“glucagon receptor”的搜索结果

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  1. Vortioxetine (Lu AA21004) hydrobromide

    Catalog No. A12602
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    5-HT Receptor modulator
    Vortioxetine (Lu AA21004) hydrobromide是一种口服多峰血清素能药物,可抑制5-HT(1A),5-HT(1B),5-HT(3A),5-HT(7)和SERT,IC50为15 nM,33 nM,3.7 nM,19 nM和1.6 nM。 了解更多
  2. PU 02

    Catalog No. A13757
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    5-HT3 Receptor Modulator
    PU 02是5-HT3受体的负变构调节剂。 了解更多
  3. CBiPES HCl

    Catalog No. A15811
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    mGlu2 receptor modulator
    CBiPES HCl是mGluR-2的选择性正变构调节剂,IC50值为98.2 nM。 了解更多
  4. Ponesimod

    Catalog No. A13307
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    S1P1 receptor modulator
    Ponesimod是一种口服活性,选择性鞘氨醇-1-磷酸受体1(S1P1)免疫调节剂,EC50为5.7 nM。 了解更多
  5. NSC-23026

    Catalog No. A17151
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    CXCR4 receptor modulator
    NSC-23026是CXCR4受体调节剂。 了解更多
  6. VU0652835

    Catalog No. A18885
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    mGlu5 modulator
    VU0652835 is a metabotropic glutamate receptor subtype 5 (mGlu5) negative allosteric modulator with an IC50 of 81 nM. 了解更多
  7. Lu AF21934

    Catalog No. A12140
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    mGlu4 receptor modulator
    Lu AF21934 is a selective and brain-penetrant mGlu4 receptor positive allosteric modulator with an IC50 of 500 nM for human mGlu4. 了解更多
  8. Endothelin Mordulator 1

    Catalog No. A13040
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    endothelin receptor modulator
    Endothelin Mordulator 1 is a endothelin receptor modulator, used for the research of endothelin-mediated disorders. 了解更多
  9. TCN238

    Catalog No. A21191
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    mGlu4 receptor modulator
    TCN238 is a positive allosteric mGlu4 receptor modulator with an EC50 of 1 μM. 了解更多
  10. LUF6000

    Catalog No. A21532
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    A3 adenosine receptor allosteric modulator
    LUF6000 is an allosteric modulator of the human A3 adenosine receptor (AR). 了解更多
  11. VU 0361737

    Catalog No. A12467
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    mGlu4 receptors modulator
    VU 0361737是mGluR-4的选择性正变构调节剂(人和大鼠受体的EC50值分别为240和110 nM)。 了解更多
  12. VU 0364770

    Catalog No. A12139
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    mGlu4 receptors modulator
    VU 0364770是mGlu4受体的正变构调节剂,在表达mGlu4的HEK 293细胞中EC50值为290 nM。 了解更多
  13. E1R

    Catalog No. A18825
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    sigma-1 receptors modulator
    E1R is a novel positive allosteric modulator of sigma-1 receptors. 了解更多
  14. VU0453379

    Catalog No. A18796
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    GLP-1R modulator
    VU0453379 is a CNS-penetrant glucagon-like peptide 1 receptor (GLP-1R) positive allosteric modulator (PAM) with an EC50 of 1.3 μM. 了解更多
  15. NNC0640

    Catalog No. A18900
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    GLP-1R modulator
    NNC0640 is a negative allosteric modulator of glucagon-like peptide-1 receptor (GLP-1R). 了解更多

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