“ADM Hydrochloride”的搜索结果

产品 101 到 147 共 147个

每页
页面:
  1. 1
  2. 2
  3. 3

设置降序顺序
  1. Ractopamine HCl

    Catalog No. A17372
    Quick View
    beta-Adrenergic agonist
    Ractopamine HCl is a beta-Adrenergic agonist. It acts by being a full agonist at the TAAR1. 了解更多
  2. Antazoline HCl

    Catalog No. A16411
    Quick View
    Histamine H1 receptor 抑制剂
    Antazoline HCl是第一代抗组胺药,可与组胺H1受体结合并阻断内源性组胺的作用。 了解更多
  3. SKF38393 HCl

    Catalog No. A15839
    Quick View
    Dopamine Receptor 激动剂?
    SKF38393 HCl是D1激动剂,IC50为110 nM。 了解更多
  4. Xylazine HCl

    Catalog No. A13434
    Quick View
    Adrenergic Receptor 激动剂
    Xylazine hydrochloride是α2A-AR、α2B-AR和α2C-AR的活化剂。 了解更多
  5. S(-)-Propranolol HCl

    Catalog No. A13428
    Quick View
    β-adrenergic blocker
    S(-)-Propranolol HCl是一种非选择性的β-肾上腺素能受体(βAR)拮抗剂,对β1AR和β2AR具有高亲和力,Ki值分别为1.8 nM和0.8 nM。 盐酸普萘洛尔抑制[3H] -DHA与大鼠脑膜制剂的结合,IC50为12 nM。 了解更多
  6. Atomoxetine HCl

    Catalog No. A13424
    Quick View
    norepinephrine (NE) transporter 抑制剂
    Atomoxetine HCl是SLC6A2的一种竞争性特异性抑制剂,同时在大鼠下丘脑突触体中显示出微弱的ST和DAT抑制作用。 了解更多
  7. Dexmedetomidine HCl

    Catalog No. A11846
    Quick View
    alpha2-adrenoceptor 激动剂
    Dexmedetomidine hydrochloride是美托咪啶的活性异构体,它充当有效的,高度选择性的α2-AR(α2-肾上腺素受体)激动剂。 了解更多
  8. MPEP HCl

    Catalog No. A13236
    Quick View
    mGlu5 receptor 拮抗剂
    MPEP HCl是对mGlu5a受体亚型(IC50 = 36 nM)的有效,高度选择性的非竞争性拮抗剂,但在浓度高达30 uM的mGlu1b受体上无激动剂或拮抗剂活性。 了解更多
  9. Ivabradine HCl (Procoralan)

    Catalog No. A11868
    Quick View
    Ivabradine Hydrochloride,也称为S-16257,是缓动剂伊伐布雷定的盐酸盐制剂。 了解更多
  10. Haloperidol hydrochloride

    Catalog No. A18304
    Quick View
    dopamine D2 receptor antagonist
    Haloperidol hydrochloride is a potent dopamine D2 receptor antagonist, widely used as an antipsychotic. 了解更多
  11. Chlorcyclizine hydrochloride

    Catalog No. A18025
    Quick View
    histamine H1 antagonist
    Chlorcyclizine hydrochloride is a histamine H1 antagonist. 了解更多
  12. Trimethobenzamide hydrochloride

    Catalog No. A17648
    Quick View
    D2 receptor blocker
    Trimethobenzamide hydrochloride is a blocker of the D2 receptor. Trimethobenzamide is an antiemetic used to prevent nausea and vomiting. 了解更多
  13. Moxisylyte hydrochloride

    Catalog No. A17725
    Quick View
    alpha-adrenergic blocking agent
    Moxisylyte hydrochloride is an alpha-adrenergic blocking agent that is used in Raynaud's disease. It is also used locally in the eye to reverse the mydriasis caused by phenylephrine and other sympathomimetic agents. 了解更多
  14. Cyproheptadine hydrochloride

    Catalog No. A16169
    Quick View
    serotonin/histamine2 拮抗剂
    Cyproheptadine hydrochloride是抗组胺药,是5-羟色胺和组胺的拮抗剂。 了解更多
  15. Alosetron Hydrochloride

    Catalog No. A14989
    Quick View
    5HT3-receptor 拮抗剂
    Alosetron Hydrochloride是一种5-羟色胺5HT3受体拮抗剂,可用于治疗肠易激综合症。 了解更多
  16. SB-408124 HCl

    Catalog No. A15231
    Quick View
    OX Receptor 拮抗剂
    SB408124 Hydrochloride是OX1受体的非肽拮抗剂,全细胞和膜的Ki分别为57 nM和27 nM。表现出比OX2受体高50倍的选择性。 了解更多
  17. rac-Rotigotine Hydrochloride

    Catalog No. A15217
    Quick View
    D2 receptor 激动剂
    rac-Rotigotine Hydrochloride是D-2受体的高效效价和选择性激动剂,Ki为0.69 nM。 了解更多
  18. Pitolisant hydrochloride

    Catalog No. A15213
    Quick View
    Nonimidazole inverse 激动剂
    Pitolisant hydrochloride是一种在重组人H3受体(Ki = 0.16 nM)处新颖,有效且选择性的壬二唑反向激动剂。 了解更多
  19. MTEP hydrochloride

    Catalog No. A15174
    Quick View
    mGlu5 拮抗剂
    MTEP hydrochloride是一种有效的,选择性和非竞争性的mGlu5拮抗剂,IC50和Ki分别为5 nM和16 nM。 了解更多
  20. Guanfacine hydrochloride

    Catalog No. A15098
    Quick View
    α2A-adrenoceptor 激动剂
    Guanfacine hydrochloride是一种抗高血压药,是一种选择性的α2A肾上腺素受体激动剂,Kd为31 nM,选择性是α2B肾上腺素受体的60倍。 了解更多
  21. Clemizole hydrochloride

    Catalog No. A15047
    Quick View
    H1 histamine receptor 拮抗剂
    Clemizole hydrochloride是H1组胺受体的拮抗剂,对NS4B RNA结合的IC50值为8 mM。 了解更多
  22. Siramesine Hydrochloride

    Catalog No. A12479
    Quick View
    Sigma-2 receptor 激动剂
    Siramesine Hydrochloride是一种选择性sigma-2受体激动剂,已被证明可触发癌细胞的细胞死亡并在体内表现出强大的抗癌活性。 了解更多
  23. CP 945598 HCl (Otenabant HCl)

    Catalog No. A11942
    Quick View
    CB1 拮抗剂
    CP 945598 HCl (Otenabant HCl)是一种有效且高度选择性的CB1拮抗剂。 了解更多
  24. Ozagrel hydrochloride

    Catalog No. A11742
    Quick View
    Thromboxane A2 synthesis 抑制剂
    Ozagrel hydrochloride是一种抗血小板剂,用作血栓烷a2合成抑制剂。 了解更多
  25. Terazosin hydrochloride

    Catalog No. A11740
    Quick View
    Terazosin hydrochloride是一种选择性α1拮抗剂,用于治疗前列腺肥大(BPH)症状。 了解更多
  26. Betaxolol hydrochloride

    Catalog No. A11733
    Quick View
    Betaxolol hydrochloride是β1肾上腺素受体阻断剂,可作用于高血压和青光眼。 了解更多
  27. Cyproheptadine hydrochloride

    Catalog No. A11709
    Quick View
    Cyproheptadine hydrochloride 是 5-HT2 受体拮抗剂,IC50为0.6 nM。 了解更多
  28. Urapidil hydrochloride

    Catalog No. A11704
    Quick View
    Urapidil hydrochloride是α1肾上腺素受体拮抗剂、5-HT1A血清素受体部分激动剂和抗高血压药。 了解更多
  29. Phenylephrine HCl

    Catalog No. A11666
    Quick View
    α1-adrenergic receptor 激动剂
    Phenylephrine HCl是一种选择性的α1肾上腺素能受体激动剂,主要用作减充血剂,扩张瞳孔和增加血压的药物。 了解更多
  30. MK 3207 HCl

    Catalog No. A10598
    Quick View
    CGRP Receptor 拮抗剂
    MK 3207 hydrochloride是一种有效的CGRP受体拮抗剂,IC50为0.12 nM。 了解更多
  31. Rotigotine HCl

    Catalog No. A11118
    Quick View
    Dopamine Receptor 激动剂
    Rotigotine hydrochloride是一种多巴胺D2和D3受体激动剂。D2和D3的Ki值分别为13和0.71 nM。 了解更多
  32. BRL 52537 HCl

    Catalog No. A11210
    Quick View
    Opioid Receptors 激动剂
    BRL 52537 hydrochloride是一种高度选择性和有效的κ阿片类激动剂(Ki = 0.24 nM)。比吗啡强25倍。 了解更多
  33. Nefazodone hydrochloride

    Catalog No. A17622
    Quick View
    5-HT2 receptors inhibitor
    Nefazodone HCl is an inhibitor of 5-HT2 receptors, SERT, NET, and hERG K+ channels used to treat mood disorders. It decreases immobility time in the forced swim test. 了解更多
  34. Melitracen hydrochloride

    Catalog No. A17494
    Quick View
    dopamine D1/2 receptor antagonist
    Melitracen HCl ia potential dopamine D1/2 receptor antagonist used to treat depression. It is often co-administered with flupenthixol as a treatment for trigeminal neuralgia. It does not effect cardiovascular function. 了解更多
  35. Rimonabant hydrochloride

    Catalog No. A11548
    Quick View
    CB1 receptor inverse 激动剂
    Rimonabant hydrochloride是CB1受体反向激动剂。 了解更多
  36. Azasetron HCl

    Catalog No. A16417
    Quick View
    5-HT3 receptor 拮抗剂
    Azasetron HCl是一种选择性的5-HT3受体拮抗剂,IC50为0.33 nM,用于治疗癌症化学疗法引起的恶心和呕吐。 了解更多
  37. Lidocaine hydrochloride

    Catalog No. A16132
    Quick View
    Histamine H1-receptor 激动剂
    Lidocaine hydrochloride是用作抗心律不齐药物的局部麻醉药和心脏抑制剂。 了解更多
  38. CBiPES HCl

    Catalog No. A15811
    Quick View
    mGlu2 receptor modulator
    CBiPES HCl是mGluR-2的选择性正变构调节剂,IC50值为98.2 nM。 了解更多
  39. SCH 23390 HCl

    Catalog No. A13066
    Quick View
    D1/D5 receptor 拮抗剂
    SCH 23390 HCl是一种有效的多巴胺受体拮抗剂(D1和D5受体亚型的Ki值分别为0.2 nM和0.3 nM)。 了解更多
  40. Atrasentan HCl

    Catalog No. A15007
    Quick View
    Endothelin 拮抗剂 receptor
    Atrasentan hydrochloride是一种开发用于治疗前列腺癌的内皮素拮抗剂受体(IC50 = 0.0551 nM,ETA)。 了解更多
  41. Asenapine HCl

    Catalog No. A15002
    Quick View
    adrenergic receptor/5-HT receptor 抑制剂
    Asenapine hydrochloride抑制肾上腺素能受体(α1,α2A,α2B,α2C)的Ki为0.25-1.2 nM,还抑制5-HT受体(1A,1B,2A,2B,2C,5A,6、7),Ki为0.03- 4.0 nM。 了解更多
  42. Tamsulosin hydrochloride

    Catalog No. A14936
    Quick View
    α1 receptor 拮抗剂
    Tamsulosin hydrochloride是一种选择性的α1受体拮抗剂,是用于良性前列腺增生的药物。 了解更多
  43. Oxymetazoline hydrochloride

    Catalog No. A10686
    Quick View
    alpha-1 adrenergic 激动剂
    Oxymetazoline是一种选择性的α-1激动剂和部分α-2激动剂局部减充血剂,以盐酸羟甲唑啉的形式使用。 了解更多
  44. Roxatidine acetate hydrochloride

    Catalog No. A11921
    Quick View
    Roxatidine acetate hydrochloride是一种用于溃疡治疗的组胺H2受体拮抗剂。 了解更多
  45. Dobutamine hydrochloride

    Catalog No. A10325
    Quick View
    Adrenoceptors 激动剂
    Dobutamine hydrochloride是一种直接作用剂,其主要活性来自刺激心脏的β1肾上腺素能受体,增加收缩力和心输出量。 了解更多
  46. Clomipramine HCl

    Catalog No. A10231
    Quick View
    5-HT Receptor 激动剂
    Clomipramine HCl是下列转运蛋白的阻滞剂:5-羟色胺转运蛋白 (SERT)(Ki = 0.14 nM),去甲肾上腺素转运蛋白(NET)(Ki = 54 nM),多巴胺转运蛋白(DAT)(Ki = 3,020 nM),甘氨酸转运蛋白(GlyT/LeuT)。 了解更多
  47. Thioridazine hydrochloride

    Catalog No. A11119
    Quick View
    Thioridazine hydrochloride是一种多巴胺受体拮抗剂,具有抗精神病活性。 最近还报道了硫代哒嗪能够成功杀死人类癌症干细胞。 了解更多

产品 101 到 147 共 147个

每页
页面:
  1. 1
  2. 2
  3. 3

设置降序顺序
Rewards