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Tianeptine sodium
Catalog No. A10931 -
Tropisetron (ICS 205930)
Catalog No. A11226 -
WIN 55,212-2 mesylate
Catalog No. A11932 CB receptor 激动剂WIN 55,212-2 mesylate是一种有效的cannabinoid receptor激动剂，在神经性疼痛的大鼠模型中具有有效的镇痛作用。它通过受体介导的信号激活p42和p44 MAP激酶。 了解更多 -
CP 945598 HCl (Otenabant HCl)
Catalog No. A11942 -
Dopamine hydrochloride
Catalog No. A10331 Dopamine hydrochloride (abbreviated as DA)是儿茶酚胺家族中的一种简单的有机化学物质，是一种单胺类神经递质，一种由神经细胞释放以向其他神经细胞发送信号的化学物质。 了解更多 -
Rimonabant (SR141716)
Catalog No. A11547 Rimonabant是CB1的选择性拮抗剂，在hCB1转染的HEK 293膜中的IC50为13.6 nM，EC50为17.3 nM。 了解更多 -
Aripiprazole (Abilify)
Catalog No. A11801 5-HT1A receptor 激动剂Aripiprazole (Abilify)是人5-HT1A受体部分激动剂，Ki为4.2 nM。 了解更多 -
Ivabradine HCl (Procoralan)
Catalog No. A11868 Ivabradine Hydrochloride,也称为S-16257，是缓动剂伊伐布雷定的盐酸盐制剂。 了解更多 -
Mirabegron
Catalog No. A12861 β3 adrenergic receptor activatorMirabegron是一种选择性的beta3-adrenoceptor（β3肾上腺素受体）激动剂，EC50为22.4 nM。是有效的膀胱松弛药和糖尿病药物。 了解更多 -
AM 2201
Catalog No. A14174 -
Labetalol HCl
Catalog No. A14239 alpha1/beta adrenergic receptors 拮抗剂Labetalol HCl是选择性α1-肾上腺素能受体和非选择性β-肾上腺素能受体的双重拮抗剂。 了解更多 -
Tropisetron HCL
Catalog No. A14375 5-HT3 receptor 拮抗剂Tropisetron HCL是选择性的5-HT3受体拮抗剂和α7烟碱样受体激动剂，对5-HT3受体的IC50为70.1±0.9 nM。 了解更多 -
Atrasentan
Catalog No. A13779 ETA 拮抗剂Atrasentan是一种实验药物，正在研究中，用于治疗各种类型的癌症，包括非小细胞肺癌。它是对A型亚型（ETA）有选择性的内皮素受体拮抗剂,对ETA的IC50为0.0551 nM。 了解更多 -
Guanabenz acetate
Catalog No. A13635 -
HOKU-81
Catalog No. A15117 -
Otenabant
Catalog No. A15200 -
Atrasentan HCl
Catalog No. A15007 Endothelin 拮抗剂 receptorAtrasentan hydrochloride是一种开发用于治疗前列腺癌的内皮素拮抗剂受体（IC50 = 0.0551 nM，ETA）。 了解更多 -
ACR 16 hydrochloride
Catalog No. A16074 dopaminergic stabilizerACR 16 hydrochloride是一种多巴胺能稳定剂（对于D2（低）和D2（高），Ki值分别为17550 nM和7521），通过功能性多巴胺D2受体拮抗作用和皮质谷氨酸功能的双重作用，稳定地稳定精神运动活动。在各种情况下神经传递受到干扰。 了解更多 -
Rimonabant hydrochloride
Catalog No. A11548 -
Dinoprost tromethamine
Catalog No. A17505 Prostaglandin Receptor inhibitorDinoprost Tromethamine, also known as Dinoprost Trometamol, is a naturally occurring prostaglandin used in medicine to induce labor and as an abortifacient. 了解更多 -
Hydroxyzine pamoate
Catalog No. A17712 Histamine H1 receptor antagonistHydroxyzine pamoate is an histamine H1 receptor antagonist that is effective in the treatment of chronic urticaria, dermatitis, and histamine-mediated pruritus. Unlike its major metabolite CETIRIZINE, it does cause drowsiness. 了解更多 -
Trimebutine maleate
Catalog No. A18115 ?- opioid receptor agonistTrimebutine Maleate is a drug with antimuscarinic and weak mu opioid agonist effects. Trimebutine Maleate modulates the calcium and potassium channels, relieves abdominal pain in patients with irritable bowel syndrome. 了解更多 -
Kynurenic acid
Catalog No. A16581 GPR35/CXCR8 拮抗剂Kynurenic acid, an endogenous tryptophan metabolite, is a broad-spectrum antagonist targeting NMDA, glutamate, α7 nicotinic acetylcholine receptor. Kynurenic acid is also an agonist of GPR35/CXCR8. 了解更多 -
Alosetron (Hydrochloride(1:X))
Catalog No. A11309 Serotonin 5HT3-receptor antagonistAlosetron Hydrochloride(1:X) (GR 68755 Hydrochloride(1:X)) is a Serotonin 5HT3-receptor antagonist that is used in treatment of irritable bowel syndrome. 了解更多 -
Semaglutide
Catalog No. A18908 GLP-1 receptor agonistSemaglutide, a long-acting GLP-1 analogue, is a glucagon-like peptide-1 (GLP-1) receptor agonist that can be used in the treatment of type 2 diabetes. 了解更多 -
CB1 antagonist 2
Catalog No. A18810 CB1 antagonistCB1 antagonist 2 is caimabinoid 1 (CB1) antagonist extracted from patent WO2016184310A1, compound 3, inhibits CB1 in vivo with an IC50 of 25.5 nM. 了解更多 -
GPR35 agonist 1
Catalog No. A12462 GPR35/CXCR8 agonistGPR35 agonist 1 (compound 50) is a potent and specific G protein-coupled receptor-35 (GPR35)/CXCR8 agonist with an EC50 of 5.8 nM, displays good druggability. 了解更多 -
β3-AR agonist 1
Catalog No. A12777 β3-adrenergic receptor agonistβ3-AR agonist 1 (compound 15) is a highly potent, selective, and orally available β3-adrenergic receptor (β3-AR) agonist (EC50=18 nM), being inactive to β1-, β2-, and α1A-AR (β1/β3, β2/β3, and α1A/β3>556-fold). 了解更多 -
Kynurenic acid sodium
Catalog No. A20000 GPR35/CXCR8 agonistKynurenic acid sodium, an endogenous tryptophan metabolite, is a broad-spectrum antagonist targeting NMDA, glutamate, α7 nicotinic acetylcholine receptor. Kynurenic acid sodium is also an agonist of GPR35/CXCR8. 了解更多 -
Taranabant
Catalog No. A11578 CB1 receptor inverse agonistTaranabant is a highly potent and selective cannabinoid 1 (CB1) receptor inverse agonist that inhibits the binding and functional activity of various agonists, with a binding Ki of 0.13 nM for the human CB1R in vitro. 了解更多 -
Cutamesine
Catalog No. A21152 sigma 1 receptor agonistCutamesine (SA4503; AGY-94806) is a selective sigma 1 receptor(??1R) agonist; high affinity for the sigma 1 receptor subtype labeled by (+)-[3H]pentazocine (IC50= 17.4??1.9 nM); 100-fold less affinity for the sigma 2 receptor. 了解更多 -
GPR40 Activator 1
Catalog No. A21154 GPR40 activatorGPR40 Activator 1 is a potent GPR40 activator for treatment of type 2 diabetes. 了解更多 -
L-371,257
Catalog No. A21219 oxytocin receptor antagonistL-371,257 is an orally bioavailable, non-blood-brain barrier penetrant, selective and competitive antagonist of oxytocin receptor (pA2=8.4) with high affinity at both the oxytocin receptor (Ki=19 nM) and vasopressin V1a receptor (Ki=3.7 nM). 了解更多
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