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Bivalirudin
Catalog No. A15023 -
Dabigatran etexilate mesylate
Catalog No. A15057 direct thrombin 抑制剂Dabigatran etexilate mesylate是达比加群的口服活性前药。达比加群是一种可逆的选择性直接凝血酶抑制剂（DTI），Ki值为4.5 nM。 了解更多 -
Dabigatran ethyl ester
Catalog No. A15058 -
Ximelagatran
Catalog No. A12509 -
Melagatran
Catalog No. A19083 Thrombin inhibitorMelagatran is a direct and orally active inhibitor of thrombin, without interacting with any other enzymes in the coagulation cascade or fibrinolytic enzymes aside from thrombin. 了解更多 -
RWJ-445167
Catalog No. A12154 dual inhibitor of thrombin and factor XaRWJ-445167 (3DP-10017) is a dual inhibitor of thrombin and factor Xa with Ki of 4.0 nM and 230 nM, respectively, exhibiting potent antithrombotic activity. 了解更多 -
Thrombin Inhibitor 2
Catalog No. A21814 thrombin inhibitorThrombin Inhibitor 2 is a small molecule direct thrombin inhibitor, extracted from US8541580B2. Thrombin Inhibitor 2 has antithrombotic activity. 了解更多 -
CHR2797 (Tosedostat)
Catalog No. A10208 Aminopeptidase 抑制剂CHR2797 (Tosedostat)是一种新型金属酶抑制剂，在体内和体外对多种肿瘤细胞系均具有抗增殖作用，并表现出选择性。 了解更多 -
Bestatin Methyl Ester
Catalog No. A13592 Aminopeptidase 抑制剂Bestatin Methyl Ester是Bestatin的细胞可渗透衍生物，其对中性氨肽酶的抑制比Bestatin稍强，但对碱性氨肽酶的活性弱得多。 了解更多 -
Fumagillin
Catalog No. A15299 Aminopeptidase 抑制剂Fumagillin是一种复杂的天然产物抗生素，它与II型蛋氨酸氨基肽酶（MetAP-2）的关键组氨酸残基共价结合，抑制内皮细胞增殖和血管生成。 了解更多 -
Nafamostat mesylate
Catalog No. A10617 serine protease 抑制剂Nafamostat mesylate是一种抗凝剂。广谱丝氨酸蛋白酶抑制剂。在哮喘小鼠模型中减少嗜酸性粒细胞浸润，肥大细胞活化和气道反应性。 了解更多 -
BCX 1470
Catalog No. A11331 -
BCX 1470 methanesulfonate
Catalog No. A11325 Serine protease 抑制剂BCX 1470 methanesulfonate是丝氨酸蛋白酶抑制剂。BCX 1470在体外阻断补体酶CLs和因子D的酯酶和溶血活性。 了解更多 -
Sivelestat sodium salt
Catalog No. A14073 Neutrophil elastase 抑制剂Sivelestat sodium salt是一种选择性白细胞弹性蛋白酶抑制剂（IC50 = 44 nM），在一系列其他蛋白酶中均无活性。它在体外抑制NF-κB活化和LTB4诱导的中性粒细胞转运。 了解更多 -
Alvelestat
Catalog No. A12779 neutrophil elastase 抑制剂Avelestat，也称为AZD9668，是可口服的,高度选择性neutrophil elastase (NE)抑制剂，IC50和Ki分别为12 nM和9.4 nM,其选择性超过其他丝氨酸蛋白酶至少600倍。 了解更多 -
AEBSF HCl
Catalog No. A14270 -
Sivelestat
Catalog No. A14184 Neutrophil elastase 抑制剂Sivelestat是一种可渗透细胞的磺酰苯胺化合物，可作为中性粒细胞弹性蛋白酶的强效，底物竞争性和高度特异性抑制剂（大鼠，兔，仓鼠，人类和小鼠白细胞弹性蛋白酶的IC50 = 19-49 nM）。 了解更多 -
SSR 69071
Catalog No. A15315 -
PMSF
Catalog No. A11901 -
Sivelestat sodium hydrate (ONO-5046 sodium hydrate)
Catalog No. A16137 Neutrophil elastase 抑制剂Sivelestat sodium hydrate (ONO-5046 sodium hydrate)是人嗜中性粒细胞弹性蛋白酶的竞争性抑制剂，还抑制从兔，大鼠，仓鼠和小鼠获得的白细胞弹性蛋白酶。 了解更多 -
Fumonisin B1
Catalog No. A15379 serine/threonine phosphatase 抑制剂Fumonisin B1是由镰孢镰刀菌（Fusarium moniliforme）产生的真菌代谢产物，已显示可抑制蛋白质丝氨酸/苏氨酸磷酸酶（PP1，PP2A，PP2B，PP2C和PP5/T/K/H），并且对PP5最有效。 了解更多 -
Nafamostat hydrochloride
Catalog No. A20828 serine protease inhibitorNafamostat hydrochloride is an anticoagulant. Broad spectrum serine protease inhibitor. Reduces eosinophil infiltration, mast cell activation and airway responsiveness in a murine model of asthma. 了解更多 -
Nafamostat
Catalog No. A20827 serine protease inhibitorNafamostat is an anticoagulant. Broad spectrum serine protease inhibitor. Reduces eosinophil infiltration, mast cell activation and airway responsiveness in a murine model of asthma. 了解更多 -
Odanacatib (MK-0822)
Catalog No. A11265 -
CA-074
Catalog No. A13256 -
E 64d (Aloxistatin)
Catalog No. A13259 Cysteine Protease 抑制剂E 64d (Aloxistatin)是组织蛋白酶B和L的抑制剂，具有溶酶体和细胞渗透性。 了解更多 -
Leupeptin hemisulfate
Catalog No. A14145 -
Loxistatin Acid (E64-C)
Catalog No. A13258 -
E-64
Catalog No. A13257 -
CA-074 Methyl Ester
Catalog No. A13593 Cathepsin B 抑制剂CA-074 Methyl Ester是CA-074的细胞渗透性类似物，用作不可逆组织蛋白酶B抑制剂。据报道，CA-074甲酯在啮齿动物模型中抑制骨吸收，并显示在体外抑制B16黑素瘤细胞侵袭。 了解更多 -
Z-FL-COCHO
Catalog No. A13502 -
SID 26681509
Catalog No. A15313 -
Balicatib
Catalog No. A12020 -
MG-101
Catalog No. A14220 -
PD 151746
Catalog No. A14245 -
Calpain Inhibitor II, ALLM
Catalog No. A14911 Calpain 抑制剂Calpain Inhibitor II, ALLM是钙蛋白酶I，钙蛋白酶II，组织蛋白酶L和组织蛋白酶B的细胞可渗透抑制剂，Ki值分别为120 nM，230 nM，0.6 nM和100 nM。 了解更多 -
Acetyl-Calpastatin (184-210) (human)
Catalog No. A15290 Selective calpain 抑制剂Acetyl-Calpastatin (184-210) (human)选择性钙蛋白酶抑制剂。强烈抑制钙蛋白酶I（Ki = 0.2 nM）和II，但不抑制木瓜蛋白酶，胰蛋白酶和组织蛋白酶L（Ki = 6 uM）。增加淀粉样β蛋白（Aβ）42，Aβ40和Aβ42比率的分泌。 了解更多 -
Calpeptin
Catalog No. A15295
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