Epigenetics
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I-BRD9
Catalog No. A15872 -
(E)-ZL0420
Catalog No. A20136 BRD4 inhibitorZL0420 is a potent and selective bromodomain-containing protein 4 (BRD4) inhibitor with IC50 values of 27 nM against BRD4 BD1 and 32 nM against BRD4 BD2. 了解更多 -
BMS-986158
Catalog No. A19442 Bromodomain inhibitorBMS-986158 is an inhibitor of the bromodomain and extra-terminal (BET) proteins. 了解更多 -
Bromodomain IN-1
Catalog No. A18845 Bromodomain inhibitorBromodomain IN-1 is a Bromodomain inhibitor extracted from patent WO2016069578A1, compound 4 . 了解更多 -
BRD4 Inhibitor-10
Catalog No. A18679 BRD4-BD1 inhibitorBRD4 Inhibitor-10 is a potent BRD4-BD1 inhibitor extracted from patent WO2015022332A1, Compound II-25, has an IC50 of 8 nM. 了解更多 -
(Rac)-BAY1238097
Catalog No. A21598 BET inhibitor(Rac)-BAY1238097 is a BET inhibitor, with an IC50 of 1.02 μM for BRD4. Used in cancer research. 了解更多 -
INCB054329 Racemate
Catalog No. A21609 -
CPI-0610 carboxylic acid
Catalog No. A21714 BET inhibitorCPI-0610 carboxylic acid is a potent bromodomain and extra-terminal (BET) protein inhibitor. CPI-0610 carboxylic acid has the potential in the therapy of multiple myeloma. 了解更多 -
AZD5153 6-Hydroxy-2-naphthoic acid
Catalog No. A21852 BET/BRD4 bromodomain inhibitorAZD5153 6-Hydroxy-2-naphthoic acid is the 6-Hydroxy-2-naphthoic acid of AZD5153. AZD5153 is a potent, selective, and orally available BET/BRD4 bromodomain inhibitor; disrupts BRD4 with an IC50 of 1.7 nM. 了解更多 -
Molibresib besylate
Catalog No. A21855 BET bromodomain inhibitorMolibresib besylate (GSK 525762C; I-BET 762 besylate) is a BET bromodomain inhibitor with IC50 of 32.5-42.5 nM. 了解更多 -
Fisetin (Fustel)
Catalog No. A10388 Fisetin (Fustel)是有效的Sirtuin活化化合物(STAC),可以调节Sirtuin。 了解更多 -
OSS-128167
Catalog No. A17048 -
Thiomyristoyl
Catalog No. A17166 -
PROTAC Sirt2 Degrader-1
Catalog No. A20005 Sirt2 degraderPROTAC Sirt2 Degrader-1 is a SirReal-based PROTAC, acts as a Sirt2 degrader, composed of a highly potent and isotype-selective Sirt2 inhibitor, a linker, and a bona fide cereblon ligand for E3 ubiquitin ligase. 了解更多 -
SRT 1720 Hydrochloride
Catalog No. A21143 SIRT1 activator ofSRT 1720 Hydrochloride is a selective activator of SIRT1 with an EC50 of 0.10 μM, and shows less potent activities on SIRT2 and SIRT3. 了解更多 -
Sirt2-IN-1
Catalog No. A19348 Sirt2 inhibitorSirt2-IN-1 (Compound 9) is a sirtuin 2 (Sirt2) inhibitor with an IC50 of 163 nM. 了解更多 -
JFD00244
Catalog No. A19517 -
SIRT5 inhibitor 1
Catalog No. A19841 SIRT5 inhibitorSIRT5 inhibitor 1 is a potent Human Sirtuin 5 deacylase inhibitor, with an IC50 of 0.11 μM. 了解更多 -
SirReal1-O-propargyl
Catalog No. A20091 Sirt2 inhibitorSirReal1-O-propargyl is a selective and highly potent Sirtuin 2 (Sirt2) inhibitor, with an IC50 of 2.4 μM. 了解更多 -
SRT1720 HCl
Catalog No. A10862 SIRT1 ActivatorSRT1720 HCl是一种抑制剂,旨在作为瑟土因亚型SIRT1的小分子活化剂。 了解更多 -
EX 527 (Selisistat)
Catalog No. A10377 SIRT1 抑制剂EX 527 (Selisistat)是一种有效的选择性SIRT1 III类组蛋白脱乙酰基酶抑制剂,在无细胞分析中的IC50为38 nM。 了解更多 -
SRT2104 (GSK2245840)
Catalog No. A14188 SIRT1 activatorSRT2104 (GSK2245840)是一种选择性sirt1激活剂,参与能量稳态的调节。 了解更多