微信关注
Total item
Cart Subtotal
￥ 0.00 “Akt Inhibitor”的搜索结果
-
AKT Kinase Inhibitor
Catalog No. A11285 Akt kinase inhibitorAKT Kinase Inhibitor is an Akt kinase inhibitor with anti-tumor activity. 了解更多 -
AKT-IN-1
Catalog No. A21009 -
AKT inhibitor VIII (AKTI-1/2)
Catalog No. A11286 AKT 抑制剂AKT inhibitor VIII (AKTI-1/2)是一种细胞可渗透且可逆的喹喔啉化合物，在体外激酶测定中，该化合物有效和选择性地抑制Akt1/Akt2活性（对于Akt1，Akt2和Akt3，IC50分别为58 nM，210 nM和2.12μM）。 了解更多 -
Akt-l-1
Catalog No. A12435 -
Ipatasertib dihydrochloride
Catalog No. A21734 pan-Akt inhibitorIpatasertib dihydrochloride (GDC-0068 dihydrochloride) is a highly selective pan-Akt inhibitor targeting Akt1/2/3 with IC50 of 5/18/8 nM, 620-fold selectivity over PKA. 了解更多 -
Solenopsin
Catalog No. A21087 ATP-competitive AKT inhibitorSolenopsin is an ATP-competitive AKT inhibitor with IC50 value of 10 μM . 了解更多 -
Isobavachalcone
Catalog No. A11453 Akt inhibitorIsobavachalcone (Corylifolinin) is derived from Psoralea corylifolia Linn. and is a potent inhibitor of Akt signaling pathway, which induces apoptosis in human cancer cells (Inhibits OVCAR-8 cell growth with an IC50 value of 7.92 μM). 了解更多 -
Borussertib
Catalog No. A13364 Akt inhibitorBorussertib is a covalent-allosteric and first-in-class inhibitor of protein kinase Akt, with an IC50 of 0.8 nM and a Ki of 2.2 nM for Aktwt. 了解更多 -
Miransertib hydrochloride
Catalog No. A22376 Akt inhibitorMiransertib hydrochloride (ARQ-092 hydrochloride) is a potent, orally active, selective and allosteric Akt inhibitor with IC50s of 2.7 nM, 14 nM and 8.1 nM for Akt1, Akt2, Akt3, respectively. 了解更多 -
10-DEBC HCl
Catalog No. A13590 AKT/PKB 抑制剂?10-DEBC HCl是Akt/PKB的选择性抑制剂。它抑制IGF-1刺激的磷酸化和Akt的激活（在2.5μM时完全抑制），抑制mTOR，p70 S6激酶的下游激活。 了解更多 -
Palomid 529 (P529)
Catalog No. A10693 -
Histone Acetyltransferase Inhibitor II
Catalog No. A12331 cell permeable p300 inhibitorHistone Acetyltransferase Inhibitor II is a potent and cell permeable p300 inhibitor, with an IC50 of 5 ?M; Histone Acetyltransferase Inhibitor II can be used in cancer research. 了解更多 -
Src Inhibitor 1
Catalog No. A12299 Src tyrosine kinase inhibitorSrc Inhibitor 1 is a potent and selective dual site Src tyrosine kinase inhibitor with IC50 values of 44 nM for Src and 88nM for Lck. 了解更多 -
CPA inhibitor
Catalog No. A11369 -
GSK3 Inhibitor XIII
Catalog No. A22128 ATP-binding site inhibitor of GSK-3GSK3 Inhibitor XIII (GSK3i XIII) is an ATP-binding site inhibitor of GSK-3. 了解更多 -
ATR inhibitor 2
Catalog No. A22162 ATR inhibitorATR inhibitor 2 is an ATP-competitive, orally active, and selective ATR inhibitor, with a Ki of <150 pM. 了解更多 -
LMPTP INHIBITOR 1 dihydrochloride
Catalog No. A22227 LMPTP inhibitorLMPTP INHIBITOR 1 (dihydrochloride) is a selective inhibitor of low molecular weight protein tyrosine phosphatase (LMPTP), with an IC50 of 0.8 μM LMPTP-A. 了解更多 -
VPS34 inhibitor 1 (Compound 19)
Catalog No. A22378 VPS34 inhibitorVPS34 inhibitor 1 (Compound 19, PIK-III analogue) is a potent and selective inhibitor of VPS34 with an IC50 of 15 nM. 了解更多 -
Selective PI3Kδ Inhibitor 1 (compound 7n)
Catalog No. A22381 PI3Kδ inhibitorSelective PI3Kδ Inhibitor 1 (compound 7n) is an inhibitor of PI3Kδ with an IC50 of 0.9 nM and >1000-fold selectivity against other class I PI3K isoforms [PI3K α/γ/β=3670/1460/21300 nM]. 了解更多 -
BTK inhibitor 1 (Compound 27)
Catalog No. A22445 BTK inhibitorBTK inhibitor 1 (compound 27) is an inhibitor of BTK with an IC50 of 0.11 nM for Btk and inhibits B cell activation in hWB with an IC50 of 2 nM. 了解更多 -
Multi-kinase inhibitor 1
Catalog No. A22645 multi-kinase inhibitorMulti-kinase inhibitor 1 is a potent multi-kinase inhibitor. Multi-kinase inhibitor 1 has the potential for diseases or disorders associated with abnormal or deregulated tyrosine kinase activity, particularly diseases associated with the activity of PDGF-R, c-Kit and Bcr-abl. 了解更多 -
Diacylglycerol acyltransferase inhibitor-1
Catalog No. A20315 DGAT1 inhibitorDiacylglycerol acyltransferase inhibitor-1 is a diacylglycerol acyltransferase (DGAT1) inhibitor. 了解更多 -
MAT2A inhibitor 2
Catalog No. A20171 MAT2A inhibitorMAT2A inhibitor 2 is a methionine adenosyltransferase 2A (MAT2A) inhibitor. 了解更多 -
DAAO inhibitor-1
Catalog No. A20117 DAAO inhibitorDAAO inhibitor-1 is a potent D-amino acid oxidase (DAAO) inhibitor with an IC50 of 0.12 μM. 了解更多 -
Grp94 Inhibitor-1
Catalog No. A20073 Grp94 inhibitorGrp94 Inhibitor-1 is a potent, selective Grp94 inhibitor with an IC50 value of 2 nM, and over 1000-fold selectivity to Grp94 against Hsp90α. 了解更多 -
mTOR inhibitor-1
Catalog No. A20029 mTOR inhibitormTOR inhibitor-1 is a novel mTOR pathway inhibitor which can suppress cells proliferation and inducing autophagy. 了解更多 -
Tubulin inhibitor 1
Catalog No. A19998 tubulin inhibitorTubulin inhibitor 1 is a tubulin inhibitor, inhibits tubulin polymerization. 了解更多 -
YAP/TAZ inhibitor-1
Catalog No. A19976 YAP/TAZ inhibitorYAP/TAZ inhibitor-1 is a YAP/TAZ inhibitor extracted from patent WO2017058716A1, Compound 1, has an IC50 of <0.100 μμ in firefly luciferase assay. 了解更多 -
SIRT5 inhibitor 1
Catalog No. A19841 SIRT5 inhibitorSIRT5 inhibitor 1 is a potent Human Sirtuin 5 deacylase inhibitor, with an IC50 of 0.11 μM. 了解更多 -
BET bromodomain inhibitor
Catalog No. A19831 BET inhibitorBET bromodomain inhibitor is a potent BET inhibitor extracted from patent WO/2015/153871A2, compound example 11. 了解更多 -
TRAF-STOP inhibitor 6877002
Catalog No. A19758 CD40-TRAF6 interaction inhibitorTRAF-STOP inhibitor 6877002, is a selective inhibitor of CD40-TRAF6 interaction, compound VII, shows inhibition of NF-κB activation in RAW cells, extracted from patent WO2014033122A1. 了解更多 -
Glutaminyl Cyclase Inhibitor 1
Catalog No. A19723 glutaminyl cyclase inhibitorGlutaminyl Cyclase Inhibitor 1 is a glutaminyl cyclase inhibitor with an IC50 of 0.5 μM. 了解更多 -
PKC-theta inhibitor
Catalog No. A19712 PKC-θ inhibitorPKC-theta inhibitor is a selective PKC-θinhibitor, with an IC50 of 12 nM. 了解更多 -
LRRK2 inhibitor 1
Catalog No. A19701 LRRK2 inhibitorLRRK2 inhibitor 1 is a potent, selective and oral LRRK2 inhibitor with an pIC50 of 6.8 nM. 了解更多 -
PDGFRα kinase inhibitor 1
Catalog No. A19632 type II PDGFRα kinase inhibitorPDGFRα kinase inhibitor 1 is a highly selective type II PDGFRα kinase inhibitor with IC50s of 132 nM and 6115 nM for PDGFRα and PDGFRβ, respectively. 了解更多 -
HIV-1 integrase inhibitor 3
Catalog No. A19628 INST inhibitorHIV-1 integrase inhibitor 3 is a HIV-1 integrase strand transfer (INST) inhibitor with an IC50 of 2.7 nM. 了解更多 -
PI3K/mTOR Inhibitor-2
Catalog No. A19621 dual pan-PI3K/mTOR inhibitorPI3K/mTOR Inhibitor-2 is a potent dual pan-PI3K/mTOR inhibitor with IC50s of 3.4/34/16/1 nM for PI3Kα/PI3Kβ/PI3Kδ/PI3Kγ and 4.7 nM for mTOR. Antitumor activity. 了解更多 -
HIV-1 integrase inhibitor 4
Catalog No. A19617 INST inhibitorHIV-1 integrase inhibitor 4 is a HIV-1 integrase strand transfer (INST) inhibitor with an IC50 of 3.7 nM. 了解更多 -
Neurotoxin Inhibitor
Catalog No. A19507 -
Aurora Kinase Inhibitor 3
Catalog No. A19448 Aurora A kinase inhibitorAurora Kinase Inhibitor 3 is a strong and selective Aurora A kinase inhibitor with an IC50 of 42 nM, and weakly inhibits EGFR with an IC50>10 μM. 了解更多 -
p38α inhibitor 1
Catalog No. A19182 p38α inhibitorp38α inhibitor 1 is a p38α inhibitor extracted from patent WO 2008076265 A1. 了解更多 -
Bromodomain inhibitor-8
Catalog No. A19161 BET bromodomain inhibitorBromodomain inhibitor-8 (Intermediate 21) is a BET bromodomain inhibitor for treating autoimmune and inflammatory diseases. 了解更多
ADOOQ 产品质量保证
We promise all products to perform as described.