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CGS-15943
Catalog No. A14327 -
Preladenant
Catalog No. A13504 -
DPCPX
Catalog No. A16104 -
Vipadenant (BIIB-014)
Catalog No. A13963 A2A receptor 拮抗剂Vipadenant，也称为BIIB014，CEB-4520，是针对帕金森氏症的有效，选择性和口服腺苷A2A受体拮抗剂。Vipadenant在帕金森氏病的常用模型中显示出强大的口服活性。 了解更多 -
Theophylline-7-acetic acid
Catalog No. A16822 -
Proxyphylline
Catalog No. A16821 A1 adenosine receptors 拮抗剂Proxyphylline是茶碱的衍生物，由于其心血管特性而被用作支气管扩张剂。它与A2腺苷受体（对于血小板，Ki = 850μM）选择性拮抗A1腺苷受体（对于牛脑，Ki = 82 nM）。 了解更多 -
AZD-4635 (HTL1071)
Catalog No. A16820 -
MRS1177
Catalog No. A16871 -
MRS1186
Catalog No. A16870 -
A2A receptor antagonist 1
Catalog No. A12567 adenosine A2A/A1 receptor antagonistA2A receptor antagonist 1 (CPI-444 analog) is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively. 了解更多 -
Tonapofylline
Catalog No. A21328 adenosine A1 receptor antagonistTonapofylline (BG 9928) is an orally active and selective adenosine A1 receptor antagonist with a Ki of 7.4 nM for human adenosine A1 receptor (hA1), which displays 915-fold selectivity versus human adenosine A2A receptor and 12-fold selectivity versus human adenosine A2B receptor and is used in development for the treatment of heart failure. 了解更多 -
Rolofylline
Catalog No. A21649 adenosine A1 receptor antagonistRolofylline (KW-3902) is a potent, selective adenosine A1 receptor antagonist that is under development for the treatment of patients with acute congestive heart failure and renal impairment. 了解更多 -
Derenofylline
Catalog No. A21990 adenosine A1 receptor antagonistDerenofylline (SLV 320) is a potent, selective and orally active adenosine A1 receptor antagonist, with Ki values of 1 nM, 200 nM and 398 nM for human A1, A3 and A2A receptors respectively. 了解更多 -
BAY-u 3405
Catalog No. A13751 -
MF498
Catalog No. A15532 -
PF-04418948
Catalog No. A12894 -
TG6-10-1
Catalog No. A15968 -
Grapiprant (CJ-023423)
Catalog No. A15964 prostaglandin EP4 receptor 拮抗剂Grapiprant (CJ-023423)是一种具有抗痛觉过敏特性的新型，有效且选择性的前列腺素EP4受体拮抗剂。 了解更多 -
GSK-269984A
Catalog No. A17096 -
CAY10471 Racemate
Catalog No. A11760 Prostaglandin D2 receptor CRTH2 antagonistCAY10471 Racemate (TM30089 Racemate) is a potent and highly selective prostaglandin D2 receptor CRTH2 antagonist. 了解更多 -
ONO-AE3-208
Catalog No. A11516 EP4 antagonistONO-AE3-208 is an EP4 antagonist, and suppresses cell invasion, migration, and metastasis of prostate cancer. 了解更多 -
MK-2894 sodium salt
Catalog No. A11498 EP4 antagonistMK-2894 sodium salt is a highly potent and selective second generation EP4 antagonist. 了解更多 -
Terutroban
Catalog No. A20884 thromboxane-prostaglandin receptor antagonistTerutroban is a thromboxane-prostaglandin receptor antagonist. 了解更多 -
CJ-42794
Catalog No. A21948 EP4 antagonistCJ-42794 is a selective prostaglandin E receptor subtype 4 (EP4) antagonist, inhibits [3H]-PGE2 binding to the human EP4 receptor with a mean pKi of 8.5, a binding affinity that was at least 200-fold more selective for the human EP4 receptor than other human EP receptor subtypes (EP1, EP2, and EP3). 了解更多 -
Ki16198
Catalog No. A11966 -
AM095 free base
Catalog No. A14180 LPA1 Receptor 拮抗剂AM095 free base是一种新型，有效且口服可生物利用的溶血磷脂酸1型受体（LPA1）拮抗剂，对小鼠或重组人LPA1的IC50值分别为0.73和0.98μM。 了解更多 -
ONO-7300243
Catalog No. A16644 LPA1 antagonistONO-7300243 is a novel, potent lysophosphatidic acid receptor 1 (LPA1) antagonist with IC50 of 0.16 μM. 了解更多 -
LPA1 antagonist 1
Catalog No. A21301 LPA1 antagonistLPA1 antagonist 1 is a highly selective Lysophosphatidic Acid receptor-1 (LPA1) antagonist with an IC50 of 25 nM. 了解更多 -
LPA2 antagonist 1
Catalog No. A21308 -
BMS-986020 sodium
Catalog No. A21842 LPA1 antagonistBMS-986020 sodium is a high-affinity lysophosphatidic acid receptor 1 (LPA1) antagonist. 了解更多 -
Zibotentan (ZD4054)
Catalog No. A11006 ETA-receptor 拮抗剂Zibotentan (ZD4054)是一种有效且特异性的ETA受体（内皮素A受体）拮抗剂（IC50 = 21 nM），对ETB没有抑制活性。 了解更多 -
Ambrisentan (BSF 208075)
Catalog No. A11291 EndothelinA receptor 拮抗剂Ambrisentan (BSF 208075)充当内皮素受体拮抗剂，对A型内皮素受体（ETA）具有选择性。 了解更多 -
Avosentan (SPP301)
Catalog No. A11301 -
Sitaxsentan sodium (TBC-11251)
Catalog No. A11564 ETA receptor 拮抗剂Sitaxsentan sodium (TBC-11251)是一种选择性内皮素受体A拮抗剂，IC50和Ki分别为1.4 nM和0.43 nM。 了解更多
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