你的浏览器似乎禁用了 JavaScript。
您必须在浏览器中启用JavaScript才能使用本网站的功能。

微信关注
申请试用装

主页 /
Products On Sale

Products On Sale

Quick View
Flupirtine maleate

Catalog No. A10251
Quick View

添加到收藏
NMDA 拮抗剂

Flupirtine maleate是Flupirine的盐形式，是一种非阿片类中枢性镇痛药，是一种选择性的神经元钾离子通道开放剂，也具有NMDA受体拮抗剂特性。了解更多

Bulk Inquiry Free Sample
Quick View
Tamoxifen Citrate

Catalog No. A10885
Quick View

添加到收藏
Estrogen receptor 拮抗剂

Tamoxifen Citrate是哺乳动物甾醇异构酶的选择性和有效抑制剂。了解更多

Product Citations (4)

Bulk Inquiry Free Sample
- Renu Sudhakar, .et al. Bazedoxifene, a Postmenopausal Drug, Acts as an Antimalarial and Inhibits Hemozoin Formation, Microbiol Spectr, 2022, Jun 29;10(3) PMID: 35616371
- Takashi Azuma, .et al. Removal of pharmaceuticals in water by introduction of ozonated microbubbles, SEP PURIF TECHNOL, 2019, Apr; 212: 483-489
- Azuma T, .et al. Distribution of six anticancer drugs and a variety of other pharmaceuticals, and their sorption onto sediments, in an urban Japanese river, Environ Sci Pollut Res Int, 2017, Aug;24(23):19021-19030 PMID: 28660504
- Azuma T, .et al. Detection of pharmaceuticals and phytochemicals together with their metabolites in hospital effluents in Japan, and their contribution to sewage treatment plant influents, Sci Total Environ, 2016, Apr 1;548-549:189-197 PMID: 26802347
Quick View
Paliperidone

Catalog No. A10691
Quick View

添加到收藏
Dopamine Receptor 拮抗剂

Paliperidone (Invega)是一种非典型的抗精神病药。了解更多

Product Citations (1)

Bulk Inquiry Free Sample
- Reiko Watanabe, .et al. Development of an In Silico Prediction Model for P-glycoprotein Efflux Potential in Brain Capillary Endothelial Cells toward the Prediction of Brain Penetration, J Med Chem, 2021, Mar 11;64(5):2725-2738 PMID: 33619967
Quick View
JNJ-31020028

Catalog No. A14332
Quick View

添加到收藏
neuropeptide Y Y2 receptor 拮抗剂

JNJ-31020028是一种新型的选择性脑渗透神经肽Y Y2受体拮抗剂。了解更多

Bulk Inquiry Free Sample
Quick View
Bicalutamide (Casodex)

Catalog No. A10142
Quick View

添加到收藏
Androgen Receptor 拮抗剂

Bicalutamide (Casodex)是一种口服非甾体抗雄激素，用于治疗前列腺癌和多毛症。了解更多

Product Citations (5)

Bulk Inquiry Free Sample
- Mi Chen, .et al. TRIM33 drives prostate tumor growth by stabilizing androgen receptor from Skp2-mediated degradation, EMBO Rep, 2022, Aug 3;23(8):e53468 PMID: 35785414
- Takashi Azuma, .et al. Removal of pharmaceuticals in water by introduction of ozonated microbubbles, SEP PURIF TECHNOL, 2019, Apr; 212: 483-489
- Anowara Khatun, .et al. Transcriptional Repression and Protein Degradation of the Ca2+-Activated K+ Channel KCa1.1 by Androgen Receptor Inhibition in Human Breast Cancer Cells, Front Physiol, 2018, 9: 312 PMID: 29713287
- Azuma T, .et al. Distribution of six anticancer drugs and a variety of other pharmaceuticals, and their sorption onto sediments, in an urban Japanese river, Environ Sci Pollut Res Int, 2017, Aug;24(23):19021-19030 PMID: 28660504
- Azuma T, .et al. Detection of pharmaceuticals and phytochemicals together with their metabolites in hospital effluents in Japan, and their contribution to sewage treatment plant influents, Sci Total Environ, 2016, Apr 1;548-549:189-197 PMID: 26802347
Quick View
Ki16425

Catalog No. A10501
Quick View

添加到收藏
LPA Receptor 拮抗剂

ki16425是对LPA1和LPA3具有选择性的LPA受体拮抗剂，对人LPA1、LPA2和LPA3受体分别显示Ki值为0.34、6.5和0.93 μM。了解更多

Product Citations (5)

Bulk Inquiry Free Sample
- Maria F Fernandes, .et al. Glucagon-like Peptide-1 Secretion Is Inhibited by Lysophosphatidic Acid, Int J Mol Sci, 2022, Apr 9;23(8):4163 PMID: 35456981
- Rieko Suenaga, .et al. Lateral access mechanism of LPA receptor probed by molecular dynamics simulation, PLoS One, 2022, Feb 3;17(2):e0263296 PMID: 35113924
- Inoue A, .et al. Illuminating G-Protein-Coupling Selectivity of GPCRs, Cell, 2019, Jun 13;177(7):1933-1947 PMID: 31160049
- Taniguchi R, .et al. Structural insights into ligand recognition by the lysophosphatidic acid receptor LPA6, Nature, 2017, Aug 17;548(7667):356-360 PMID: 28792932
- T. HASHIMOTO, .et al. Generalized pruritus in primary sclerosing cholangitis: implications of histamine release by lysophosphatidic acid., Br J Dermatol., 2015, Nov;173(5):1334-6 PMID: 26122943
Quick View
Memantine hydrochloride

Catalog No. A11708
Quick View

添加到收藏
NMDA receptor 拮抗剂

Memantine hydrochloride是nmda受体的拮抗剂，与离子通道位点结合。它还是CYP2B6和CYP2D6抑制剂，作用于重组CYP2B6和CYP2D6，Ki分别为0.51 nM和94.9 μM。它被用于治疗帕金森综合征。了解更多

Bulk Inquiry Free Sample
Quick View
Reversine

Catalog No. A13250
Quick View

添加到收藏
human A3 adenosine receptor 拮抗剂 /Aurora 抑制剂

Reversine是一种有效的人A3腺苷受体拮抗剂，Ki为0.66μM，是一种泛光A/B/C激酶抑制剂，IC50分别为12 nM/13 nM/20 nM。也用于干细胞去分化。了解更多

Product Citations (1)

Bulk Inquiry Free Sample
- Hazheen K, .et al. BuGZ facilitates loading of spindle assembly checkpoint proteins to kinetochores in early mitosis, J Biol Chem, 2020, August 20
Quick View
Otenabant

Catalog No. A15200
Quick View

添加到收藏
CB1 receptor 拮抗剂

Otenabant是最近发现的选择性，高亲和力，竞争性CB1受体拮抗剂，Ki为0.7 nM。了解更多

Bulk Inquiry Free Sample
Quick View
Cyproterone acetate

Catalog No. A11409
Quick View

添加到收藏
Androgen Receptor 拮抗剂

Cyproterone acetate是17-羟孕酮的合成衍生物，可作为雄激素受体拮抗剂以及具有弱孕激素和糖皮质激素活性的弱孕激素受体激动剂。了解更多

Bulk Inquiry Free Sample
Quick View
AMD 3465 Hexahydrobromide

Catalog No. A11953
Quick View

添加到收藏
CXCR4 拮抗剂

AMD 3465 Hexahydrobromide是一种有效的选择性CXCR4拮抗剂。了解更多

Product Citations (1)

Bulk Inquiry Free Sample
- Kentaro Suzuki, .et al. C-terminal-modifed LY2510924: a versatile scafold for targeting C-X-C chemokine receptor type 4, Sci Rep, 2019, 9: 15284
Quick View
MDL 29951

Catalog No. A13729
Quick View

添加到收藏
NMDA receptor 拮抗剂

MDL-29951是在体外和体内均能激活NMDA受体的新型甘氨酸拮抗剂（Ki = 0.14 mM，[3H]甘氨酸结合）。了解更多

Bulk Inquiry Free Sample
Quick View
Endoxifen

Catalog No. A12639
Quick View

添加到收藏
Estrogen receptor 拮抗剂

Endoxifen是他莫昔芬的次生代谢产物。它是负责他莫昔芬在ER阳性乳腺癌中有效性的主要代谢物。Endoxifen Z-isomer抑制hERG, 这种作用具有浓度依赖性, IC50值为1.6μM。了解更多

Product Citations (2)

Bulk Inquiry Free Sample
- Marina Arino Martin, .et al. Photolytic fate of (E)- and (Z)-endoxifen in water and treated wastewater exposed to sunlight, Environ Res, 2021, Apr 3;197:111121 PMID: 33823193
- Martin MA, .et al. Photodegradation of (E)- and (Z)-Endoxifen in water by ultraviolet light: Efficiency, kinetics, by-products, and toxicity assessment, Water Res, 2019, Dec 29;171:115451 PMID: 31901682
Quick View
Nutlin-3

Catalog No. A10657
Quick View

添加到收藏
Mdm2 拮抗剂

Nutlin-3是一种有效的，选择性Mdm2(它自身和p53的环指依赖性泛素蛋白连接酶)拮抗剂，是有效的凋亡诱导剂。了解更多

Product Citations (4)

Bulk Inquiry
- Maxime Parisotto, .et al. PTEN deletion in luminal cells of mature prostate induces replication stress and senescence in vivo, J Exp Med, 2018, Jun 4; 215(6): 1749-1763 PMID: 29743291
- Ohmuro-Matsuyama Y, .et al. Evaluation of protein-ligand interactions using the luminescent interaction assay FlimPIA with streptavidin-biotin linkage, Anal Biochem, 2018, Dec 15;563:61-66 PMID: 30316750
- Alisa A. Garaeva, .et al. Mitochondrial dysfunction induces SESN2 gene expression through Activating Transcription Factor 4, Cell Cycle, 2016, 15(1): 64-71 PMID: 26771712
- A G Evstafieva, .et al. A sustained deficiency of mitochondrial respiratory complex III induces an apoptotic cell death through the p53-mediated inhibition of pro-survival activities of the activating transcription factor 4, Cell Death Dis., 2014, 5(11): e1511. PMID: 25375376
Quick View
MK-0517 (Fosaprepitant)

Catalog No. A11756
Quick View

添加到收藏
neurokinin-1 receptor 拮抗剂

MK-0517 (Fosaprepitant,L-758,298)是Aprepitant的水溶性磷酰基前药，它是NK1拮抗剂。了解更多

Bulk Inquiry Free Sample
Quick View
S1RA (E-52862)

Catalog No. A12504
Quick View

添加到收藏
sigma-1 receptor 拮抗剂

S1RA是一种选择性sigma-1受体拮抗剂，据报道其结合亲和力为Ki = 17.0±7.0 nM，对sigma-2受体具有选择性，并且对其他170种受体，酶，转运蛋白和离子通道具有选择性。了解更多

Bulk Inquiry Free Sample
Quick View
AZD1283

Catalog No. A15443
Quick View

添加到收藏
P2Y12 receptor 拮抗剂

AZD1283是P2Y12受体的有效拮抗剂，EC50为3.0 ug/kg/min，TI> 10；结合IC50为11 nM。了解更多

Bulk Inquiry
Quick View
Biperiden HCl

Catalog No. A10147
Quick View

添加到收藏
Muscarinic receptor antagonist

Biperiden HCl是毒蕈碱受体拮抗剂，对M1亚型表现出一定的选择性。了解更多

Bulk Inquiry Free Sample
Quick View
MK-4305 (Suvorexant)

Catalog No. A11500
Quick View

添加到收藏
OX receptor 拮抗剂

Suvorexant (MK-4305)是OX1R和OX2R的有效，选择性和口服可生物利用的拮抗剂，目前正在临床研究中作为失眠的新疗法。了解更多

Product Citations (9)

Bulk Inquiry Free Sample
- Richard L Spinieli, .et al. Orexin contributes to eupnea within a critical period of postnatal development, Am J Physiol Regul Integr Comp Physiol, 2021, Oct 1;321(4):R558-R571 PMID: 34405704
- Jacob W Clark, .et al. Manipulation of REM sleep via orexin and GABAA receptor modulators differentially affects fear extinction in mice: effect of stable versus disrupted circadian rhythm, Sleep, 2021, Mar 15;zsab068 PMID: 33720375
- Zhang B, .et al. Hypothalamic orexin and mechanistic target of rapamycin activation mediate sleep dysfunction in a mouse model of tuberous sclerosis complex, Neurobiol Dis, 2019, Oct 9;134:104615 PMID: 31605778
- Obara K, .et al. Assessment of Inhibitory Effects of Hypnotics on Acetylcholine-Induced Contractions in Isolated Rat Urinary Bladder Smooth Muscle, Biol Pharm Bull, 2019, 42(2):280-288 PMID: 30713259
- James B Jaggard, .et al. Hypocretin underlies the evolution of sleep loss in the Mexican cavefish, eLife, 2018, 7: e32637 PMID: 29405117
- Skillman B, .et al. Quantification of suvorexant in blood using liquid chromatography-quadrupole/time of flight (LC-Q/TOF) mass spectrometry, J Chromatogr B Analyt Technol Biomed Life Sci, 2018, Aug 1;1091:87-95 PMID: 29859493
- Clark L, .et al. On the use of Pichia pastoris for isotopic labeling of human GPCRs for NMR studies, J Biomol NMR, 2018, Aug;71(4):203-211 PMID: 30121871
- Sullinger S, .et al. Identification of Suvorexant in Urine Using Liquid Chromatography-Quadrupole/Time-of-Flight Mass Spectrometry (LC-Q/TOF-MS), J Anal Toxicol, 2017, Apr 1;41(3):224-229 PMID: 28035034
- Carson M, .et al. Quantification of suvorexant in urine using gas chromatography/mass spectrometry, J Chromatogr B Analyt Technol Biomed Life Sci, 2017, Jan 1;1040:289-294 PMID: 27825624
Quick View
XCT 790

Catalog No. A13299
Quick View

添加到收藏
ERRα 拮抗剂/inverse 激动剂

XCT 790是ERRα的强效特异性反向激动剂。了解更多

Bulk Inquiry
Quick View
A-804598

Catalog No. A16066
Quick View

添加到收藏
P2X7 receptor 拮抗剂

A-804598是一种P2X7选择性竞争性拮抗剂，对人，大鼠和小鼠通道的IC50值分别为11、10和9 nM。了解更多

Bulk Inquiry Free Sample
Quick View
Alvimopan (ADL 8-2698)

Catalog No. A11292
Quick View

添加到收藏
Opioid 拮抗剂

Alvimopan (ADL 8-2698)表现为外周作用的opioid拮抗剂，Alvimopan竞争性结合胃肠道中的mu-opioid receptor。了解更多

Bulk Inquiry Free Sample
Quick View
Birinapant (TL32711)

Catalog No. A12738
Quick View

添加到收藏
XIAP/cIAP1 拮抗剂

Birinapant (TL32711)是第二个线粒体衍生的胱天蛋白酶（SMAC）激活剂和IAP（凋亡蛋白抑制剂）家族蛋白抑制剂的合成小分子和肽类似物，对cIAP1最有效，无细胞试验中Kd为<1 nM，具有潜在的抗肿瘤活性。了解更多

Bulk Inquiry Free Sample
Quick View
SB-742457

Catalog No. A14092
Quick View

添加到收藏
5-HT6 receptor 拮抗剂

SB-742457是一种选择性的5-HT6受体拮抗剂，具有认知，记忆和增强学习的作用。了解更多

Bulk Inquiry Free Sample
Quick View
Alosetron

Catalog No. A11310
Quick View

添加到收藏
5-HT3 拮抗剂

Alosetron是一种5-HT3拮抗剂，对胃肠道肠道神经系统的5-HT3受体具有拮抗作用。了解更多

Bulk Inquiry Free Sample
Quick View
GSK 0660

Catalog No. A12392
Quick View

添加到收藏
PPARδ 拮抗剂

GSK 0660是一种选择性PPARβ拮抗剂（在PPARβ，PPARα和PPARγ处，IC50值分别为0.155，> 10和≥10 ?M）。了解更多

Bulk Inquiry Free Sample
Quick View
AM966

Catalog No. A13982
Quick View

添加到收藏
LPA1 receptor 拮抗剂

AM966是LPA1受体（溶血磷脂酸受体）的高亲和力，选择性口服拮抗剂，IC50值为17 nM。了解更多

Product Citations (1)

Bulk Inquiry Free Sample
- Maria F Fernandes, .et al. Glucagon-like Peptide-1 Secretion Is Inhibited by Lysophosphatidic Acid, Int J Mol Sci, 2022, Apr 9;23(8):4163 PMID: 35456981
Quick View
MDV3100

Catalog No. A10562
Quick View

添加到收藏
Androgen receptor 拮抗剂

MDV3100(Enzalutamide)是一种androgen-receptor (AR)拮抗剂。在AR研究中强烈推荐的抑制剂。了解更多

Product Citations (3)

Bulk Inquiry Free Sample
- Shiv Verma, .et al. Increased cytokine gene expression and cognition risk associated with androgen deprivation therapy, Prostate, 2022, Oct;82(14):1389-1399 PMID: 35821621
- Mi Chen, .et al. TRIM33 drives prostate tumor growth by stabilizing androgen receptor from Skp2-mediated degradation, EMBO Rep, 2022, Aug 3;23(8):e53468 PMID: 35785414
- Prem P Kushwaha, .et al. Role of solute carrier transporters SLC25A17 and SLC27A6 in acquired resistance to enzalutamide in castration-resistant prostate cancer, Mol Carcinog, 2021, Dec 22 PMID: 34939235
Quick View
SB269970 HCl

Catalog No. A11925
Quick View

添加到收藏
5-HT7 receptor 拮抗剂

SB269970 HCl是有效的选择性5-HT7受体拮抗剂。了解更多

Bulk Inquiry Free Sample
Quick View
ICI 118,551 hydrochloride

Catalog No. A13225
Quick View

添加到收藏
β2 adrenergic 拮抗剂

ICI 118,551 hydrochloride是选择性的β2 adrenergic receptor 拮抗剂,结合 β2，β1 和 β3 肾上腺素能受体的Ki 值分别为 0.7，49.5 和 611 nM。了解更多

Bulk Inquiry Free Sample
Quick View
(-)-MK 801 maleate

Catalog No. A13435
Quick View

添加到收藏
NMDA receptor 拮抗剂.

(-)-MK 801 maleate是一种有效的、选择性的、非竞争性的NMDA受体拮抗剂。它通过与NMDA相关离子通道内的一个位点结合而起作用。了解更多

Bulk Inquiry Free Sample
Quick View
LY2940680 (Taladegib)

Catalog No. A11048
Quick View

添加到收藏
SMO 拮抗剂

LY2940680 (Taladegib)已显示可影响由Hedgehog（Hh）蛋白引发的癌细胞信号通路。了解更多

Bulk Inquiry Free Sample
Quick View
SB-705498

Catalog No. A11143
Quick View

添加到收藏
TRPV1 拮抗剂

SB-705498是有效，选择性和口服生物利用的TRPV1拮抗剂，抑制TRPV1的Capsaicin，酸和热激活，IC50分别为3 nM， 0.1 nM和6 nM，该作用具有一定的电压依赖性，作用于TRPV1比作用于TRPM8选择性高100倍以上。了解更多

Bulk Inquiry Free Sample
Quick View
Buflomedil HCl

Catalog No. A11737
Quick View

添加到收藏
VEGFR 拮抗剂

Buflomedil HCl是一种用于治疗外周血管疾病的血管活性剂。了解更多

Bulk Inquiry Free Sample
Quick View
AR7

Catalog No. A12905
Quick View

添加到收藏
RARα 拮抗剂.

AR7是视黄酸受体α(RARα)拮抗剂。了解更多

Bulk Inquiry
Quick View
WAY-100635 maleate salt

Catalog No. A15282
Quick View

添加到收藏
5HT1A 拮抗剂

WAY-100635 maleate salt是一种有效的、选择性的5-羟色胺1A拮抗剂，对5-HT的IC50为0.95-0.12 nM。了解更多

Bulk Inquiry
Quick View
5-hydroxymethyl tolterodine (PNU 200577)

Catalog No. A11166
Quick View

添加到收藏
muscarinic receptor 拮抗剂

5-hydroxymethyl tolterodine (PNU 200577)是托特罗定的代谢产物，tolterodine是一种用于治疗尿失禁的毒蕈碱受体拮抗剂。了解更多

Bulk Inquiry Free Sample
Quick View
Dyphylline

Catalog No. A10339
Quick View

添加到收藏
Adenosine receptor 拮抗剂

Dyphylline是黄嘌呤衍生物，具有支气管扩张药和血管扩张药的作用。它充当腺苷受体拮抗剂和磷酸二酯酶抑制剂。了解更多

Bulk Inquiry Free Sample
Quick View
SIB 1757

Catalog No. A13758
Quick View

添加到收藏
mGluR 拮抗剂

SIB 1757是mGlu5代谢型谷氨酸受体亚型的高度选择性拮抗剂。了解更多

Bulk Inquiry Free Sample
Quick View
(+)-MK 801 Maleate

Catalog No. A12761
Quick View

添加到收藏
NMDA receptor 拮抗剂

(+)-MK 801 Maleate是NMDA的有效拮抗剂，Ki值为30.5nM。了解更多

Bulk Inquiry Free Sample
Quick View
Ginkgolide B

Catalog No. A10429
Quick View

添加到收藏
PAFR 拮抗剂

Ginkgolide B (BN 52021)是一种PAFR拮抗剂，IC50为3.6 μM。了解更多

Bulk Inquiry Free Sample
Quick View
Granisetron Hydrochloride

Catalog No. A10437
Quick View

添加到收藏
5-HT3 receptor 拮抗剂

Granisetron Hydrochloride是血清素5-ht3受体拮抗剂。了解更多

Bulk Inquiry Free Sample
Quick View
JNJ7777120

Catalog No. A12713
Quick View

添加到收藏
Histamine 拮抗剂

JNJ7777120是有效的，选择性的非咪唑histamine H4 receptor拮抗剂。了解更多

Product Citations (2)

Bulk Inquiry Free Sample
- K Yamamoto, .et al. Activation of orexinergic and histaminergic pathway involved in therapeutic effect of histamine H4 receptor antagonist against cisplatin-induced anorexia in mice, Naunyn-Schmiedeberg's Arch Pharmacol, 2019, pp 1-12
- Yamamoto K, .et al. Effects of a histamine H4 receptor antagonist on cisplatin-induced anorexia in mice, Neurosci Lett, 2018, May 29;676:103-107 PMID: 29655943
Quick View
Flutamide

Catalog No. A10402
Quick View

添加到收藏
Androgen receptor 拮抗剂

Flutamide是一种抗雄激素药物，其活性代谢洛丽塔与Ki值为55nM的雄激素受体结合，可作用于前列腺癌。了解更多

Bulk Inquiry Free Sample
Quick View
Solifenacin succinate

Catalog No. A11215
Quick View

添加到收藏
muscarinic M3 receptor antagoinst

Solifenacin succinate是毒蕈碱M3受体拮抗剂，用于治疗尿失禁。了解更多

Bulk Inquiry Free Sample
Quick View
SB-408124

Catalog No. A11567
Quick View

添加到收藏
OX Receptor 拮抗剂

SB-408124是一种选择性的非肽orexin OX1受体拮抗剂(人OX1和OX2受体的Kb值分别为21.7和1405 nM)。体内口服后阻断orexin-A诱导的修饰。了解更多

Bulk Inquiry Free Sample
Quick View
RU 58841

Catalog No. A11541
Quick View

添加到收藏
AR 拮抗剂

RU 58841，也称为PSK-3841或HMR-3841，是一种非甾体类抗雄激素药物。了解更多

Bulk Inquiry
Quick View
SYN-115 (Tozadenant)

Catalog No. A11560
Quick View

添加到收藏
A2a receptor 拮抗剂

SYN115是口服，有效和选择性的腺苷2a（A2a）受体抑制剂，作用于人类和恒河猴的 adenosine A2A 受体，Ki 值分别为 11.5 nM 和 6 nM。了解更多

Bulk Inquiry Free Sample
Quick View
Firategrast (SB 683699)

Catalog No. A12787
Quick View

添加到收藏
α4β1/α4β7 integrin 拮抗剂

Firategrast (SB 683699)是一种口服可生物利用的alpha4 beta1/alpha4 beta7整联蛋白拮抗剂，旨在减少淋巴细胞向中枢神经系统（CNS）的运输。了解更多

Product Citations (1)

Bulk Inquiry Free Sample
- Higuchi S, .et al. Inhibition of the integrin signal constitutes a mouse iPS cell niche, Dev Growth Differ, 2016, Sep;58(7):586-99 PMID: 27633818
Quick View
SB225002

Catalog No. A14209
Quick View

添加到收藏
CXCR2 拮抗剂

SB225002是一种有效的选择性CXCR2拮抗剂，IC50为22 nM，可抑制白介素IL-8与CXCR2的结合，选择性是其他测试的7-TMR的150倍以上。了解更多

Bulk Inquiry

联系我们

Not your Region? View all Distributors

溶液配制计算器

分子量计算器

稀释计算器

摩尔浓度计算器

ADOOQ 产品质量保证

Guaranteed product quality, 365 days Unconditional Return & Replacement

We promise all products to perform as described.