“AZ 960”的搜索结果

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  1. Clinafloxacin

    Catalog No. A16458
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    DNA gyrase and topoisomerase IV 抑制剂
    Clinafloxacin是一种氟喹诺酮,可双重抑制肺炎链球菌中的DNA促旋酶和拓扑异构酶IV。 了解更多
  2. Lincomycin hydrochloride (U-10149A)

    Catalog No. A10532
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    Lincomycin hydrochloride是Lincomycin的一水盐,是从林肯链霉菌中分离的林肯酰胺抗生素,据报道其抑制细菌蛋白质合成并依赖于浓度。 了解更多
  3. Dexrazoxane

    Catalog No. A17714
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    topoisomerase IIα inhibitor
    Dexrazoxane is an intracellular iron chelator and an inhibitor of topoisomerase IIα. 了解更多
  4. Zoliflodacin

    Catalog No. A22032
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    DNA gyrase/topoisomerase inhibitor
    Zoliflodacin (ETX0914;AZD0914) is a novel spiropyrimidinetrione bacterial DNA gyrase/topoisomerase inhibitor. 了解更多
  5. PARP-2-IN-1

    Catalog No. A20240
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    PARP-2 inhibitor
    PARP-2-IN-1 is a potent and selective PARP-2 inhibitor with an IC50 of 11.5 nM. 了解更多
  6. Talazoparib tosylate

    Catalog No. A20238
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    PARP1/2 inhibitor
    Talazoparib tosylate (BMN 673ts) is a novel, potent and orally available PARP1/2 inhibitor with an IC50 of 0.57 nM for PARP1. 了解更多
  7. RTS-V5

    Catalog No. A20099
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    HDAC/proteasome inhibitor
    RTS-V5 is a dual HDAC/proteasome inhibitor with IC50s of 6.9, 18, 15, 0.27, 0.53 μM for HDAC1, HDAC2, HDAC3, HDAC6, HDAC8, respectively. 了解更多
  8. FT895

    Catalog No. A19615
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    HDAC11 inhibitor
    FT895 is a potent and selective HDAC11 inhibitor with an IC50 of 3 nM. 了解更多
  9. HDAC-IN-5

    Catalog No. A20972
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    HDAC inhibitor
    HDAC-IN-5 is a histone deacetylase (HDAC) inhibitor. 了解更多
  10. SIRT-IN-1

    Catalog No. A20962
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    SIRT1/2/3 inhibitor
    SIRT-IN-1 is a potent inhibitor of SIRT1/2/3, with IC50s of 15, 10, 33 μM, respectively. 了解更多
  11. SIRT-IN-2

    Catalog No. A20961
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    SIRT1/2/3 inhibitor
    SIRT-IN-2 is a potent inhibitor of SIRT1/2/3, with IC50s of 4, 4, 7 μM, respectively. 了解更多
  12. MB-7133

    Catalog No. A22007
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    DNA synthesis inhibitor
    MB-7133 is a DNA synthesis inhibitor. 了解更多
  13. TAS-103

    Catalog No. A21954
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    DNA topoisomerase I/II inhibitor
    TAS-103 is a dual inhibitor of DNA topoisomerase I/II, used for cancer research. 了解更多
  14. Daunorubicin

    Catalog No. A21903
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    topoisomerase II inhibitor
    Daunorubicin (Daunomycin; RP 13057; Rubidomycin) is a topoisomerase II inhibitor with potent antineoplastic activities. 了解更多
  15. Dehydroaltenusin

    Catalog No. A21804
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    eukaryotic DNA polymerase α inhibitor
    Dehydroaltenusin is a small molecule selective inhibitor of eukaryotic DNA polymerase α, a type of antibiotic produced by a fungus with an IC50 value of 0.68 μM. 了解更多
  16. Nanatinostat

    Catalog No. A21625
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    HDAC inhibitor
    Nanatinostat (CHR-3996) is a potent, class I selective and orally active histone deacetylase (HDAC) inhibitor with an IC50 of 8 nM. 了解更多
  17. Givinostat hydrochloride

    Catalog No. A21487
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    HDAC inhibitor
    Givinostat hydrochloride (ITF-2357 hydrochloride) is a HDAC inhibitor with an IC50 of 198 and 157 nM for HDAC1 and HDAC3, respectively. 了解更多
  18. Gepotidacin

    Catalog No. A21086
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    topoisomerase II inhibitor
    Gepotidacin (GSK2140944) is a novel triazaacenaphthylene bacterial type II topoisomerase inhibitor. 了解更多
  19. CG-200745

    Catalog No. A20939
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    HDAC inhibitor
    CG-200745 is a potent HDAC inhibitor which has the hydroxamic acid moiety to bind zinc at the bottom of catalytic pocket. 了解更多
  20. KU 59403

    Catalog No. A20928
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    ATM inhibitor
    KU 59403 is a potent ATM inhibitor, with an IC50 of 3 nM. 了解更多
  21. Top1 inhibitor 1

    Catalog No. A13304
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    human topoisomerase I (Top1) inhibitor
    Top1 inhibitor 1 (compound 28) is a potent human topoisomerase I (Top1) inhibitor with an IC50 value of 29 nM. 了解更多
  22. MAC glucuronide phenol-linked SN-38

    Catalog No. A18403
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    DNA topoisomerase I inhibitor
    MAC glucuronide phenol-linked SN-38 is a pH-susceptible lactone MAC glucuronide phenol-linked SN-38 (DNA topoisomerase I inhibitor) drug linker. MAC glucuronide phenol-linked SN-38 is cytotoxic across L540cy cells and Ramos cells with IC50 values of 113 and 67 ng/mL, respectively. 了解更多
  23. MAC glucuronide α-hydroxy lactone-linked SN-38

    Catalog No. A18407
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    Topoisomerase I inhibitor
    MAC glucuronide α-hydroxy lactone-linked SN-38 (Topoisomerase I inhibitor) is a stabilized lactone MAC glucuronide α-hydroxy lactone-linked SN-38 drug linker. 了解更多
  24. PARP14 inhibitor H10

    Catalog No. A18616
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    PARP14 抑制剂
    PARP14 inhibitor H10, compound H 10, is a selective inhibitor against PARP14 (IC50=490 nM), over other PARPs (??24 fold over PARP1). PARP14 inhibitor H10 induces caspase-3/7-mediated cell apoptosis. 了解更多
  25. ddATP

    Catalog No. A18898
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    DNA polymerase 抑制剂
    dATP is a dideoxynucleotide, acts as a chain-elongating inhibitor of DNA polymerase, used for Sanger method for DNA sequencing. 了解更多
  26. CL2-SN-38

    Catalog No. A18945
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    DNA topoisomerase I inhibitor
    CL2-SN-38 is a part of the antibody drug conjugate (ADC), can conjugate with the anti-Trop-2-humanized antibody hRS7. SN-38 is a DNA topoisomerase I inhibitor. 了解更多
  27. AZD-7648

    Catalog No. A20049
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    DNA-PK inhibitor
    AZD-7648 is a potent and selective DNA-PK inhibitor. Anti-tumor activity. 了解更多
  28. AZD1390

    Catalog No. A16798
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    ATM 抑制剂
    AZD1390是一流的口服中枢神经渗透性ATM抑制剂,在细胞中的IC50为0.78 nM,对PIKK酶家族中密切相关的成员具有10,000倍以上的选择性,并且在多种激酶中均具有出色的选择性。 了解更多
  29. AZ31

    Catalog No. A16813
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    ATM 抑制剂
    AZ31是一种新的选择性ATM抑制剂,IC50<0.0012 uM,对密切相关的酶具有良好的选择性(对DNA-PK和PI3Kα的选择性大于500倍,对mTOR、PI3Kβ和PI3Kγ的选择性大于1000倍)。 了解更多
  30. AZ32

    Catalog No. A16814
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    ATM 抑制剂
    AZ32是ATM激酶的特异性抑制剂,对小鼠具有良好的BBB渗透性,ATM酶的IC50值<0.0062 uM。它对ATR有足够的选择性,并且具有较高的细胞通透性。 了解更多
  31. AZD0156

    Catalog No. A16419
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    ATM 抑制剂
    AZD0156是有效且选择性的ATM激酶抑制剂,具有潜在的化学/放射致敏和抗肿瘤活性。 了解更多
  32. Tubercidin

    Catalog No. A13285
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    Tubercidin是一种腺苷类似物,是一种从结核链霉菌获得的抗生素。 了解更多
  33. Saccharin 1-methylimidazole

    Catalog No. A16114
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    DNA and RNA synthesis activator
    Saccharin 1-methylimidazole被认为是DNA和RNA合成的通用活化剂。 了解更多
  34. AZ6102

    Catalog No. A15873
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    TNKS1/2 抑制剂
    AZ6102是有效的TNKS1/2抑制剂,对其他PARP家族酶具有100倍的选择性,对DLD-1细胞中Wnt途径的抑制作用的IC50为5 nM。 了解更多
  35. AZD6738 (Ceralasertib)

    Catalog No. A15794
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    ATR 抑制剂
    AZD6738是一种有效的ATR激酶抑制剂,对分离的酶的IC50为1 nM,对细胞中ATR激酶依赖性CHK1磷酸化的IC50为74 nM。 了解更多
  36. TH588

    Catalog No. A15537
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    MTH1 抑制剂
    TH588是一流的nudix水解酶家族抑制剂,可有效和选择性地参与并抑制细胞中的MTH1(IC50 = 5 nM)。 了解更多
  37. TH287

    Catalog No. A15536
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    MTH1 抑制剂
    TH287是一种有效的MTH1(NUDT1)抑制剂,IC50值为0.8 nM,对MTH2,NUDT5,NUDT12,NUDT14和NUDT16的效力较低。 了解更多
  38. 4-HQN

    Catalog No. A15370
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    PARP 抑制剂
    4-HQN已显示抑制PARP(聚(ADP-核糖)合成酶),该酶催化NAD+的ADP-核糖部分与各种蛋白质的共价结合。 了解更多
  39. CRT0044876

    Catalog No. A14304
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    APE1 抑制剂
    CRT0044876是一种有效的选择性APE1抑制剂,IC50约为3μM。 了解更多
  40. AZ-20

    Catalog No. A13205
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    ATR kinase 抑制剂
    AZ20是一种有效的选择性ATR抑制剂,IC50值为5 nM。 了解更多
  41. Apaziquone

    Catalog No. A12406
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    Apaziquone是吲哚醌生物还原前药和丝裂霉素C类似物,具有潜在的抗肿瘤和放射增敏活性。 了解更多
  42. AZD-2461

    Catalog No. A12393
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    PARP 抑制剂
    AZD2461是新型有效的PARP抑制剂,对P-糖蛋白的亲和力较低。 了解更多
  43. Azithromycin (Zithromax)

    Catalog No. A11803
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  44. Dacarbazine

    Catalog No. A10281
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    Dacarbazine是一种用于治疗各种癌症的抗肿瘤化学治疗药物。Dacarbazine是烷基化剂类别的成员,其通过向其DNA中添加烷基(CnH2n+1)来破坏癌细胞。 了解更多
  45. Pyroxamide (NSC 696085)

    Catalog No. A10764
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    HDAC 抑制剂
    Pyroxamide (NSC 696085)是亲和纯化的HDAC1的有效抑制剂,可导致乙酰化核心组蛋白在用该试剂培养的MEL细胞中积累。 了解更多
  46. Olaparib (AZD2281)

    Catalog No. A10111
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    PARP 抑制剂
    Olaparib (AZD2281)是聚ADP核糖聚合酶(PARP)的抑制剂,该酶是一种与DNA修复有关的酶。 了解更多

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