“betaine hydrochloride”的搜索结果

产品 1 到 50 共 54个

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  1. Tamsulosin hydrochloride

    Catalog No. A14936
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    α1 receptor 拮抗剂
    Tamsulosin hydrochloride是一种选择性的α1受体拮抗剂,是用于良性前列腺增生的药物。 了解更多
  2. Atrasentan HCl

    Catalog No. A15007
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    Endothelin 拮抗剂 receptor
    Atrasentan hydrochloride是一种开发用于治疗前列腺癌的内皮素拮抗剂受体(IC50 = 0.0551 nM,ETA)。 了解更多
  3. SCH 23390 HCl

    Catalog No. A13066
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    D1/D5 receptor 拮抗剂
    SCH 23390 HCl是一种有效的多巴胺受体拮抗剂(D1和D5受体亚型的Ki值分别为0.2 nM和0.3 nM)。 了解更多
  4. Azasetron HCl

    Catalog No. A16417
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    5-HT3 receptor 拮抗剂
    Azasetron HCl是一种选择性的5-HT3受体拮抗剂,IC50为0.33 nM,用于治疗癌症化学疗法引起的恶心和呕吐。 了解更多
  5. Melitracen hydrochloride

    Catalog No. A17494
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    dopamine D1/2 receptor antagonist
    Melitracen HCl ia potential dopamine D1/2 receptor antagonist used to treat depression. It is often co-administered with flupenthixol as a treatment for trigeminal neuralgia. It does not effect cardiovascular function. 了解更多
  6. MK 3207 HCl

    Catalog No. A10598
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    CGRP Receptor 拮抗剂
    MK 3207 hydrochloride是一种有效的CGRP受体拮抗剂,IC50为0.12 nM。 了解更多
  7. CP 945598 HCl (Otenabant HCl)

    Catalog No. A11942
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    CB1 拮抗剂
    CP 945598 HCl (Otenabant HCl)是一种有效且高度选择性的CB1拮抗剂。 了解更多
  8. Clemizole hydrochloride

    Catalog No. A15047
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    H1 histamine receptor 拮抗剂
    Clemizole hydrochloride是H1组胺受体的拮抗剂,对NS4B RNA结合的IC50值为8 mM。 了解更多
  9. MTEP hydrochloride

    Catalog No. A15174
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    mGlu5 拮抗剂
    MTEP hydrochloride是一种有效的,选择性和非竞争性的mGlu5拮抗剂,IC50和Ki分别为5 nM和16 nM。 了解更多
  10. SB-408124 HCl

    Catalog No. A15231
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    OX Receptor 拮抗剂
    SB408124 Hydrochloride是OX1受体的非肽拮抗剂,全细胞和膜的Ki分别为57 nM和27 nM。表现出比OX2受体高50倍的选择性。 了解更多
  11. Alosetron Hydrochloride

    Catalog No. A14989
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    5HT3-receptor 拮抗剂
    Alosetron Hydrochloride是一种5-羟色胺5HT3受体拮抗剂,可用于治疗肠易激综合症。 了解更多
  12. Cyproheptadine hydrochloride

    Catalog No. A16169
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    serotonin/histamine2 拮抗剂
    Cyproheptadine hydrochloride是抗组胺药,是5-羟色胺和组胺的拮抗剂。 了解更多
  13. Chlorcyclizine hydrochloride

    Catalog No. A18025
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    histamine H1 antagonist
    Chlorcyclizine hydrochloride is a histamine H1 antagonist. 了解更多
  14. Haloperidol hydrochloride

    Catalog No. A18304
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    dopamine D2 receptor antagonist
    Haloperidol hydrochloride is a potent dopamine D2 receptor antagonist, widely used as an antipsychotic. 了解更多
  15. MPEP HCl

    Catalog No. A13236
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    mGlu5 receptor 拮抗剂
    MPEP HCl是对mGlu5a受体亚型(IC50 = 36 nM)的有效,高度选择性的非竞争性拮抗剂,但在浓度高达30 uM的mGlu1b受体上无激动剂或拮抗剂活性。 了解更多
  16. BRL-15572 dihydrochloride

    Catalog No. A11178
    5-HT1D receptor 拮抗剂
    BRL-15572是一种选择性的h5-HT1D拮抗剂,相对于h5-HT1B表现出60倍的选择性,对一系列其他受体类型的亲和力很小或没有亲和力。 了解更多
  17. Naftopidil 2HCl

    Catalog No. A10619
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    5-HT1A and α1-adrenergic receptor 拮抗剂
    Naftopidil 2HCl是选择性5-HT1A和α1-肾上腺素能受体拮抗剂,IC50分别为0.1μM和0.2μM。 了解更多
  18. cis-(Z)-Flupentixol dihydrochloride

    Catalog No. A12347
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    Dopamine receptor 拮抗剂
    cis-(Z)-Flupentixol dihydrochloride是多巴胺受体拮抗剂、抗精神病药物、抗精神病药物。 了解更多
  19. SB 399885 HCl

    Catalog No. A14102
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    5-HT6 拮抗剂
    SB 399885 hydrochloride是一种有效的,脑渗透剂和口服活性的SR-6拮抗剂。它对SR-6的选择性比其他血清素受体高200倍(对于人类重组,天然大鼠和天然人类SR-6受体,pKi值分别为9.11、8.81和9.02)。 了解更多
  20. Atipamezole HCl

    Catalog No. A13902
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    α2 adrenergic receptor 拮抗剂
    Atipamezole hydrochloride是一种选择性α2肾上腺素受体拮抗剂(α2A、α2B、α2C、α1A和α1B受体的Ki值分别为1.1、1.0、0.89、1300和6500nm)。已经被证明是大脑的渗透剂。 了解更多
  21. SB 258585 HCl

    Catalog No. A14026
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    5-HT6 serotonin receptor 拮抗剂
    SB 258585 hydrochloride是一种选择性和有效的SR-6拮抗剂。该化合物显示出比其他5-羟色胺受体亚型高160倍的选择性。 了解更多
  22. Bavisant dihydrochloride

    Catalog No. A15015
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    H3 receptor 拮抗剂
    Bavisant dihydrochloride是一种人类H3受体的高选择性,口服活性拮抗剂。 了解更多
  23. Bavisant dihydrochloride hydrate

    Catalog No. A15016
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    H3 receptor 拮抗剂
    Bavisant dihydrochloride hydrate是人类H3受体的高度选择性口服活性拮抗剂。 了解更多
  24. Levocetirizine Dihydrochloride

    Catalog No. A17440
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    L-isomer of cetirizine and histamine H1 receptor antagonist
    Levocetirizine dihydrochloride is a L-isomer of cetirizine and histamine H1 receptor antagonist. It incrases levels of CD4+ CD25+ T cells and decreases levels of eosinophils, decreasing allergy symptoms. 了解更多
  25. SB-277011 dihydrochloride

    Catalog No. A21353
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    dopamine D3 receptor antagonist
    SB-277011 dihydrochloride (SB-277011A dihydrochloride) is a potent, selective, orally bioavailable and brain penetrate dopamine D3 receptor antagonist, with pKis of 8.0, 6.0, <5.2 and 5.9 for D3, D2, 5-HT1B, and 5-HT1D receptors, respectively. 了解更多
  26. JNJ-37822681 dihydrochloride

    Catalog No. A21470
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    dopamine D2 receptor antagonist
    JNJ-37822681 dihydrochloride is a potent, specific, centrally active, fast-dissociating dopamine D2 receptor antagonist with a moderate binding affinity for the dopamine D2L receptor (Ki =158 nM), which has potential for the treatment of schizophrenia and bipolar disorder. 了解更多
  27. Vofopitant dihydrochloride

    Catalog No. A21543
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    NK1 receptor antagonist
    Vofopitant dihydrochloride (GR 205171A) is a potent, selective and orally available tachykinin neurokinin 1(NK1) receptor antagonist. 了解更多
  28. Granisetron Hydrochloride

    Catalog No. A10437
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    5-HT3 receptor 拮抗剂
    Granisetron Hydrochloride是血清素5-ht3受体拮抗剂。 了解更多
  29. Phenoxybenzamine hydrochloride

    Catalog No. A10719
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    α-adrenergic (AR) 拮抗剂/CaM 抑制剂
    Phenoxybenzamine hydrochloride是一种细胞可渗透的,非特异性的,不可逆的α-肾上腺素(AR)拮抗剂,也可作为CaM抑制剂。 了解更多
  30. ICI 118,551 hydrochloride

    Catalog No. A13225
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    β2 adrenergic 拮抗剂
    ICI 118,551 hydrochloride是选择性的β2 adrenergic receptor 拮抗剂,结合 β2,β1 和 β3 肾上腺素能受体的Ki 值分别为 0.7,49.5 和 611 nM。 了解更多
  31. HEAT hydrochloride (BE 2254)

    Catalog No. A13408
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    Adrenergic α1 Receptor 拮抗剂
    HEAT hydrochloride (BE 2254)是一种选择性很强的α1-肾上腺素受体拮抗剂,是3-[125I]-衍生物的前体。肾上腺素受体或肾上腺素能受体是参与多种交感神经系统过程的G蛋白偶联受体。 了解更多
  32. Idazoxan Hydrochloride

    Catalog No. A13409
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    α2- adrenoceptor 拮抗剂 / I2 imidazoline receptor 激动剂
    Idazoxan hydrochloride 是α2-AR肾上腺素受体拮抗剂和潜在I2咪唑啉受体激动剂。还显示I1咪唑啉受体拮抗剂活性。(I1、I2和α的公钥基础设施值分别为5.90、7.22、8.01、7.43和7.7)。 了解更多
  33. AMD-070 HCl

    Catalog No. A14997
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    CXCR4 拮抗剂
    在CXCR4 125I-SDF抑制结合试验中,AMD-070 HCl是一种有效的选择性CXCR4拮抗剂,IC50值为13 nM,抑制T-4型HIV-1(NL4.3株)在MT-4细胞中的复制和PBMC。 了解更多
  34. LY 334370 hydrochloride

    Catalog No. A17027
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    5-HT1F 激动剂
    LY 334370 hydrochloride是一种选择性的5-HT1F受体激动剂(Ki值为1.87、16.4,> 100 (IC50))。CAS:199673-74-0(LY 334370盐酸盐);182563-08-2(LY 334370游离碱) 了解更多
  35. Metoclopramide hydrochloride hydrate

    Catalog No. A18072
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    Dopamine D2 antagonist
    Metoclopramide hydrochloride hydrate is a dopamine D2 antagonist that is used as an antiemetic. 了解更多
  36. GSK1521498 free base (hydrochloride)

    Catalog No. A21792
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    μ-opioid receptor (MOR) antagonist
    GSK1521498 free base (hydrochloride) is a potent and selective μ-opioid receptor (MOR) antagonist. 了解更多
  37. Mianserin hydrochloride

    Catalog No. A10588
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    5-HT2/5-HT1 拮抗剂
    Mianserin hydrochloride是5-HT2/5-HT1拮抗剂。对5-HT6非选择性5-HT2受体拮抗剂具有中等亲和力。对5-HT6具有中等亲和力。 了解更多
  38. 5-HT1A receptor 拮抗剂
    NAD 299 hydrochloride (Robalzotan)是一种选择性的,高亲和力的5-HT1A受体拮抗剂(体外Ki = 0.6 nM)。 了解更多
  39. Alprenolol hydrochloride

    Catalog No. A17781
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    5-HT1A receptor antagonist
    Alprenolol (hydrochloride) is a non-selective beta blocker as well as 5-HT1A receptor antagonist. 了解更多
  40. Metipranolol hydrochloride

    Catalog No. A18064
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    β-adrenergic receptor antagonist
    Metipranolol (hydrochloride) is a non-selective β-adrenergic receptor (β-AR) antagonist. Formulations containing metipranolol have been used in the treatment of elevated IOP in patients with ocular hypertension or glaucoma. 了解更多
  41. SB 271046 Hydrochloride

    Catalog No. A11573
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    5-HT6 receptor antagonist
    SB271046 Hydrochloride is a potent, selective and orally active 5-HT6 receptor antagonist with pKi of 8.9. 了解更多
  42. Ziprasidone hydrochloride

    Catalog No. A16790
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    5-HT (serotonin)/dopamine receptor antagonist
    Ziprasidone Hcl(CP-88059 Hcl) is a combined 5-HT (serotonin) and dopamine receptor antagonist which exhibits potent effects of antipsychotic activity. 了解更多
  43. Sarpogrelate hydrochloride

    Catalog No. A17295
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    5-HT2 antagonist
    Sarpogrelate hydrochloride (MCI-9042), a selective 5-HT2 antagonist, has been widely used as an anti-platelet agent for the treatment of PAD. 了解更多
  44. SB 242084 hydrochloride

    Catalog No. A21349
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    5-HT2C receptor antagonist
    SB 242084 hydrochloride is a 5-HT2C receptor antagonist(pKi=9.0) that displays 158- and 100-fold selectivity over 5-HT2A and 5-HT2B receptors respectively. 了解更多
  45. Risperidone hydrochloride

    Catalog No. A21458
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    dopamine D2 receptor antagonist
    Risperidone hydrochloride is a serotonin 5-HT2 receptor blocker and a potent dopamine D2 receptor antagonist, with Kis of 0.16, 1.4 nM for 5-HT2 and D2 receptor, respectively. 了解更多
  46. SB-224289 hydrochloride

    Catalog No. A21920
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    5-HT1B receptor antagonist
    SB-224289 hydrochloride is a selective 5-HT1B receptor antagonist, with anxiolytic effect. 了解更多
  47. Amisulpride hydrochloride

    Catalog No. A21994
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    dopamine D2/D3 receptor antagonist
    Amisulpride hydrochloride is a dopamine D2/D3 receptor antagonist with Kis of 2.8 and 3.2 nM for human dopamine D2 and D3, respectively. 了解更多
  48. Cariprazine hydrochloride

    Catalog No. A15036
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    D3/D2 Dopamine Receptor 拮抗剂
    Cariprazine hydrochloride是一种新型的抗精神病药物,对多巴胺D3(Ki = 0.09 nM)和D2(Ki = 0.5 nM)受体具有高选择性和亲和力,对5-羟色胺5-HT(1A)受体具有中等亲和力。 了解更多
  49. Talnetant hydrochloride

    Catalog No. A15255
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    NK3 receptor 拮抗剂
    Talnetant Hydrochloride是一种有效且选择性的NK3受体拮抗剂(ki = 1.4 nM,hNK-3-CHO);对hNK-3受体的选择性是对hNK-2受体的100倍,在浓度高达100 uM时对hNK-1没有亲和力。 了解更多
  50. SB-269970 hydrochloride

    Catalog No. A21889
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    5-HT7 receptor antagonist
    SB269970 hydrochloride (SB-269970A) is a hydrochloride salt form of SB-269970, which is a 5-HT7 receptor antagonist with the pKi of 8.3, exhibits >50-fold selectivity against other receptors. 了解更多

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