“jwh 307”的搜索结果

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  1. PD173074

    Catalog No. A10703
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    FGFR1/VEGFR2 抑制剂
    PD173074是有效的,细胞可渗透的和ATP竞争性的FGFR和VEGFR抑制剂。 了解更多
  2. SL 0101-1

    Catalog No. A11160
    RSK 抑制剂
    SL 0101-1是p90核糖体S6激酶(RSK)的选择性抑制剂(对于RSK2,IC50 = 89 nM)。 了解更多
  3. Diclofenac sodium

    Catalog No. A10304
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    COX 抑制剂
    Diclofenac Sodium是一种非选择性的COX抑制剂,完整细胞中的COX-1和-2的IC50分别为0.5μg/ml和0.5μg/ml,作用于绵羊COX-1和COX-2, IC50分别为60和220 nM,用作非甾体类抗炎药(NSAID)来减轻疼痛和减轻疼痛 肿胀发炎。 了解更多
  4. Avanafil

    Catalog No. A12619
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    PDE5 抑制剂
    Avanafil是用于治疗勃起功能障碍的PDE5抑制剂,IC50为5.2 nM,对PDE1,PDE6和PDE11活性较低。 了解更多
  5. NSC 405020

    Catalog No. A13072
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    MT1-MMP 抑制剂
    NSC-405020是一种膜1型基质金属蛋白酶(MT1-MMP)抑制剂(IC50> 100μmol/ L)。 了解更多
  6. Donepezil

    Catalog No. A13079
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    AChE 抑制剂
    Donepezil是一种非竞争性乙酰胆碱酯酶抑制剂,可以很容易地穿过血脑屏障并增加皮质乙酰胆碱的浓度。众所周知,多奈哌齐是研究阿尔茨海默病的有用工具。 了解更多
  7. PSI-7977

    Catalog No. A11529
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    HCV Nucleotide 抑制剂
    PSI-7977是PSI-7851的氨基磷酸酯前药,PSI-7851是核苷类似物,当磷酸化时,抑制丙型肝炎病毒的RNA依赖性RNA聚合酶(EC50 = 92 nM)。 了解更多
  8. Y-33075

    Catalog No. A11610
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    ROCK 抑制剂
    Y-33075是ROCK(Rho相关的卷曲螺旋形成蛋白激酶)抑制剂。 了解更多
  9. NH125

    Catalog No. A14307
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    eEF-2 抑制剂
    NH125是选择性eEF-2激酶抑制剂。 了解更多
  10. CFTRinh-172

    Catalog No. A12897
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    CFTR 抑制剂
    CFTRinh-172是电压无关的选择性CFTR抑制剂。在2分钟内可逆地抑制CFTR短路电流的 Ki 值为300 nM。 了解更多
  11. CL-82198

    Catalog No. A13597
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    MMP-13 抑制剂
    CL-82198是人胶原酶3(也称为基质金属蛋白酶13(MMP-13))的选择性抑制剂,在10 mg/ml时产生89%的抑制作用。 了解更多
  12. PD 166793

    Catalog No. A15307
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    Broad spectrum MMP 抑制剂
    PD166793是一种细胞可渗透的化合物,可强烈抑制MMP(基质金属蛋白酶)-2,-3和-13,而弱抑制AMP脱氨酶,MMP-1,-7,-9和-14。 了解更多
  13. WAY 170523

    Catalog No. A15317
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    MMP-13 抑制剂
    WAY 170523是MMP-13的选择性强效抑制剂。 了解更多
  14. CC-223

    Catalog No. A13078
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    mTOR 抑制剂
    CC-223是一种有效的mTOR激酶抑制剂(IC50 = 16 nM),其敏感性是相关脂质激酶PI3K-alpha(IC50 = 4 uM)的> 150倍。 了解更多
  15. MRT68921

    Catalog No. A15880
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    Autophagy ULK1/2 抑制剂
    MRT68921是一种有效的双重自噬激酶ULK1/2抑制剂,IC50分别为2.9 nM和1.1 nM。 了解更多
  16. MRT67307

    Catalog No. A11485
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    SIK/TBK-1/IKKe 抑制剂
    MRT67307是一种强效双IKK?和TBK1抑制剂,IC50分别为160和19 nM。 了解更多
  17. Rebeprazole sodium

    Catalog No. A16147
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    proton pump 抑制剂
    Rebeprazole sodium是质子泵抑制剂中的一种抗溃疡药。 了解更多
  18. PCI 29732

    Catalog No. A16262
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    BTK 抑制剂
    PCI 29732是一种选择性且不可逆的Btk抑制剂,在基于FRET的生化酶检测中,IC50为8.2 nM。 了解更多
  19. TC-E 5002

    Catalog No. A16373
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    KDM2/7 抑制剂
    TC-E 5002是一种选择性组蛋白脱甲基酶KDM2/7亚家族抑制剂(KDM7A,KDM7B,KDM2A,KDM5A,KDM4C,KDM6A和KDM4A的IC50值分别为0.2、1.2、6.8、55、83,> 100和> 120 uM)。在体外抑制HeLa和KYSE-150癌细胞的生长。 了解更多
  20. GRL0617

    Catalog No. A18780
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    SARS PLPro inhibitor
    GRL0617 is a potent, selective and competitive noncovalent inhibitor of SARS PLPro, with an IC50 of 0.6 μM, and with a Ki of 0.49 μM. 了解更多
  21. ODM-203

    Catalog No. A19098
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    FGFR/VEGFR 抑制剂
    ODM-203 is a potent FGFR and VEGFR families inhibitor with IC50s of 11, 16, 6, 35 nM towards recombinant FGFR1, FGFR2, FGFR3 and FGFR4 as well as 26, 9, 5 nM towards VEGFR1, VEGFR2 and VEGFR3, respectively. 了解更多
  22. Enzaplatovir

    Catalog No. A20830
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    RSV fusion protein inhibitor
    Enzaplatovir is an inhibitor of Respiratory Syncytial Virus (RSV). It can be used as a viral fusion protein inhibitor. 了解更多
  23. STF-083010

    Catalog No. A16720
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    IRE1α inhibitor
    STF-083010 is a specific IRE1α inhibitor. STF-083010 inhibits Ire1 endonuclease activity, without affecting its kinase activity, after endoplasmic reticulum stress. 了解更多
  24. BAY885

    Catalog No. A13765
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    ERK5 inhibitor
    BAY885 is a novel ERK5 inhibitor. 了解更多
  25. GSK2593074A

    Catalog No. A13600
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    necroptosis inhibitor
    GSK2593074A (GSK??074) is a necroptosis inhibitor with dual targeting ability to both RIP1 and RIP3. 了解更多
  26. NMDI14

    Catalog No. A12958
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    NMD inhibitor
    NMDI14 is a nonsense mediated RNA decay (NMD) inhibitor. 了解更多
  27. Y-33075 dihydrochloride

    Catalog No. A11611
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    ROCK inhibitor
    Y-33075 dihydrochloride is a selective ROCK inhibitor with an IC50 of 3.6 nM. 了解更多
  28. Diclofenac

    Catalog No. A17814
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    COX inhibitor
    Diclofenac is a potent and nonselective anti-inflammatory agent, acts as a COX inhibitor, with IC50s of 4 nM, 1.3 nM for human COX-1 and COX-2 in CHO cells, and 5.1, 0.84 μM for ovine COX-1 and COX-2, respectively. 了解更多
  29. Emiglitate

    Catalog No. A20917
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    α-glucoside hydrolase inhibitor
    Emiglitate (BAY o 1248) is a potent, selective and competitive inhibitor of α-glucoside hydrolase. 了解更多
  30. (R)-Simurosertib

    Catalog No. A21894
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    CDC7 kinase inhibitor
    (R)-Simurosertib ((R)-TAK-931) is the (R)-enantiomer of Simurosertib, Simurosertib (TAK-931) is a selective cycle 7 (CDC7) kinase inhibitor, with an IC50<0.3 nM. 了解更多
  31. PLpro inhibitor

    Catalog No. A21044
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    Plpro inhibitor
    PLpro inhibitor is a potent inhibitor of papain-like protease (PLpro) with IC50 of 2.6 uM. 了解更多
  32. Flumatinib

    Catalog No. A16258
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    multi-kinase 抑制剂
    Flumatinib是一种多激酶抑制剂,对c-Abl,PDGFRbeta和c-Kit的IC50值分别为1.2 nM,307.6 nM和2662 nM。 了解更多

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