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“glucagon receptor”的搜索结果

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  1. AZD9496 maleate
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    AZD9496 maleate

    Catalog No. A21726
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    estrogen receptor (ERα) antagonist
    AZD9496 maleate is a potent and selective estrogen receptor (ERα) antagonist with IC50 of 0.28 nM. AZD9496 maleate is an orally bioavailable selective oestrogen receptor degrader (SERD). 了解更多
  2. Fimasartan
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    Fimasartan

    Catalog No. A17477
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    non-peptide angiotensin II receptor antagonist
    Fimasartan is a non-peptide angiotensin II receptor antagonist (ARB) used for the treatment of hypertension and heart failure. Through oral administration, fimasartan blocks angiotensin II receptor type 1 (AT1 receptors), reducing pro-hypertensive actions of angiotensin II, such as systemic vasoconstriction and water retention by the kidneys. 了解更多
  3. Enclomiphene citrate
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    Enclomiphene citrate

    Catalog No. A21830
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    oestrogen receptor antagonist
    Enclomiphene citrate is a potent and orally active oestrogen receptor antagonist, with antioestrogenic property. 了解更多
  4. H3B-6545 Hydrochloride
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    H3B-6545 Hydrochloride

    Catalog No. A21629
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    estrogen receptor covalent antagonist
    H3B-6545 Hydrochloride is an oral, selective estrogen receptor covalent antagonist (SERCA). 了解更多
  5. Azilsartan D5
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    Azilsartan D5

    Catalog No. A21600
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    angiotensin II type 1 receptor antagonist
    Azilsartan D5 is the deuterium labeled Azilsartan(TAK-536), which is a specific and potent angiotensin II type 1 receptor antagonist. 了解更多
  6. Losartan (D4 Carboxylic Acid)
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    Losartan (D4 Carboxylic Acid)

    Catalog No. A21578
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    angiotensin II receptor antagonist
    Losartan D4 Carboxylic Acid is the deuterium labeled Losartan(EXP-3174), which is an angiotensin II receptor antagonist. 了解更多
  7. Fulvestrant R enantiomer
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    Fulvestrant R enantiomer

    Catalog No. A21545
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    estrogen receptor antagonist
    Fulvestrant R enantiomer (ICI 182780 R enantiomer; ZD 9238 R enantiomer; ZM 182780 R enantiomer) is the less active R enantiomer of Fulvestrant. Fulvestrant is a potent estrogen receptor antagonist with an IC50 of 9.4 nM. 了解更多
  8. Sparsentan
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    Sparsentan

    Catalog No. A20879
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    angiotensin II and endothelin A receptor antagonist
    Sparsentan (RE-021) is a highly potent dual angiotensin II and endothelin A receptor antagonist with Kis of 0.8 and 9.3 nM, respectively. 了解更多
  9. Azilsartan medoxomil monopotassium
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    Azilsartan medoxomil monopotassium

    Catalog No. A20860
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    angiotensin II receptor type 1 antagonist
    Azilsartan medoxomil monopotassium is an orally administered angiotensin II receptor type 1 antagonist with IC50 of 0.62 nM, which used in the treatment of adults with essential hypertension. 了解更多
  10. Valsartan
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    Valsartan

    Catalog No. A10962
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    angiotensin II receptor antagonist
    Valsartan (CGP-48933) is an angiotensin II receptor antagonist for the treatment of high blood pressure and heart failure. 了解更多
  11. SL910102
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    SL910102

    Catalog No. A13591
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    Angiotensin AT1 receptor antagonist
    SL910102 is a nonpeptide angiotensin AT1 receptor antagonist. 了解更多
  12. H3B-6545
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    H3B-6545

    Catalog No. A20100
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    Estrogen receptor antagonist
    H3B-6545 is an oral, selective estrogen receptor covalent antagonist (SERCA). 了解更多
  13. OP-3633
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    OP-3633

    Catalog No. A18468
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    Glucocorticoid Receptor Antagonist
    OP-3633 is a Potent Steroidal Glucocorticoid Receptor Antagonist with Enhanced Selectivity against the Progesterone and Androgen Receptors (IC50 = 29 nM). 了解更多
  14. Losartan
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    Losartan

    Catalog No. A17510
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    Angiotensin II receptor antagonist
    Losartan is an angiotensin II receptor antagonist, competing with the binding of angiotensin II to AT1 receptors with IC50 of 20 nM. 了解更多
  15. MDV3100
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    MDV3100

    Catalog No. A10562
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    Androgen receptor 拮抗剂
    MDV3100(Enzalutamide)是一种androgen-receptor (AR)拮抗剂。在AR研究中强烈推荐的抑制剂。 了解更多
  16. (R)-Elagolix
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    (R)-Elagolix

    Catalog No. A21184
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    GnRHR antagonist
    Elagolix is a highly potent, selective, orally-active, short-duration, non-peptide antagonist of the gonadotropin-releasing hormone receptor (GnRHR) (KD = 54 pM). 了解更多
  17. Azilsartan Medoxomil
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    Azilsartan Medoxomil

    Catalog No. A16420
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    angiotensin II receptor type 1 拮抗剂
    Azilsartan medoxomil是一种口服给药的1型血管紧张素II受体拮抗剂，IC50为0.62 nM。 了解更多
  18. Flutamide
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    Flutamide

    Catalog No. A10402
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    Androgen receptor 拮抗剂
    Flutamide是一种抗雄激素药物，其活性代谢洛丽塔与Ki值为55nM的雄激素受体结合，可作用于前列腺癌。 了解更多
  19. (E/Z)-4-hydroxy Tamoxifen
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    (E/Z)-4-hydroxy Tamoxifen

    Catalog No. A12532
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    Estrogen receptor 拮抗剂
    (E/Z)-4-hydroxy Tamoxifen是他莫昔芬的活性代谢产物，是一种选择性雌激素受体（ER）调节剂，广泛用于乳腺癌的治疗和化学预防治疗。 了解更多
  20. RU43044
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    RU43044

    Catalog No. A14340
    Glucocorticoid receptor 拮抗剂
    RU43044在骨肉瘤细胞而非人乳腺癌细胞中发挥显着的激动剂活性并激活MMTV-Luc转录。 了解更多
  21. BIBS39
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    BIBS39

    Catalog No. A14154
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    angiotensin II receptor 拮抗剂
    BIBS39是一种非肽血管紧张素II（AII）受体拮抗剂，可从其特异性结合位点置换[125I] AII，其AII亚型（AT1）受体和K（i）的K（i）值为29+/-7 nM。）AII亚型2（AT2）受体的480+/-110 nM）值。 了解更多
  22. EXP-3174
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    EXP-3174

    Catalog No. A15451
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    AT1 receptor 拮抗剂
    EXP-3174是一种有效的选择性非竞争性AT1受体拮抗剂，IC50值为37 nM。 了解更多
  23. AZD9496
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    AZD9496

    Catalog No. A15822
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    estrogen receptor downregulator and 拮抗剂
    AZD9496是一种有效的生物选择性雌激素受体下调剂和拮抗剂。 了解更多
  24. EPI-001
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    EPI-001

    Catalog No. A15814
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    Androgen Receptor 拮抗剂
    EPI-001是雄激素受体（AR）的拮抗剂，它通过与AR的N末端结构域（NTD）共价结合并阻断AR及其剪接变体（转录因子IC50）的转录活性所需的蛋白质相互作用抑制AR NTD反式激活6μM） 了解更多
  25. ODM-201
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    ODM-201

    Catalog No. A15797
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    Androgen receptor 拮抗剂
    ODM-201是一种有效且完全的人类AR（hAR）拮抗剂，IC50值为26 nM。 了解更多
  26. NIBR189
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    NIBR189

    Catalog No. A15775
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    EBI2 (GPR183) receptor 拮抗剂
    NIBR189是爱泼斯坦-巴尔病毒诱导的基因2（EBI2；GPR183）受体的小分子拮抗剂，IC50为16 nM（结合）和11 nM（功能性）。 了解更多
  27. Endoxifen
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    Endoxifen

    Catalog No. A12639
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    Estrogen receptor 拮抗剂
    Endoxifen是他莫昔芬的次生代谢产物。它是负责他莫昔芬在ER阳性乳腺癌中有效性的主要代谢物。Endoxifen Z-isomer抑制hERG, 这种作用具有浓度依赖性, IC50值为1.6μM。 了解更多
  28. N-desMethyl EnzalutaMide
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    N-desMethyl EnzalutaMide

    Catalog No. A13964
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    androgen-receptor (AR) 拮抗剂
    N-desMethyl EnzalutaMide用于治疗涉及雄激素，雌激素和孕激素受体的疾病。 了解更多
  29. Lonaprisan
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    Lonaprisan

    Catalog No. A14130
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    progesterone receptor 拮抗剂
    Lonaprisan是米非司酮相关类固醇的口服生物可利用的五氟乙基衍生物，具有抗孕激素活性。 了解更多
  30. Tasosartan
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    Tasosartan

    Catalog No. A10891
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    Angiotensin II receptor 拮抗剂
    Tasosartan是一种血管紧张素II受体拮抗剂。 了解更多
  31. AZD1981
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    AZD1981

    Catalog No. A13186
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    CRTH2 receptor 拮抗剂
    AZD1981作为疾病相关细胞系统的有效拮抗剂，可抑制DK-PGD2诱导的人嗜酸性粒细胞CD11b表达，IC50为10 nM。 了解更多
  32. PD 123319 ditrifluoroacetate
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    PD 123319 ditrifluoroacetate

    Catalog No. A13201
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    angiotensin AT2 receptor 拮抗剂
    PD 123319 ditrifluoroacetate是一种有效的，选择性的非肽血管紧张素AT2受体拮抗剂。大鼠肾上腺组织和大脑的IC50值分别为34和210 nM。 了解更多
  33. Tamoxifen Citrate
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    Tamoxifen Citrate

    Catalog No. A10885
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    Estrogen receptor 拮抗剂
    Tamoxifen Citrate是哺乳动物甾醇异构酶的选择性和有效抑制剂。 了解更多
  34. Eprosartan
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    Eprosartan

    Catalog No. A11121
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    AT1 receptor 拮抗剂
    Eprosartan是一种用于治疗高血压的血管紧张素II受体拮抗剂。 了解更多
  35. Cyproterone acetate
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    Cyproterone acetate

    Catalog No. A11409
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    Androgen Receptor 拮抗剂
    Cyproterone acetate是17-羟孕酮的合成衍生物，可作为雄激素受体拮抗剂以及具有弱孕激素和糖皮质激素活性的弱孕激素受体激动剂。 了解更多
  36. Bicalutamide (Casodex)
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    Bicalutamide (Casodex)

    Catalog No. A10142
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    Androgen Receptor 拮抗剂
    Bicalutamide (Casodex)是一种口服非甾体抗雄激素，用于治疗前列腺癌和多毛症。 了解更多
  37. (R)-Bicalutamide
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    (R)-Bicalutamide

    Catalog No. A10008
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    Androgen Receptor 拮抗剂
    (R)-Bicalutamide是一种活性的竞争性非甾体雄激素受体拮抗剂，对MDA 453细胞的IC50为0.17μM。 了解更多

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