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￥ 0.00 “kinase+inhibitor”的搜索结果
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AKT Kinase Inhibitor
Catalog No. A11285 Akt kinase inhibitorAKT Kinase Inhibitor is an Akt kinase inhibitor with anti-tumor activity. 了解更多 -
Multi-kinase inhibitor 1
Catalog No. A22645 multi-kinase inhibitorMulti-kinase inhibitor 1 is a potent multi-kinase inhibitor. Multi-kinase inhibitor 1 has the potential for diseases or disorders associated with abnormal or deregulated tyrosine kinase activity, particularly diseases associated with the activity of PDGF-R, c-Kit and Bcr-abl. 了解更多 -
Src Inhibitor 1
Catalog No. A12299 Src tyrosine kinase inhibitorSrc Inhibitor 1 is a potent and selective dual site Src tyrosine kinase inhibitor with IC50 values of 44 nM for Src and 88nM for Lck. 了解更多 -
RIP1 kinase inhibitor 1
Catalog No. A20154 RIP1 kinase inhibitorRIP1 kinase inhibitor 1 (compound 22) is a highly potent, orally available, and brain-penetrating RIP1 kinase inhibitor (pKi=9.04). 了解更多 -
PDGFRα kinase inhibitor 1
Catalog No. A19632 type II PDGFRα kinase inhibitorPDGFRα kinase inhibitor 1 is a highly selective type II PDGFRα kinase inhibitor with IC50s of 132 nM and 6115 nM for PDGFRα and PDGFRβ, respectively. 了解更多 -
Aurora Kinase Inhibitor 3
Catalog No. A19448 Aurora A kinase inhibitorAurora Kinase Inhibitor 3 is a strong and selective Aurora A kinase inhibitor with an IC50 of 42 nM, and weakly inhibits EGFR with an IC50>10 μM. 了解更多 -
Tie2 kinase inhibitor
Catalog No. A10932 -
IRAK inhibitor 2
Catalog No. A11456 interleukin-1 receptor associated kinase inhibitorIRAK inhibitor 2 is interleukin-1 receptor associated kinase inhibitor . 了解更多 -
RIP2 Kinase Inhibitor 3
Catalog No. A20109 RIP2 inhibitorRIP2 Kinase Inhibitor 3 is a highly potent and selective inhibitor of receptor interacting protein-2 (RIP2) Kinase with an IC50 of 1 nM . 了解更多 -
RIP2 kinase inhibitor 2
Catalog No. A16313 RIP2 kinase 抑制剂RIP2 kinase inhibitor 2 是从专利WO/2014043437 A1（化合物实施例9）中提取的受体相互作用蛋白2（RIP2）激酶抑制剂。 了解更多 -
RIP2 kinase inhibitor 1
Catalog No. A16312 RIP2 kinase 抑制剂RIP2 kinase inhibitor 1 是从专利WO/2014043446 A1（化合物实施例1）中提取的受体相互作用蛋白2（RIP2）激酶抑制剂。 了解更多 -
Ehp inhibitor 2
Catalog No. A22325 Eph family tyrosine kinase inhibitorEhp inhibitor 2 is a Eph family tyrosine kinase inhibitor. 了解更多 -
Raf inhibitor 2
Catalog No. A22641 raf kinase inhibitorRaf inhibitor 2 is a potent raf kinase (IC50<1.0 μM) inhibitor, compound 32, extracted from patent EP1003721B1. Raf inhibitor 2 can be used for cancer research. 了解更多 -
ROCK inhibitor
Catalog No. A15225 ROCK 抑制剂ROCK inhibitor是人类ROCK-1和ROCK-2同工酶的高效抑制剂，IC50值分别为0.6和1.1 nM。 了解更多 -
cGMP Dependent Kinase Inhibitor Peptid
Catalog No. A16052 PKG/PKA 抑制剂cGMP Dependent Kinase Inhibitor Peptid是一种特定的cGKI（环GMP依赖性蛋白激酶）抑制剂。数据表明，它不阻断完整组蛋白的环状GMP依赖性蛋白激酶磷酸化，已被用于研究恶性疟原虫。 了解更多 -
B-Raf inhibitor 1 dihydrochloride
Catalog No. A21834 Raf kinase inhibitorB-Raf inhibitor 1 dihydrochloride is a potent Raf kinase inhibitor with Kis of 1 nM, 1 nM, and 0.3 nM for B-RafWT, B-RafV600E, and C-Raf, respectively. 了解更多 -
Tyrosine kinase-IN-1
Catalog No. A12486 multi-targeted tyrosine kinase inhibitorTyrosine kinase-IN-1 is a multi-targeted tyrosine kinase inhibitor with IC50s of 4, 20, 4, 2 nM for KDR, Flt-1, FGFR1 and PDGFRα, respectively. 了解更多 -
Tyrosine kinase inhibitor
Catalog No. A15267 Tyrosine kinase 抑制剂Tyrosine kinase inhibitor是一种抑制酪氨酸激酶的药物。酪氨酸激酶是负责通过信号转导级联反应激活许多蛋白质的酶。 了解更多 -
Bozitinib
Catalog No. A18554 c-MET kinase inhibitorBozitinib (PLB-1001) is a highly selective c-MET kinase inhibitor with blood-brain barrier permeability. Bozitinib (PLB-1001) is a ATP-competitive small-molecule inhibitor, binds to the conventional ATP-binding pocket of the tyrosine kinase superfamily. 了解更多 -
Pim1/AKK1-IN-1
Catalog No. A11476 multi-kinase inhibitorPim1/AKK1-IN-1 is a potent multi-kinase inhibitor with Kd values of 35 nM/53 nM/75 nM/380 nM for Pim1/AKK1/MST2/LKB1 respectively, and also inhibits MPSK1 and TNIK. 了解更多 -
RIPK1-IN-4
Catalog No. A21029 RIP1 kinase inhibitorRIPK1-IN-4 (compound 8) is a potent and selective type II kinase inhibitor of receptor interacting protein 1 (RIP1) kinase and binds to a DLG-out inactive form of RIP1 with an IC50s of 16 nM and 10 nM for RIP1 and ADP-Glo kinase. 了解更多 -
Tesevatinib
Catalog No. A21875 multi-target tyrosine kinase inhibitorTesevatinib (XL-647; EXEL-7647; KD-019) is an orally available, multi-target tyrosine kinase inhibitor; inhibits EGFR, ErbB2, KDR, Flt4 and EphB4 kinase with IC50s of 0.3, 16, 1.5, 8.7, and 1.4 nM. 了解更多 -
Rigosertib
Catalog No. A21868 multi-kinase inhibitorRigosertib (ON-01910) is a multi-kinase inhibitor and a selective anti-cancer agent, which induces apoptosis by inhibition the PI3 kinase/Akt pathway, promots the phosphorylation of histone H2AX and induces G2/M arrest in cell cycle. 了解更多 -
Cenisertib
Catalog No. A11262 multi-kinase inhibitorCenisertib (AS-703569) is a multi-kinase inhibitor that blocks the activity of Aurora-kinase-A/B, ABL1, AKT, STAT5 and FLT3. 了解更多 -
c-Fms-IN-1
Catalog No. A21047 FMS kinase inhibitorc-Fms-IN-1 is a FMS kinase inhibitor with an IC50 of 0.0008 μM. 了解更多 -
Ilorasertib
Catalog No. A20982 ATP-competitive multitargeted kinase inhibitorIlorasertib (ABT-348) is a potent and ATP-competitive multitargeted kinase inhibitor, which inhibits Aurora C, Aurora B, and Aurora A with IC50s of 1 nM, 7 nM, 120 nM, respectively. 了解更多 -
Sulfatinib
Catalog No. A21915 tyrosine kinase inhibitorSulfatinib (HMPL-012) is a potent and highly selective tyrosine kinase inhibitor against VEGFR1/2/3, FGFR1 and CSF1R with IC50s of in a range of 1 to 24 nM. 了解更多 -
(R)-Simurosertib
Catalog No. A21894 CDC7 kinase inhibitor(R)-Simurosertib ((R)-TAK-931) is the (R)-enantiomer of Simurosertib, Simurosertib (TAK-931) is a selective cycle 7 (CDC7) kinase inhibitor, with an IC50<0.3 nM. 了解更多 -
Rigosertib sodium
Catalog No. A21824 multi-kinase inhibitorRigosertib sodium (ON-01910 sodium) is a multi-kinase inhibitor and a selective anti-cancer agent, which induces apoptosis by inhibition the PI3K/Akt pathway, promotes the phosphorylation of histone H2AX and induces G2/M arrest in cell cycle. 了解更多 -
DDR1-IN-1 dihydrochloride
Catalog No. A21813 DDR1 receptor tyrosine kinase inhibitorDDR1-IN-1 dihydrochloride is a potent and selective DDR1 receptor tyrosine kinase inhibitor with an IC50 of 105 nM; 4-fold less potent for DDR2 (IC50 = 413 nM). 了解更多 -
BAY1217389
Catalog No. A21595 MPS1 kinase inhibitorBAY 1217389 is a potent, and selective inhibitor of the monopolar spindle 1 (MPS1) kinase with an IC50 value less than 10 nM. 了解更多 -
ENMD-2076 Tartrate
Catalog No. A21583 multi-targeted kinase inhibitorENMD-2076 Tartrate is a multi-targeted kinase inhibitor with IC50s of 1.86, 14, 58.2, 15.9, 92.7, 70.8, 56.4 nM for Aurora A, Flt3, KDR/VEGFR2, Flt4/VEGFR3, FGFR1, FGFR2, Src, PDGFRα, respectively. 了解更多 -
Amuvatinib hydrochloride
Catalog No. A21503 multi-targeted tyrosine kinase inhibitorAmuvatinib hydrochloride (MP470 hydrochloride) is an orally bioavailable multi-targeted tyrosine kinase inhibitor with potent activity against mutant c-Kit, PDGFRα, Flt3, c-Met and c-Ret. 了解更多 -
Acumapimod
Catalog No. A21325 p38 MAP kinase inhibitorAcumapimod (BCT197) is an orally active p38 MAP kinase inhibitor, with an IC50 of less than 1 μM for p38α.385.42 了解更多 -
B-Raf IN 1
Catalog No. A21055 B-Raf kinase inhibitorB-Raf IN 1 is a potent and selective B-Raf kinase inhibitor with an IC50 of 24 nM. 了解更多 -
Lenvatinib mesylate
Catalog No. A17567 multi-targeted tyrosine kinase inhibitorLenvatinib mesylate (E7080 mesylate), an oral, multi-targeted tyrosine kinase inhibitor that inhibits VEGFR1-3, FGFR1-4, PDGFR, KIT, and RET, shows potent antitumor activities. 了解更多 -
CHMFL-ABL/KIT-155
Catalog No. A12421 ABL/c-KIT dual kinase inhibitorCHMFL-ABL/KIT-155 (CHMFL-ABL-KIT-155; compound 34) is a highly potent and orally active type II ABL/c-KIT dual kinase inhibitor. 了解更多
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