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“rasgap ras p21”的搜索结果

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  1. Tipifarnib (Zarnestra)
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    Tipifarnib (Zarnestra)

    Catalog No. A10935
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    FTase 抑制剂
    Tipifarnib (Zarnestra)是一种法尼基转移酶抑制剂，可在激酶途径变得过度活跃之前的翻译后修饰步骤中抑制Ras激酶。 了解更多
  2. Decitabine
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    Decitabine

    Catalog No. A10292
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    DNA Methyltransferase 抑制剂
    Decitabine是一种次甲基化剂，它通过抑制DNA甲基转移酶来使DNA次甲基化。 了解更多
  3. Rasagiline
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    Rasagiline

    Catalog No. A11111
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    MAO B 抑制剂
    Rasagiline是MAO-B（单胺氧化酶-B）的选择性不可逆抑制剂。 了解更多
  4. Ibudilast (KC-404)
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    Ibudilast (KC-404)

    Catalog No. A11019
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    PDE 抑制剂
    Ibudilast (KC-404)是一种相对非选择性的phosphodiesterase抑制剂，具有抗炎和神经保护活性。 了解更多
  5. Dorzolamide HCL
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    Dorzolamide HCL

    Catalog No. A10333
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    carbonic anhydrase 抑制剂
    Dorzolamide HCl是一种碳酸酐酶抑制剂。它是一种抗青光眼剂，以滴眼剂的形式局部使用。盐酸度尔佐胺用于降低开角型青光眼和高眼压患者的眼内压升高。 了解更多
  6. Tioxolone
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    Tioxolone

    Catalog No. A11673
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    Carbonic anhydrase 抑制剂
    Tioxolone是一种抗痤疮制剂。 了解更多
  7. Brinzolamide
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    Brinzolamide

    Catalog No. A11765
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    Carbonic anhydrase 抑制剂
    Brinzolamide是一种碳酸酐酶抑制剂，IC50为3.19 nM。 了解更多
  8. Rasagiline mesylate
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    Rasagiline mesylate

    Catalog No. A11722
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    Monoamine oxidase 抑制剂
    Rasagiline mesylate是一种不可逆的单胺氧化酶抑制剂，在早期帕金森氏病中用作单一疗法，在较晚期的病例中用作辅助疗法。对于B型MAO，它对A型的选择性是14倍。 了解更多
  9. Diclofenamide
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    Diclofenamide

    Catalog No. A10303
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    Carbonic anhydrase 抑制剂
    Diclofenamide (or dichlorphenamide)是一种磺酰胺和间二氨磺酰苯类的碳酸酐酶抑制剂。 了解更多
  10. Indisulam (E7070)
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    Indisulam (E7070)

    Catalog No. A12325
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    Carbonic anhydrase inhbitor
    Indisulam (E7070)是一种碳酸酐酶抑制剂，也是一种靶向细胞周期G1期的新型合成磺酰胺。 了解更多
  11. SC-26196
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    SC-26196

    Catalog No. A12318
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    Δ6 desaturase 抑制剂
    SC-26196选择性δ6去饱和酶抑制剂(IC50 = 0.2 μM 体外)。 了解更多
  12. Erastin
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    Erastin

    Catalog No. A13822
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    VDAC 抑制剂
    Erastin是一种细胞可渗透的哌嗪基-喹唑啉酮化合物，在具有H-Ras突变的细胞中表现出癌基因选择性致死性。 了解更多
  13. Punicalagin
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    Punicalagin

    Catalog No. A12105
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    Carbonic anhydrase 抑制剂
    Punicalagin是一种鞣花单宁，一种酚类化合物。它是一种高活性碳酸酐酶抑制剂。 了解更多
  14. Punicalin
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    Punicalin

    Catalog No. A12106
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    Carbonic anhydrase 抑制剂
    Punicalin是一种高活性碳酸酐酶抑制剂。 了解更多
  15. Deltarasin HCl
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    Deltarasin HCl

    Catalog No. A13722
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    PDE-KRAS 抑制剂
    Deltarasin HCl是一种新型的抑制KRASPDEδ相互作用从而破坏致癌性KRAS信号的小分子。 了解更多
  16. DTP348
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    DTP348

    Catalog No. A14410
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    CAIX 抑制剂/ radiosensitizer
    DTP348是双重CAIX抑制剂/放射增敏剂。 了解更多
  17. U-104
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    U-104

    Catalog No. A14959
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    Carbonic anhydrase (CA) 抑制剂
    U-104是碳酸酐酶IX（CAIX）的新型脲基磺酰胺抑制剂。 了解更多
  18. FTI-277 HCl
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    FTI-277 HCl

    Catalog No. A14439
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    FTase 抑制剂
    FTI-277 HCl是法呢基转移酶（FTase）的抑制剂。一种高效的Ras CAAX拟肽药物，可拮抗H-Ras和K-Ras致癌信号。 了解更多
  19. Acetazolamide
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    Acetazolamide

    Catalog No. A15859
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    Carbonic Anhydrase 抑制剂
    Acetazolamide是一种有效的碳酸酐酶（CA）抑制剂，在临床实践中通常用作迅速降低眼内压（IOP）的直接且容易获得的选择。 了解更多
  20. Benzenesulfonamide
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    Benzenesulfonamide

    Catalog No. A13594
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    Carbonic anhydrase 抑制剂
    Benzenesulfonamide是碳酸酐酶的抑制剂。 了解更多
  21. Vorasidenib
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    Vorasidenib

    Catalog No. A16908
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    IDH1 抑制剂
    Vorasidenib (AG-881)是一种有效且选择性的口服抑制剂，可抑制细胞质中异柠檬酸脱氢酶1型(IDH1，IDH1 [NADP+]可溶)和2型（IDH2异柠檬酸脱氢酶[NADP+]）的突变形式。线粒体中的线粒体，具有潜在的抗肿瘤活性。 了解更多
  22. Ethoxzolamide
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    Ethoxzolamide

    Catalog No. A17359
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    Carbonic anhydrase inhibitor
    Ethoxzolamide is a carbonic anhydrase inhibitor with Ki of 1 nM. 了解更多
  23. Minaprine dihydrochloride
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    Minaprine dihydrochloride

    Catalog No. A17722
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    MAO-A inhibitor
    Minaprine is a reversible inhibitor of MAO-A; weakly inhibit acetylcholinesterase; an antidepressant for treatment of depression. 了解更多
  24. Lodenafil
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    Lodenafil

    Catalog No. A18029
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    PDE5 inhibitor
    Lodenafil is a potent phosphodiesterase type 5 (PDE5) inhibitor for the treatment of erectile dysfunction (ED). 了解更多
  25. Fosphenytoin disodium
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    Fosphenytoin disodium

    Catalog No. A18184
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    PDE3 inhibitor
    Fosphenytoin Sodium is the sodium salt form of fosphenytoin, a prodrug that is hydrolyzed to the anticonvulsant phenytoin. It is an PDE3 (phosphodiesterase 3) inhibitor. 了解更多
  26. CM-675
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    CM-675

    Catalog No. A18741
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    PDE5/HDAC-1 inhibitor
    CM-675 is a dual phosphodiesterase 5 (PDE5) and class I histone deacetylases-selective inhibitor, with IC50 values of 114 nM and 673 nM for PDE5 and HDAC1, respectively. CM-675 has potential to treat Alzheimer??s disease. 了解更多
  27. BPN14770
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    BPN14770

    Catalog No. A18663
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    PDE4D inhibitor
    BPN14770 is a selective phosphodiesterase 4D (PDE4D) allosteric inhibitor with IC50s of 7.8 nM and 7.4 nM for PDE4D7 and PDE4D3, respectively. 了解更多
  28. MT-3014
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    MT-3014

    Catalog No. A18580
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    PDE 10A inhibitor
    MT-3014 is a potent, highly selective and brain-penetrated phosphodiesterase 10A (PDE 10A) inhibitor, with IC50s of 0.062 nM and 0.09 nM for human PDE 10A and bovine PDE 10A, respectively. 了解更多
  29. PDE12-IN-3
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    PDE12-IN-3

    Catalog No. A18579
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    PDE12 inhibitor
    PDE12-IN-3 is a phosphodiesterase 12 (PDE12) inhibitor with a pXC50 of 7.68. Antiviral activity. 了解更多
  30. VP3.15
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    VP3.15

    Catalog No. A18538
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    dual PDE7/GSK-3 inhibitor
    VP3.15 is a potent, orally bioavailable and CNS-penetrant dual phosphodiesterase (PDE)7- glycogen synthase kinase (GSK)3 inhibitor, with IC50s of 1.59 μM and 0.88 μM for PDE7 and GSK-3, respectively. VP3.15 has neuroprotective and neuroreparative activities, thus as potential combined anti-inflammatory and pro-remyelinating therapies for multiple sclerosis (MS). 了解更多
  31. A939572
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    A939572

    Catalog No. A13298
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    SCD1 inhibitor
    A939572 is a potent, and orally bioavailable stearoyl-CoA desaturase1 (SCD1) inhibitor with IC50 values of <4 nM and 37 nM for mSCD1 and hSCD1, respectively. 了解更多
  32. PF-05085727
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    PF-05085727

    Catalog No. A20098
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    PDE2A inhibitor
    PF-05085727 is a potent, selective and brain penetrant Phosphodiesterase 2A (PDE2A) inhibitor with an IC50 of 2 nM. 了解更多
  33. PF-05180999
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    PF-05180999

    Catalog No. A13006
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    PDE2A inhibitor
    PF-05180999 is a phosphodiesterase 2A (PDE2A) inhibitor, with an IC50 of 1.6 nM. 了解更多
  34. Sildenafil citrate
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    Sildenafil citrate

    Catalog No. A10841
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    PDE5 inhibitor
    Sildenafil citrate is a potent phosphodiesterase type 5 (PDE5) inhibitor with IC50 of 5.22 nM. 了解更多
  35. Mirodenafil dihydrochloride
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    Mirodenafil dihydrochloride

    Catalog No. A18047
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    PDE-5 inhibitor
    Mirodenafil dihydrochloride (SK3530 dihydrochloride) is a phosphodiesterase type 5 (PDE-5) inhibitor developed for the treatment of erectile dysfunction. 了解更多
  36. Mirodenafil
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    Mirodenafil

    Catalog No. A21260
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    PDE-5 inhibitor
    Mirodenafil(SK3530) is a phosphodiesterase type 5 (PDE-5) inhibitor developed for the treatment of erectile dysfunction. 了解更多
  37. Rasagiline 13C3 mesylate racemic
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    Rasagiline 13C3 mesylate racemic

    Catalog No. A21350
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    Monoamine oxidase inhibitor
    Rasagiline 13C3 mesylate racemic is the deuterium labeled Rasagiline, which is an irreversible inhibitor of monoamine oxidase. 了解更多
  38. Saterinone hydrochloride
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    Saterinone hydrochloride

    Catalog No. A21402
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    PDE3 inhibitor
    Saterinone hydrochloride is a phosphodiesterase III (PDE III) inhibitor. 了解更多
  39. CVT-12012
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    CVT-12012

    Catalog No. A21447
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    SCD inhibitor
    CVT-12012 is a potent and orally bioavailable stearoyl-coA desaturase (SCD) inhibitor, with IC50s of 38 nM, 6.1 nM for rat microsomal and human HEPG2, respectively. 了解更多
  40. AMG 579
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    AMG 579

    Catalog No. A21478
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    PDE10A inhibitor
    AMG 579 is a potent, selective, and efficacious inhibitor of phosphodiesterase 10A (PDE10A) with an IC50 of 0.1 nM. 了解更多
  41. BAY 73-6691 racemate
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    BAY 73-6691 racemate

    Catalog No. A21745
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    PDE9 inhibitor
    BAY 73-6691 racemate is a phosphodiesterase 9 inhibitor extracted from patent WO 2017070293 A1. 了解更多
  42. VP3.15 dihydrobromide
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    VP3.15 dihydrobromide

    Catalog No. A21789
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    PDE7/GSK3 inhibitor
    VP3.15 dihydrobromide is a potent, orally bioavailable and CNS-penetrant dual phosphodiesterase (PDE)7- glycogen synthase kinase (GSK)3 inhibitor, with IC50s of 1.59 μM and 0.88 μM for PDE7 and GSK-3, respectively. 了解更多
  43. R 80123
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    R 80123

    Catalog No. A21836
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    phosphodiesterase inhibitor
    R 80123 is the Z-isomer of R 79595, is also a highly selective phosphodiesterase inhibitor. 了解更多
  44. IBMX
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    IBMX

    Catalog No. A21847
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    PDE inhibitor
    IBMX is a broad-spectrum phosphodiesterase (PDE) inhibitor, with IC50s of 6.5, 26.3 and 31.7 μM for PDE3, PDE4 and PDE5, respectively. 了解更多
  45. Olprinone
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    Olprinone

    Catalog No. A21869
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    PDE3 inhibitor
    Olprinone(Loprinone) is a selective phosphodiesterase 3 (PDE3) inhibitor. 了解更多
  46. MF-438
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    MF-438

    Catalog No. A20963
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    SCD1 inhibitor
    MF-438 is a potent and orally bioavailable stearoyl-CoA desaturase 1 (SCD1) inhibitor with an EC50 of 2.3 nM for rSCD1. 了解更多
  47. RSL3
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    RSL3

    Catalog No. A15865
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    Ferroptosis inhibitor
    RSL3 is a ferroptosis activator in a VDAC-independent manner,exhibiting selectivity for tumor cells bearing oncogenic RAS. 了解更多
  48. Lonafarnib (SCH66336)
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    Lonafarnib (SCH66336)

    Catalog No. A12328
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    FPTase 抑制剂
    Lonafarnib (SCH66336)是H-ras、K-ras-4B和N-ras的选择性FPTase抑制剂，IC50分别为1.9 nM、5.2 nM和2.8 nM。 了解更多
  49. FTI 277
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    FTI 277

    Catalog No. A12368
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    FTase 抑制剂
    FTI 277是一种抑制法呢基转移酶(FTase)的抑制剂(IC50 = 0.5 nM)。抑制全细胞的 H-Ras 和 K-Ras 加工(IC50值分别为0.1和10 nM)，破坏mapk的组成型H-Ras特异性激活。在人恶性胶质瘤细胞和许多其他肿瘤细胞系中引起显著的抗增殖作用。 了解更多

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