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Letaxaban (TAK-442)
Catalog No. A12871 factor Xa 抑制剂Letaxaban (TAK-442)是一种有效的，选择性的，口服活性的Xa抑制剂，是一种四氢嘧啶-2（1H）-衍生物。TAK-442在贫血小板的人[半最大抑制浓度（IC（50））：53 nM，TAK-442]和大鼠（IC（50）：32 nM，TAK-442）血浆中抑制内源性FXa活性。 了解更多 -
TAK-242 S enantiomer
Catalog No. A15253 TLR4 抑制剂TAK-242的S对映体。TAK-242（Resatorvid），Toll样受体（TLR）4信号转导的小分子抑制剂。TAK-242用于治疗败血症和败血性休克。 了解更多 -
TAK-700 Salt (Orteronel Salt)
Catalog No. A13515 CYP17A1/androgen synthesis 抑制剂TAK-700 Salt (Orteronel Salt)是一种雄激素合成抑制剂。它选择性地抑制在睾丸，肾上腺和前列腺肿瘤组织中表达的酶CYP17A。 了解更多 -
TAK-960 hydrochloride
Catalog No. A21703 PLK1 inhibitorTAK-960 hydrochloride is an orally available, selective inhibitor of polo-like kinase 1 (PLK1), with an IC50 of 0.8 nM at 10 μM ATP; TAK-960 hydrochloride also shows inhibitory activities against PLK2 and PLK3, with IC50s of 16.9 and 50.2 nM, respectively. 了解更多 -
TAK-659 hydrochloride
Catalog No. A21885 Syk inhibitorTAK-659 hydrochloride is a potent, selective and orally available spleen tyrosine kinase (Syk) inhibitor with an IC50 of 3.2 nM. 了解更多 -
TAK-063
Catalog No. A15799 -
TAK-441
Catalog No. A11351 -
TAK-960
Catalog No. A11146 -
TAK-700 (Orteronel)
Catalog No. A11044 -
Mubritinib (TAK 165)
Catalog No. A10612 HER2/ErbB2 抑制剂Mubritinib (TAK 165)是一种有效的EGFR和p34cdc2抑制剂，IC50分别为6 nM和0.2 ?M。Mubritinib（TAK 165）也抑制p33cdk2和p33cdk5。 了解更多 -
(R)-Simurosertib
Catalog No. A21894 CDC7 kinase inhibitor(R)-Simurosertib ((R)-TAK-931) is the (R)-enantiomer of Simurosertib, Simurosertib (TAK-931) is a selective cycle 7 (CDC7) kinase inhibitor, with an IC50<0.3 nM. 了解更多 -
Lapaquistat acetate
Catalog No. A20851 squalene synthase inhibitorLapaquistat acetate (TAK-475) is a squalene synthase inhibitor, blocking the conversion of farnesyl diphosphate (FPP) to squalene. 了解更多 -
Resatorvid
Catalog No. A11543 TLR4 inhibitorResatorvid (TAK-242) is a selective Toll-like receptor 4 (TLR4) inhibitor and plays pivotal role in various inflammatory diseases. 了解更多 -
Cenicriviroc Mesylate
Catalog No. A17028 CCR2/5 receptors 抑制剂Cenicriviroc(TAK-652,TBR-652)是CCR2和CCR5受体的抑制剂，可使其充当防止病毒进入人细胞的进入抑制剂 了解更多 -
MLN1117 (Serabelisib)
Catalog No. A15529 p110α 抑制剂MLN1117，也称为INK1117和TAK-117，是具有潜在抗肿瘤活性的I类磷酸肌醇3激酶（PI3K）α同工型的生物利用抑制剂。 了解更多 -
Lapaquistat
Catalog No. A21262 cholesterol biosynthesis inhibitorLapaquistat (T-91485), a cholesterol biosynthesis inhibitor, is the active metabolite of TAK-475. Lapaquistat can decrease statin-induced myotoxicity in lipid-lowering therapy. 了解更多 -
Cenicriviroc
Catalog No. A13643 CCR2/CCR5 抑制剂Cenicriviroc是用于治疗HIV感染的实验性候选药物.Cenicriviroc是CCR2和CCR5受体的抑制剂，可使其充当阻止病毒进入人体细胞的进入抑制剂。 了解更多 -
Eplivanserin mixture
Catalog No. A21987 serotonin reuptake inhibitor/5-HT2A receptor antagonistEplivanserin mixture is a selective serotonin reuptake inhibitor and a 5-HT2A receptor antagonist, extracted from patent WO 2005/002578 A1. 了解更多 -
Vanoxerine
Catalog No. A21922 dopamine reuptake inhibitorVanoxerine (GBR-12909) is a competitive, potent, and highly selective dopamine reuptake inhibitor (Ki=1 nM). 了解更多 -
Vilazodone D8
Catalog No. A21876 SSR inhibitor / 5-HT1A receptor partial agonistVilazodone D8 is the a deuterium labeled vilazodone, which is a combined serotonin specific reuptake inhibitor (SSRI) and 5-HT1A receptor partial agonist. 了解更多 -
LY2365109 hydrochloride
Catalog No. A21779 GlyT1 inhibitorLY2365109 hydrochloride is a potent and selective GlyT1 inhibitor, with an IC50 of 15.8 nM for glycine uptake in cells over-expressing hGlyT1a. 了解更多 -
Dasotraline hydrochloride
Catalog No. A21684 triple reuptake inhibitorDasotraline hydrochloride (SEP-225289 hydrochloride) is a triple reuptake inhibitor that blocks dopamine, norepinephrine, and serotonin transporters with IC50 values of 4, 6, and 11 nM, respectively. 了解更多 -
Dasotraline
Catalog No. A21618 triple reuptake inhibitorDasotraline is a triple reuptake inhibitor that blocks dopamine, norepinephrine, and serotonin transporters with IC50 values of 4, 6, and 11 nM, respectively. 了解更多 -
Escitalopram
Catalog No. A21241 selective serotonin reuptake inhibitor (SSRI)Escitalopram is a selective serotonin reuptake inhibitor (SSRI) with Ki of 0.89 nM. 了解更多 -
Diclofensine hydrochloride
Catalog No. A20923 monoamine reuptake inhibitorDiclofensine hydrochloride (Ro-8-4650 hydrochloride) is a potent inhibitor of monoamine reuptake, blocking the uptake of dopamine, noradrenaline, and serotonin by rat brain synaptosomes with IC50 values of 0.74, 2.3, and 3.7 nM, respectively. 了解更多 -
VU 0240551
Catalog No. A20854 KCC2 inhibitorVU 0240551 is a small molecule inhibitor of the neuronal K-Cl cotransporter, KCC2 (IC50 = 560 nM for K+ uptake assay in KCC2-overexpressing cells). 了解更多 -
Escitalopram oxalate
Catalog No. A16533 Serotonin reuptake inhibitorEscitalopram oxalate ((S)-(+)Citalopram oxalate) is a selective serotonin reuptake inhibitor (SSRI) with Ki of 0.89 nM. 了解更多 -
DMT1 blocker 2
Catalog No. A18999 DMT1 inhibitorDMT1 blocker 2, Compound 12f, is a direct inhibitor of divalent metal transporter 1 (DMT1) with an IC50 of 0.83 μM, is expected to block iron uptake by enterocytes in vivo. 了解更多 -
Amezinium methylsulfate
Catalog No. A18103 norepinephrine reuptake inhibitorAmezinium Metilsulfate, also known as Regulton and LU-1631, is a norepinephrine reuptake inhibitor which exclusively affects postganglionic sympathetic neurons. Amezinium Metilsulfate is used to treat hypotension. 了解更多 -
Paroxetine mesylate
Catalog No. A17566 serotonin uptake inhibitorParoxetine Mesylate is a serotonin uptake inhibitor that is effective in the treatment of depression. 了解更多 -
Takinib
Catalog No. A16960 -
Tiagabine hydrochloride
Catalog No. A16135 -
Desvenlafaxine succinate hydrate
Catalog No. A15491 serotonin (5-HT)/norepinephrine (NE) reuptake 抑制剂Desvenlafaxine succinate hydrate是一种新型5-羟色胺(5-HT)转运蛋白 和去甲肾上腺素(NE)转运蛋白重吸收抑制剂，Ki值分别为40.2 nM和558.4 nM 了解更多 -
Azaphen dihydrochloride monohydrate
Catalog No. A15009 -
Phenylpiracetam
Catalog No. A15211 -
NG25
Catalog No. A15185 -
Bitopertin (R enantiomer)
Catalog No. A15022
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