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￥ 0.00 5-HT Receptors
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Agomelatine
Catalog No. A10048 -
BRL-15572 dihydrochloride
Catalog No. A11178 5-HT1D receptor 拮抗剂BRL-15572是一种选择性的h5-HT1D拮抗剂，相对于h5-HT1B表现出60倍的选择性，对一系列其他受体类型的亲和力很小或没有亲和力。 了解更多 -
WAY-100635
Catalog No. A11182 -
Naftopidil 2HCl
Catalog No. A10619 5-HT1A and α1-adrenergic receptor 拮抗剂Naftopidil 2HCl是选择性5-HT1A和α1-肾上腺素能受体拮抗剂，IC50分别为0.1μM和0.2μM。 了解更多 -
Puerarin (Kakonein)
Catalog No. A10759 5-HT2C receptor 拮抗剂Puerarin (Kakonein)是几种已知的异黄酮之一。Puerarin是5-HT2C受体和苯二氮卓类拮抗剂。Puerarin正在研究作为一种自微乳化药物递送系统。 了解更多 -
Tropisetron (ICS 205930)
Catalog No. A11226 -
Alosetron
Catalog No. A11310 -
SB269970 HCl
Catalog No. A11925 -
Asenapine maleate
Catalog No. A10091 H1 拮抗剂Asenapine maleate平对多种受体具有高亲和力（pKi），包括5-羟色胺5-HT1A（8.6），5-HT1B（8.4），5-HT2A（10.2），5-HT2B（9.8），5-HT2C（10.5），5 -HT5A（8.8），5-HT6（9.5）和5-HT7（9.9）受体，肾上腺素α1（8.9），α2A（8.9），α2B（9.5）和α2C（8.9）受体，多巴胺D1（ 8.9），D2（8.9），D3（9.4）和D4（9.0）受体以及组胺H1（9.0）和H2（8.2）受体。 了解更多 -
Ketanserin (Vulketan Gel)
Catalog No. A10497 5-HT2A serotonin receptor 拮抗剂Ketanserin (Vulketan Gel)是大鼠和人5-HT2A血清素受体拮抗剂，Ki为2.5 nM。 了解更多 -
Granisetron Hydrochloride
Catalog No. A10437 -
Mianserin hydrochloride
Catalog No. A10588 5-HT2/5-HT1 拮抗剂Mianserin hydrochloride是5-HT2/5-HT1拮抗剂。对5-HT6非选择性5-HT2受体拮抗剂具有中等亲和力。对5-HT6具有中等亲和力。 了解更多 -
Ondansetron HCl (GR 38032F)
Catalog No. A10674 5-HT Receptors 拮抗剂Ondansetron HCl (GR 38032F)是5-羟色胺5-HT3受体拮抗剂，主要用作止吐药，通常在化疗后用于治疗恶心和呕吐。 了解更多 -
Olanzapine (LY170053)
Catalog No. A10667 5-HT Receptors/D2 dopamine receptor 拮抗剂Olanzapine (LY170053)对5-HT2血清素和D2多巴胺受体拮抗剂具有高亲和力。 了解更多 -
Eletriptan
Catalog No. A13075 -
NAD 299 hydrochloride (Robalzotan)
Catalog No. A13092 5-HT1A receptor 拮抗剂NAD 299 hydrochloride (Robalzotan)是一种选择性的，高亲和力的5-HT1A受体拮抗剂（体外Ki = 0.6 nM）。 了解更多 -
SDZ 205-557 HCl
Catalog No. A13766 -
N-Desmethylclozapine
Catalog No. A13762 5-HT2C serotonin receptor 拮抗剂N-Desmethylclozapine是一种有效的选择性5-HT2C血清素受体拮抗剂。 了解更多 -
Lu AE58054 (Idalopirdine)
Catalog No. A12521 -
Tandospirone
Catalog No. A13293 5-HT Receptor 拮抗剂Tandospirone是5HT1A受体的部分激动剂。它以剂量依赖性方式显着降低氟哌啶醇诱导的运动迟缓。 了解更多 -
SB-742457
Catalog No. A14092 -
SB 399885 HCl
Catalog No. A14102 5-HT6 拮抗剂SB 399885 hydrochloride是一种有效的，脑渗透剂和口服活性的SR-6拮抗剂。它对SR-6的选择性比其他血清素受体高200倍（对于人类重组，天然大鼠和天然人类SR-6受体，pKi值分别为9.11、8.81和9.02）。 了解更多 -
Cyclobenzaprine HCl
Catalog No. A14255 -
Tropisetron HCL
Catalog No. A14375 5-HT3 receptor 拮抗剂Tropisetron HCL是选择性的5-HT3受体拮抗剂和α7烟碱样受体激动剂，对5-HT3受体的IC50为70.1±0.9 nM。 了解更多 -
NAN-190 hydrobromide
Catalog No. A13417 5-HT1A receptor 拮抗剂NAN-190 hydrobromide是一种广泛用于科学研究的药物和研究化学品。以前认为它是一种选择性的5-HT1A受体拮抗剂，但后来的发现表明它也能有效地阻断α2肾上腺素能受体。 了解更多 -
Clozapine N-oxide
Catalog No. A15048 5-HT1C receptor 拮抗剂Clozapine N-oxide是氯氮平的主要代谢产物，在体外可降低SR-2A（5-HT2血清素受体）密度。 了解更多 -
Ziprasidone
Catalog No. A15286 5-HT/dopamine receptor 拮抗剂Ziprasidone是5-HT（5-羟色胺）和多巴胺受体拮抗剂的组合，具有抗精神病活性。 了解更多 -
Alosetron Hydrochloride
Catalog No. A14989 -
Cyproheptadine hydrochloride
Catalog No. A16169 -
Azasetron HCl
Catalog No. A16417 5-HT3 receptor 拮抗剂Azasetron HCl是一种选择性的5-HT3受体拮抗剂，IC50为0.33 nM，用于治疗癌症化学疗法引起的恶心和呕吐。 了解更多 -
LY 334370 hydrochloride
Catalog No. A17027 5-HT1F 激动剂LY 334370 hydrochloride是一种选择性的5-HT1F受体激动剂（Ki值为1.87、16.4，> 100 (IC50)）。CAS：199673-74-0（LY 334370盐酸盐）；182563-08-2（LY 334370游离碱） 了解更多 -
Volinanserin
Catalog No. A17115 -
Dolasetron
Catalog No. A17595 5-HT3 receptor antagonistDolasetron is a serotonin 5-HT3 receptor antagonist used to treat nausea and vomiting following chemotherapy. Its main effect is to reduce the activity of the vagus nerve, which is a nerve that activates the vomiting center in the medulla oblongata. It does not have much antiemetic effect when symptoms are due to motion sickness. 了解更多 -
Dolasetron Mesylate
Catalog No. A17729 5-HT3 receptor antagonistDolasetron mesylate is a selective 5-HT3 receptor antagonist. 了解更多 -
Alprenolol hydrochloride
Catalog No. A17781 5-HT1A receptor antagonistAlprenolol (hydrochloride) is a non-selective beta blocker as well as 5-HT1A receptor antagonist. 了解更多 -
Alosetron (Hydrochloride(1:X))
Catalog No. A11309 Serotonin 5HT3-receptor antagonistAlosetron Hydrochloride(1:X) (GR 68755 Hydrochloride(1:X)) is a Serotonin 5HT3-receptor antagonist that is used in treatment of irritable bowel syndrome. 了解更多 -
SB 258585 HCl
Catalog No. A14026 5-HT6 serotonin receptor 拮抗剂SB 258585 hydrochloride是一种选择性和有效的SR-6拮抗剂。该化合物显示出比其他5-羟色胺受体亚型高160倍的选择性。 了解更多 -
Granisetron
Catalog No. A15096 -
WAY-100635 maleate salt
Catalog No. A15282 -
Ricasetron
Catalog No. A15499 -
LY278584
Catalog No. A15500 -
Lerisetron
Catalog No. A15501
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