 -
A2A receptor antagonist 1
Catalog No. A12567 adenosine A2A/A1 receptor antagonistA2A receptor antagonist 1 (CPI-444 analog) is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively. 了解更多 -
Tonapofylline
Catalog No. A21328 adenosine A1 receptor antagonistTonapofylline (BG 9928) is an orally active and selective adenosine A1 receptor antagonist with a Ki of 7.4 nM for human adenosine A1 receptor (hA1), which displays 915-fold selectivity versus human adenosine A2A receptor and 12-fold selectivity versus human adenosine A2B receptor and is used in development for the treatment of heart failure. 了解更多 -
EHNA hydrochloride
Catalog No. A21585 Adenosine deaminase inhibitorEHNA hydrochloride is a specific inhibitor of adenosine deaminase, prevents dAdo degradation and increases mitochondrial dATP levels in fibroblasts. 了解更多 -
Rolofylline
Catalog No. A21649 adenosine A1 receptor antagonistRolofylline (KW-3902) is a potent, selective adenosine A1 receptor antagonist that is under development for the treatment of patients with acute congestive heart failure and renal impairment. 了解更多 -
Derenofylline
Catalog No. A21990 adenosine A1 receptor antagonistDerenofylline (SLV 320) is a potent, selective and orally active adenosine A1 receptor antagonist, with Ki values of 1 nM, 200 nM and 398 nM for human A1, A3 and A2A receptors respectively. 了解更多 -
N6-Cyclohexyladenosine
Catalog No. A21008 A1 receptor agonistN6-Cyclohexyladenosine is a selective A1 receptor agonist (EC50 = 8.2 nM). 了解更多 -
Laropiprant (MK0524)
Catalog No. A11483 DP1 抑制剂Laropiprant (MK0524)与烟酸合用可降低血液胆固醇。是一种有效的，选择性的 DP receptor 拮抗剂，Ki 值为 0.57 nM，对 TP 受体的 Ki 值为 2.95 nM。 了解更多 -
Ozagrel hydrochloride
Catalog No. A11742 Thromboxane A2 synthesis 抑制剂Ozagrel hydrochloride是一种抗血小板剂，用作血栓烷a2合成抑制剂。 了解更多 -
Cloprostenol (sodium salt)
Catalog No. A13498 cloprostenol是前列腺素F2α（PGF2α）的合成类似物。它在仓鼠和大鼠中终止妊娠的效力分别是PGF2α的200倍和100倍，而没有与PGF2α相关的副作用。 了解更多 -
BAY-u 3405
Catalog No. A13751 -
NS-304 (Selexipag)
Catalog No. A13880 prostacyclin receptor 激动剂NS-304 (Selexipag)是一种选择性的前列环素IP1受体激动剂（人和大鼠IP受体的Ki值为260和2100 nM，EP1-4，DP，FP和TP受体的Ki值为> 10μM）。 了解更多 -
MF498
Catalog No. A15532 -
PF-04418948
Catalog No. A12894 -
CP544326 (Taprenepag)
Catalog No. A15853 -
TG6-10-1
Catalog No. A15968 -
Grapiprant (CJ-023423)
Catalog No. A15964 prostaglandin EP4 receptor 拮抗剂Grapiprant (CJ-023423)是一种具有抗痛觉过敏特性的新型，有效且选择性的前列腺素EP4受体拮抗剂。 了解更多
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