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“jwh 370”的搜索结果

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  1. BTZ043 (BTZ038, BTZ044) Racemate
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    BTZ043 (BTZ038, BTZ044) Racemate

    Catalog No. A10165
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    DprE1 抑制剂
    BTZ043 (BTZ038,BTZ044) Racemate 抑制癸二烯基磷酸基-β-d-核糖2α-表异构酶，它是一种产生致病细菌结核分枝杆菌细胞壁的酶。 了解更多
  2. Tubacin
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    Tubacin

    Catalog No. A10954
    HDAC6 抑制剂
    Tubacin (tubulin acetylation inducer)是一种高效且选择性强，可逆，可透过细胞的HDAC6抑制剂，IC50为4 nM。 了解更多
  3. KRN 633
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    KRN 633

    Catalog No. A10504
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    VEGFR 抑制剂
    KRN 633是一种细胞可渗透、可逆、ATP竞争性VEGFR激酶抑制剂，仅在较高浓度下(IC50 = 0.97 μM和4.33 μM)抑制PDGFR-α和C-Kit，对其他17种激酶无活性(IC50 ≥ 10 μM)。 了解更多
  4. MK-2461
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    MK-2461

    Catalog No. A11753
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    c-Met 抑制剂
    MK-2461是一种新型的多靶点激酶抑制剂，优先抑制活化的c-Met受体。 了解更多
  5. P505-15 (PRT062607, BIIB057)
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    P505-15 (PRT062607, BIIB057)

    Catalog No. A11952
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    Syk 抑制剂
    P505-15 (PRT062607,BIIB057)是一种新型的，高度选择性的，Syk抑制剂（SYK IC（50）= 1 nM），具有比SYK活性至少高80倍的抗SYK活性。 了解更多
  6. JNK-IN-8
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    JNK-IN-8

    Catalog No. A12749
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    JNK 抑制剂
    JNK-IN-8是第一种JNK1，JNK2和JNK4不可逆JNK抑制剂，IC50分别为4.7 nM，18.7 nM和1 nM。 了解更多
  7. BCH
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    BCH

    Catalog No. A13370
    LAT1 抑制剂
    BCH是L型氨基酸转运蛋白LAT1的抑制剂。通过激活KB，Saos2和C6癌细胞系中的半胱氨酸蛋白酶抑制生长并诱导凋亡。 了解更多
  8. Batimastat (BB-94)
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    Batimastat (BB-94)

    Catalog No. A12985
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    MMP 抑制剂
    Batimastat (BB-94)是多种基质金属蛋白酶（MMP）的强效合成抑制剂，包括间质胶原酶（IC50 = 3 nM），溶血素（IC50 = 20 nM），Mr 72,000型IV胶原酶（IC50 = 4） nM），92,000型IV胶原酶先生（IC50 = 4 nM）和基质溶素（IC50 = 6 nM）。它是一种低分子量（MW = 478）的肽样胶原蛋白底物类似物，由类似物结合而成，分别与MMP和催化活性锌原子结合在一起。 了解更多
  9. PRT062607 HCL
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    PRT062607 HCL

    Catalog No. A12731
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    Syk 抑制剂
    PRT2607，也称为PRT062607，P505-15和BIIB057，是一种新型，高度选择性且口服可生物利用的小分子SYK抑制剂（SYK IC（50）= 1 nM），具有至少80倍的抗SYK活性 大于对其他激酶的亲和力。 了解更多
  10. UNC1215
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    UNC1215

    Catalog No. A12948
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    L3MBTL3 抑制剂
    UNC1215是具有细胞活性的L3MBTL3的强效选择性拮抗剂。 了解更多
  11. Mevastatin
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    Mevastatin

    Catalog No. A13709
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    HMG-CoA reductase 抑制剂
    Mevastatin是HMG-CoA还原酶的抑制剂。 了解更多
  12. ESI-09
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    ESI-09

    Catalog No. A14233
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    EPAC1/EPAC2 抑制剂
    ESI-09是一种直接由cAMP（EPAC）抑制剂激活的特异性交换蛋白，对于EPAC1和EPAC2，IC50为3.2 uM和1.4 uM。 了解更多
  13. 1-Azakenpaullone
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    1-Azakenpaullone

    Catalog No. A14303
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    GSK-3β 抑制剂
    1-Azakenpaullone是一种有效的选择性GSK-3β抑制剂，IC50为18 nM，选择性比CDK1/cyclin B和CDK5/p25高100倍。 了解更多
  14. DTP348
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    DTP348

    Catalog No. A14410
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    CAIX 抑制剂/ radiosensitizer
    DTP348是双重CAIX抑制剂/放射增敏剂。 了解更多
  15. CAY10650
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    CAY10650

    Catalog No. A14355
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    cPLA2α 抑制剂
    CAY10650是一种高效（IC50 = 12 nM）cPLA2α抑制剂。 了解更多
  16. AK-1
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    AK-1

    Catalog No. A14370
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    SIRT2 抑制剂
    AK-1比SIRT1和SIRT3选择性抑制SIRT2。 了解更多
  17. RG108
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    RG108

    Catalog No. A13054
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    DNA methyltransferase 抑制剂
    RG108是DNA甲基转移酶的非核苷抑制剂，IC50为115 nM。 了解更多
  18. Cyclothiazide
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    Cyclothiazide

    Catalog No. A13700
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    AMPA desensitization 抑制剂
    Cyclothiazide是苯并噻二叠氮，可作为AMPA受体的增效剂，正向调节其对谷氨酸的响应（EC50 = 3.8 M）。 了解更多
  19. NBMPR
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    NBMPR

    Catalog No. A13701
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    ENT1 抑制剂
    NBMPR是一种核苷类似物，可竞争性抑制平衡的核苷转运蛋白1（大鼠和人的Kd = 0.1-1.0 nM，IC50s = 4.6和3.6 nM）。 了解更多
  20. O6-Benzylguanine
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    O6-Benzylguanine

    Catalog No. A13706
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    MGMT 抑制剂
    O6-Benzylguanine是DNA烷基转移酶的有效底物和有效灭活剂。O6-苄基鸟嘌呤是MGMT的抑制剂。 了解更多
  21. UK 370106
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    UK 370106

    Catalog No. A15316
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    MMP-3/MMP-12 Inhiibitor
    UK 370106是一种高度选择性的MMP-3和MMP-12抑制剂。 了解更多
  22. TC-H 106
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    TC-H 106

    Catalog No. A15357
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    HDAC 抑制剂
    TC-H 106是一种慢速，紧密结合的I类HDAC（组蛋白脱乙酰基酶）抑制剂。 了解更多
  23. 4-HQN
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    4-HQN

    Catalog No. A15370
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    PARP 抑制剂
    4-HQN已显示抑制PARP（聚（ADP-核糖）合成酶），该酶催化NAD+的ADP-核糖部分与各种蛋白质的共价结合。 了解更多
  24. GSK2879552
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    GSK2879552

    Catalog No. A15547
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    LSD1 抑制剂
    GSK2879552是一种可逆的赖氨酸特异性脱甲基酶1（LSD1）抑制剂，具有潜在的抗肿瘤活性。 了解更多
  25. E7820
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    E7820

    Catalog No. A15456
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    lpha-2-integrin 抑制剂
    E7820是一种小分子芳香族磺酰胺衍生物，具有潜在的抗血管生成和抗肿瘤活性。E7820通过抑制整合素α2（一种在内皮细胞上表达的细胞粘附分子）来抑制血管生成。 了解更多
  26. AZ-33
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    AZ-33

    Catalog No. A13341
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    LDHA 抑制剂
    AZ33是LDHA抑制剂。 了解更多
  27. CID 797718
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    CID 797718

    Catalog No. A13809
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    PKD1 抑制剂
    CID797718是CID755673（Adooq目录号A13804）的结构类似物。它是效力降低10倍的PKD1抑制剂，IC50值为7.0+/-0.8 uM。 了解更多
  28. CL-387785 (EKI-785)
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    CL-387785 (EKI-785)

    Catalog No. A13146
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    EGFR 抑制剂
    CL-387785是EGFR的不可逆抑制剂，IC50为370+/-120 pM；能够在功能水平上克服由T790M突变引起的抗药性。 了解更多
  29. BML-210
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    BML-210

    Catalog No. A15935
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    HDAC 抑制剂?
    BML-210是HDAC抑制剂。BML-210诱导宫颈癌细胞中的生长抑制和凋亡并调节HDAC和DAPC复合物的表达水平。 了解更多
  30. FLT3-IN-1
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    FLT3-IN-1

    Catalog No. A16249
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    FLT3 抑制剂
    FLT3-IN-1是一种新型的有效选择性Flt3抑制剂，IC50为10 nM。抗表达FLT3-ITD的MV4-11细胞，IC50为6 nM。 了解更多
  31. CI 976
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    CI 976

    Catalog No. A16370
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    ACAT/SOAT 抑制剂
    CI 976是肝和肠酰基辅酶A胆固醇酰基转移酶（ACAT）和固醇O-酰基转移酶（SOAT）的三甲氧基脂肪酸苯胺抑制剂。Cl 976降低非高密度脂蛋白（non-HDL）胆固醇并增加HDL-胆固醇浓度。 了解更多
  32. AX-024
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    AX-024

    Catalog No. A16926
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    T cell receptor 抑制剂
    AX-024是一种细胞因子释放抑制剂，可以强烈抑制白介素6（IL-6），肿瘤坏死因子-α（TNFα），干扰素-γ（IFN-γ），IL-10和IL-17A的产生。 了解更多
  33. Elbasvir (MK-8742)
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    Elbasvir (MK-8742)

    Catalog No. A16855
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    NS5A 抑制剂
    Elbasvir (MK-8742)是一种NS5A抑制剂，可预防丙型肝炎病毒RNA复制和病毒体组装。根据基因型，EC50的中值范围为0.2至3600 pmol/L。 了解更多
  34. SR-4370
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    SR-4370

    Catalog No. A16899
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    HDAC 抑制剂
    SR-4370是HDAC抑制剂。SR-4370对HDAC1，HDAC2和HDAC3的IC50值分别为0.5 uM，0.1 uM和0.06 uM。 了解更多
  35. PF-06737007
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    PF-06737007

    Catalog No. A17179
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    Trk 抑制剂
    PF-06737007是泛原肌球蛋白相关激酶（Trk）抑制剂。 了解更多
  36. SSE15206
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    SSE15206

    Catalog No. A18350
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    Microtubule/Tubulin Inhibitor
    SSE15206 is a pyrazolinethioamide derivative that has potent antiproliferative activities in cancer cell lines of different origins and overcomes resistance to microtubule-targeting agents. 了解更多
  37. Cangrelor Tetrasodium
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    Cangrelor Tetrasodium

    Catalog No. A17919
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    P2Y12 receptors inhibitor
    Cangrelor Tetrasodium is a high-affinity, reversible inhibitor of P2Y12 receptors that causes almost complete inhibition of ADP-induced platelet aggregate. It is a modified ATP derivative stable to enzymatic degradation. Unlike clopidogrel (Plavix), which is a prodrug, cangrelor is an active drug not requiring metabolic conversion. 了解更多
  38. BC-1215
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    BC-1215

    Catalog No. A18605
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    FBXO3 inhibitor
    BC-1215 is an inhibitor of F-box protein 3 (FBXO3, a ubiquitin E3 ligase component, IC50=0.9 μg/mL for IL-1β release). BC-1215 decreases Fbxo3-Fbxl2 interaction and prevents SCFFbxo3 catalyzed Fbxl2 ubiquitination. 了解更多
  39. DW14800
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    DW14800

    Catalog No. A18491
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    PRMT5 inhibitor
    DW14800 is a protein arginine methyltransferase 5 (PRMT5) inhibitor, with an IC50 of 17 nM. DW14800 reduces H4R3me2s levels and enhances the transcription of HNF4α, but does not alter PRMT5 expression. Anti-cancer activity. 了解更多
  40. ZT-12-037-01
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    ZT-12-037-01

    Catalog No. A18395
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    ATP-competitive STK19 inhibitor
    ZT-12-037-01 is a potent, selective, ATP-competitive STK19 inhibitor. ZT-12-037-01 effectively blocks oncogenic NRAS-driven melanocyte malignant transformation and melanoma growth in vitro and in vivo. 了解更多
  41. JNJ4796
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    JNJ4796

    Catalog No. A13707
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    Influenza virus inhibitor
    JNJ4796 is an oral active fusion inhibitor of influenza virus, neutralizing influenza A group 1 viruses by inhibiting hemagglutinin (HA)-mediated fusion. 了解更多
  42. RIPA-56
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    RIPA-56

    Catalog No. A12473
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    RIP1 inhibitor
    RIPA-56 is a highly potent, selective, and metabolically stable inhibitor of receptor-interacting protein 1 (RIP1) with an IC50 of 13 nM. 了解更多
  43. LDN-27219
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    LDN-27219

    Catalog No. A20844
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    hTGase inhibitor
    LDN-27219 is a potent inhibitor of hTGase(Tissue transglutaminase) with an IC50 of 0.6 uM. 了解更多
  44. Solenopsin
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    Solenopsin

    Catalog No. A21087
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    ATP-competitive AKT inhibitor
    Solenopsin is an ATP-competitive AKT inhibitor with IC50 value of 10 μM . 了解更多
  45. Ensartinib hydrochloride
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    Ensartinib hydrochloride

    Catalog No. A21719
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    ALK/MET inhibitor
    Ensartinib hydrochloride (X-396 hydrochloride) is a potent and dual ALK/MET inhibitor with IC50s of <0.4 nM and 0.74 nM, respectively. 了解更多
  46. Liarozole dihydrochloride
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    Liarozole dihydrochloride

    Catalog No. A21853
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    CYP450 dependent inhibitor
    Liarozole dihydrochloride (R75251; R85246) is a cytochrome P450 (CYP450) dependent inhibitor, orally active, it also a potent inhibitor of estrogen (via inhibition of aromatase) and testicular androgen synthesis (inhibition of 17 ,20-lyase). 了解更多
  47. MSI-1436 lactate
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    MSI-1436 lactate

    Catalog No. A21929
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    PTB1B inhibitor
    MSI-1436 lactate is a selective, non-competitive inhibitor of the enzyme protein-tyrosine phosphatase 1B (PTB1B), with an IC50 of 1 μM, 200-fold preference over TCPTP (IC50 of 224 μM). 了解更多
  48. CG-806
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    CG-806

    Catalog No. A19814
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    FLT3/BTK inhibitor
    CG-806 is an orally active, potent and non-covalent pan-FLT3/pan-BTK inhibitor with an IC50 of 0.08 μM for FLT3. CG-806 has an IC50 of 11 nM against FLT3 wild type (WT)-transfected Ba/F3 cells. 了解更多
  49. KN-92
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    KN-92

    Catalog No. A15137
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    CaMK-II 抑制剂
    KN-92是KN-93的非活性衍生物。KN-93是Ca2+/钙调蛋白依赖性激酶II（CaMKII）的选择性抑制剂，竞争性阻断CaM与激酶的结合（Ki = 370 nM）。 了解更多
  50. KN-92 phosphate
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    KN-92 phosphate

    Catalog No. A15139
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    CaMKII 抑制剂
    KN-92 phosphate是KN-93的非活性衍生物。KN-93是Ca2+/钙调蛋白依赖性激酶II（CaMKII）的选择性抑制剂，竞争性阻断CaM与激酶的结合（Ki = 370 nM）。 了解更多

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