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Acetazolamide
Catalog No. A15859 Carbonic Anhydrase 抑制剂Acetazolamide是一种有效的碳酸酐酶（CA）抑制剂，在临床实践中通常用作迅速降低眼内压（IOP）的直接且容易获得的选择。 了解更多 -
Nesbuvir
Catalog No. A11510 -
Salirasib
Catalog No. A11572 -
GSK744 (S/GSK1265744)
Catalog No. A16014 HIV integrase 抑制剂GSK744 (S/GSK1265744)是一种有效的HIV整合酶抑制剂，可作为口服导入片剂和长效注射剂，用于治疗和预防HIV感染。 了解更多 -
Dolutegravir Sodium
Catalog No. A16162 HIV integrase 抑制剂Dolutegravir Sodium是一种HIV整合酶抑制剂（IC50 = 2.7 nM），对耐raltegravir的签名突变体Y143R，Q148K，N155H和G140S/Q148H具有中等活性。 了解更多 -
Levofloxacin hydrate
Catalog No. A16167 topoisomerase II IV 抑制剂Levofloxacin hydrate是广谱的第三代氟喹诺酮类抗生素，是具有抗菌活性的氧氟沙星的旋光性L-异构体。 了解更多 -
Benzenesulfonamide
Catalog No. A13594 -
BQU57
Catalog No. A14956 -
Clinafloxacin
Catalog No. A16458 DNA gyrase and topoisomerase IV 抑制剂Clinafloxacin是一种氟喹诺酮，可双重抑制肺炎链球菌中的DNA促旋酶和拓扑异构酶IV。 了解更多 -
Pixantrone
Catalog No. A13022 -
ASP 2151 (Amenamevir)
Catalog No. A13180 herpes virus helicase-primase 抑制剂ASP 2151 (Amenamevir)是疱疹病毒解旋酶-引发酶抑制剂。在全身或局部使用后，ASP2151对单纯疱疹性角膜炎的抗HSV活性明显优于伐昔洛韦和阿昔洛韦。 了解更多 -
Topotecan
Catalog No. A16815 -
ARS-1620
Catalog No. A16809 -
Vorasidenib
Catalog No. A16908 IDH1 抑制剂Vorasidenib (AG-881)是一种有效且选择性的口服抑制剂，可抑制细胞质中异柠檬酸脱氢酶1型(IDH1，IDH1 [NADP+]可溶)和2型（IDH2异柠檬酸脱氢酶[NADP+]）的突变形式。线粒体中的线粒体，具有潜在的抗肿瘤活性。 了解更多 -
JNJ-64619178
Catalog No. A16861 Histone Methyltransferase 抑制剂JNJ-64619178是PRMT5抑制剂，在不同的体外和细胞条件下均具有高选择性和强效性（亚纳摩尔范围，PRMT5-MEP-50 IC50 = 0.14 nM），并具有良好的药代动力学和安全性。 了解更多 -
Bictegravir
Catalog No. A17011 HIV-1 integrase 抑制剂Bictegravir，也称为GS-9883，是一种有效的，未经增强的，每日一次的HIV-1整合酶链转移抑制剂（INSTI）（IC50-1.6 nM），具有改善的药代动力学和体外耐药性。 了解更多 -
CMP3a
Catalog No. A18347 NEK2 kinase inhibitorCMP3a is a NEK2 kinase inhibitor. CMP3a efficiently attenuated GBM growth in a mouse model and exhibited a synergistic effect with radiotherapy. Targeting NEK2 attenuates glioblastoma growth and radioresistance by destabilizing histone methyltransferase EZH2. 了解更多 -
Benzthiazide
Catalog No. A17355 CA9 inhibitorBenzthiazide is a long-acting diuretic and a hypertension agent. Benzthiazide is an inhibitor of carbonic anhydrase 9 (CA9), with Kis of 8.0, 8.8 and 10 nM for CA9, CA2 and CA1, respectively. Benzthiazide also suppresses proliferation of cancer cells. 了解更多 -
Ethoxzolamide
Catalog No. A17359 Carbonic anhydrase inhibitorEthoxzolamide is a carbonic anhydrase inhibitor with Ki of 1 nM. 了解更多 -
Tacrine HCl
Catalog No. A17374 AChE & butyrylcholinesterase inhibitorTacrine is a derivative of aminoacridine that functions as an inhibitor of both acetylcholinesterase (AChE) and butyrylcholinesterase (IC50s = 31 and 26.5 nM, respectively). 了解更多 -
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MLS0315771
Catalog No. A17219 MPI inhibitorMLS0315771 is a potent competitive phosphomannose isomerase (MPI) inhibitor. 了解更多 -
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Iopanoic acid
Catalog No. A17658 cholecystographic agentIopanoic acid is an inhibitor of 5'-Deiodinase and also an iodinated contrast medium. 了解更多 -
Minaprine dihydrochloride
Catalog No. A17722 MAO-A inhibitorMinaprine is a reversible inhibitor of MAO-A; weakly inhibit acetylcholinesterase; an antidepressant for treatment of depression. 了解更多 -
Drofenine Hydrochloride
Catalog No. A17724 BChE inhibitorDrofenine hydrochloride is a potent competitive inhibitor of BChE, and the ki values of Drofenine is calculated to be 3 uM. 了解更多 -
Edrophonium chloride
Catalog No. A17794 acetylcholinesterase inhibitorEdrophonium Chloride, also known as Tensilon, is an acetylcholinesterase inhibitor used in cardiac arrhythmias and in the diagnosis of myasthenia gravis. Edrophonium Chloride has also been used as an antidote to curare principles. 了解更多 -
Cangrelor Tetrasodium
Catalog No. A17919 P2Y12 receptors inhibitorCangrelor Tetrasodium is a high-affinity, reversible inhibitor of P2Y12 receptors that causes almost complete inhibition of ADP-induced platelet aggregate. It is a modified ATP derivative stable to enzymatic degradation. Unlike clopidogrel (Plavix), which is a prodrug, cangrelor is an active drug not requiring metabolic conversion. 了解更多 -
Piperidolate hydrochloride
Catalog No. A18144 antimuscarinicPiperidolate hydrochloride is an antimuscarinic, Also a potential inhibitor of human glutathione transferase P1-1. 了解更多 -
Fosphenytoin disodium
Catalog No. A18184 PDE3 inhibitorFosphenytoin Sodium is the sodium salt form of fosphenytoin, a prodrug that is hydrolyzed to the anticonvulsant phenytoin. It is an PDE3 (phosphodiesterase 3) inhibitor. 了解更多 -
AMG-510 racemate
Catalog No. A18752 KRAS G12C covalent inhibitorAMG-510 is a potent, orally bioavailable, and selective KRAS G12C covalent inhibitor with anti-tumor activity. 了解更多 -
NGI-1
Catalog No. A18706 OST inhibitorNGI-1 (ML414) is a potent oligosaccharyltransferase (OST) inhibitor, directly targeting and blocking the function of the OST catalytic subunits STT3A and STT3B. NGI-1 is a cell permeable inhibitor and can effectively reduce virus infectivity without affecting cell viability. 了解更多 -
D5D-IN-326
Catalog No. A18688 D5D inhibitorD5D-IN-326 is a selective, orally active delta-5 desaturase (D5D) inhibitor, with IC50s of 72 and 22 nM for rat and human D5D in enzymic and cell-based assays, respectively, has no effect on D6D or D9D activity. 了解更多
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