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42 个项目
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H4 Receptor antagonist 1
Catalog No. A18929 histamine H4 receptor inverse agonistH4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC50 of 19 nM. 了解更多 -
Toreforant
Catalog No. A21058 histamine H4 receptor (H4R) antagonistToreforant is a potent and selective histamine H4 receptor (H4R) antagonist, with a Ki at the human receptor of 8.4 nM. 了解更多 -
Decloxizine
Catalog No. A20964 histamine 1 receptor antagonistDecloxizine(UCB-1402; NSC289116) is a histamine 1 receptor antagonist. 了解更多 -
GSK189254A
Catalog No. A22005 histamine H3 receptor antagonistGSK189254A (GSK189254) is a novel, potent and selective histamine H3 receptor antagonist with pKi values of 9.59-9.90 and 8.51-9.17 for human and rat H3, respectively. 了解更多 -
Niperotidine
Catalog No. A21981 histamine H2-receptor antagonistNiperotidine is a histamine H2-receptor antagonist. 了解更多 -
JNJ-5207852
Catalog No. A21480 histamine H3 receptor antagonistJNJ-5207852 is a selective and potent histamine H3 receptor (H3R) antagonist, with pKis of 8.9, 9.24 for rat and human H3R, respectively. 了解更多 -
PF-03654746 Tosylate
Catalog No. A21434 histamine H3 receptor antagonistPF-03654746 Tosylate is a potent and selective histamine H3 receptor antagonist with high brain penetration. 了解更多 -
PF-03654746
Catalog No. A21429 histamine H3 receptor antagonistPF-03654746 is a potent and selective histamine H3 receptor antagonist with high brain penetration. 了解更多 -
Mebhydrolin napadisylate
Catalog No. A17997 -
Acrivastine
Catalog No. A17746 Histamine 1 receptor antagonistAcrivastine (BW825C) is a short acting histamine 1 receptor antagonist for the treatment of allergic rhinitis. 了解更多 -
Hydroxyzine pamoate
Catalog No. A17712 Histamine H1 receptor antagonistHydroxyzine pamoate is an histamine H1 receptor antagonist that is effective in the treatment of chronic urticaria, dermatitis, and histamine-mediated pruritus. Unlike its major metabolite CETIRIZINE, it does cause drowsiness. 了解更多 -
Levocetirizine Dihydrochloride
Catalog No. A17440 L-isomer of cetirizine and histamine H1 receptor antagonistLevocetirizine dihydrochloride is a L-isomer of cetirizine and histamine H1 receptor antagonist. It incrases levels of CD4+ CD25+ T cells and decreases levels of eosinophils, decreasing allergy symptoms. 了解更多 -
Terfenadine
Catalog No. A17373 H1 histamine receptor antagonistTerfenadine ((??)-Terfenadine) is a potent open-channel blocker of hERG with an IC50 of 204 nM. Terfenadine, an H1 histamine receptor antagonist, acts as a potent apoptosis inducer in melanoma cells through modulation of Ca2+ homeostasis. Terfenadine induces ROS-dependent apoptosis, simultaneously activates Caspase-4, -2, -9 and induces p73, Noxa. 了解更多 -
Fexofenadine HCl
Catalog No. A11859 COX 抑制剂/histamine H1 receptor 激动剂Fexofenadine Hydrochloride是一种抗组胺药，可抑制Cox-1，Cox-2，并且是组胺H1受体激动剂，IC50为246 nM。 了解更多 -
Mequitazine
Catalog No. A18206 Histamine H1 antagonistMequitazine is a potent histamine H1 antagonist or antihistamine. It competes with histamine for the normal H1-receptor sites on effector cells of the gastrointestinal tract, blood vessels and respiratory tract. 了解更多 -
Cyclizine 2HCl
Catalog No. A16472 -
Antazoline HCl
Catalog No. A16411 -
Alcaftadine
Catalog No. A16393 H1 histamine receptor 拮抗剂Alcaftadine是H1受体的高亲和力配体，其pKi（8.5）与其他H1抗组胺药相当。Alcaftadine还是H2和H4受体的拮抗剂，对H3受体没有亲和力。 了解更多 -
Lidocaine hydrochloride
Catalog No. A16132 -
CarbinoxaMine Maleate
Catalog No. A16129 histamine-H1 receptor blocking agentCarbinoxamine maleate是一种具有抗组胺和抗胆碱能特性的组胺-H1受体阻断剂。 了解更多 -
Bavisant dihydrochloride hydrate
Catalog No. A15016 -
Bavisant dihydrochloride
Catalog No. A15015 -
Ebrotidine
Catalog No. A15075 -
Clemizole hydrochloride
Catalog No. A15047 H1 histamine receptor 拮抗剂Clemizole hydrochloride是H1组胺受体的拮抗剂，对NS4B RNA结合的IC50值为8 mM。 了解更多 -
Cetirizine
Catalog No. A15041 -
A 943931 2HCl
Catalog No. A13442 -
Immethridine hydrobromide
Catalog No. A13641 histamine H3 receptor 激动剂Immethridine hydrobromide是一种强而高选择性的组胺H3受体激动剂（pEC50 = 9.74），其选择性是H4受体的300倍（pKi值分别为9.07和6.61）。 了解更多 -
Astemizole
Catalog No. A13899 H1-receptor 拮抗剂Astemizole是一种有效的抗组胺药物（H1-受体拮抗剂，IC50 = 4 nM），对多巴胺，5-HT和毒蕈碱乙酰胆碱受体具有选择性。该化合物显示出有效的hERG K+通道阻断活性（IC50 = 0.9 nM），在体外多药耐药菌株中具有抗疟疾活性（IC50 = 227-734 nM），并已被用作分子伴侣来纠正折叠缺陷并恢复蛋白质功能 hERG通道的某些突变形式。 了解更多 -
Promethazine HCl
Catalog No. A14248 -
Rupatadine
Catalog No. A11222 PAFR 抑制剂/H1 receptor 抑制剂Rupatadine是PAFR和组胺（H1）受体的抑制剂，Ki分别为550和102 nM。 了解更多 -
Rupatadine Fumarate
Catalog No. A12356 PAFR 抑制剂/H1 receptor 抑制剂Rupatadine Fumarate是PAFR和组胺(H1)受体的抑制剂，Ki分别为550和102 nM。 了解更多 -
Bepotastine Besilate
Catalog No. A11340 -
Orphenadrine citrate
Catalog No. A11712 -
Clemastine fumarate
Catalog No. A10226 Histamine Receptor antagonisClemastine fumarate是一种选择性的组胺H1拮抗剂。它与组胺H1受体结合，从而阻断了内源性组胺的作用，从而暂时缓解了由组胺引起的阴性症状。 了解更多 -
Ciproxifan maleate
Catalog No. A11117
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