“rasgap ras p21”的搜索结果

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  1. Resminostat hydrochloride

    Catalog No. A15220
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    HDAC 抑制剂
    Resminostat hydrochloride是HDAC1/3/6的有效抑制剂(IC50 = 43-72 nM);对HDAC8的效力较低,IC50为877 nM。 了解更多
  2. Remodelin

    Catalog No. A21985
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    acetyl-transferase protein NAT10 inhibitor
    Remodelin is a novel potent and selective inhibitor of the acetyl-transferase protein NAT10. 了解更多
  3. Entacapone sodium salt

    Catalog No. A21888
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    COMT inhibitor
    Entacapone is a specific, potent, peripherally acting catechol-O-methyltransferase (COMT) inhibitor with IC50 of 151 nM for PD treatment. 了解更多
  4. BIX-01338 hydrate

    Catalog No. A21812
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    histone lysine methyltransferase inhibitor
    BIX-01338 hydrate is a histone lysine methyltransferase inhibitor. 了解更多
  5. O6BTG-octylglucoside

    Catalog No. A11432
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    MGMT inhibitor
    O6BTG-octylglucoside is a potent O6-methylguanine-DNAmethyl-transferase (MGMT) inhibitor, with IC50s of 32 nM in vitro (cell extracts) and 10 nM in HeLa S3 cells. 了解更多
  6. Histone Acetyltransferase Inhibitor II

    Catalog No. A12331
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    cell permeable p300 inhibitor
    Histone Acetyltransferase Inhibitor II is a potent and cell permeable p300 inhibitor, with an IC50 of 5 ?M; Histone Acetyltransferase Inhibitor II can be used in cancer research. 了解更多
  7. Entacapone

    Catalog No. A10355
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    COMT inhibitor
    Entacapone is a specific, potent, peripherally acting catechol-O-methyltransferase (COMT) inhibitor with IC50 of 151 nM for PD treatment. 了解更多
  8. SIS-17

    Catalog No. A18463
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    HDAC 11 inhibitor
    SIS17 is a potent and selective HDAC 11 inhibitor with an IC50 value of 0.83 μM. SIS17, is active in cells and inhibited the demyristoylation of a known HDAC11 substrate, serine hydroxymethyl transferase 2, without inhibiting other HDACs. 了解更多
  9. P300/CBP-IN-3

    Catalog No. A18544
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    p300/CBP histone acetyltransferase inhibitor
    P300/CBP-IN-3, a p300/CBP histone acetyltransferase inhibitor. 了解更多
  10. CM-675

    Catalog No. A18741
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    PDE5/HDAC-1 inhibitor
    CM-675 is a dual phosphodiesterase 5 (PDE5) and class I histone deacetylases-selective inhibitor, with IC50 values of 114 nM and 673 nM for PDE5 and HDAC1, respectively. CM-675 has potential to treat Alzheimer??s disease. 了解更多
  11. JNJ-64619178

    Catalog No. A16861
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    Histone Methyltransferase 抑制剂
    JNJ-64619178是PRMT5抑制剂,在不同的体外和细胞条件下均具有高选择性和强效性(亚纳摩尔范围,PRMT5-MEP-50 IC50 = 0.14 nM),并具有良好的药代动力学和安全性。 了解更多
  12. WM-1119

    Catalog No. A16828
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    lysine acetyltransferase KAT6A 抑制剂
    WM-1119是赖氨酸乙酰基转移酶KAT6A的高效选择性抑制剂,IC50为0.25 uM。它对KAT6A的活性分别是对KAT5或KAT7的1100倍和250倍。 了解更多
  13. AMI5

    Catalog No. A16376
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    protein methyltransferase 抑制剂
    AMI5是一种非选择性蛋白质甲基转移酶抑制剂。 了解更多
  14. TC-E 5001

    Catalog No. A11454
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    TNKS 抑制剂
    TC-E 5001是双重tankyrase(TNKS)抑制剂(TNKS1和TNKS2的Kd值分别为79和28 nM,TNKS2的IC50 = 33 nM),在PARP1和PARP2上没有活性(IC50> 19 uM)。抑制Wnt信号并稳定Axin2水平。 了解更多
  15. AZ6102

    Catalog No. A15873
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    TNKS1/2 抑制剂
    AZ6102是有效的TNKS1/2抑制剂,对其他PARP家族酶具有100倍的选择性,对DLD-1细胞中Wnt途径的抑制作用的IC50为5 nM。 了解更多
  16. MN-64

    Catalog No. A15927
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    TNKS 抑制剂
    MN-64是Tankyrase 1和2的有效和选择性抑制剂(IC50分别为6和72 nM)。 了解更多
  17. NVP-TNKS656

    Catalog No. A15786
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    TNKS2 抑制剂
    NVP-TNKS656是一种高效,选择性和活性的TNKS2抑制剂,IC50为6 nM。对PARP1和PARP2的选择性> 300倍。 了解更多
  18. G007-LK

    Catalog No. A15528
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    TNKS 抑制剂
    G007-LK对坦科聚合酶1和2具有很高的选择性,生化IC50值分别为46 nM和25 nM,细胞IC50值为50 nM,并具有出色的小鼠药代动力学特征, 了解更多
  19. AZD1152

    Catalog No. A15011
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    Aurora B 抑制剂
    AZD1152是一种前药,可在血清中迅速经历磷酸酶介导的裂解作用,释放出Barasertib-hQPA(一种选择性的Aurora B激酶抑制剂),在急性髓细胞性白血病(AML)患者的临床研究中显示出初步活性。 了解更多
  20. AIM-100

    Catalog No. A14986
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    Ack1 (TNK2) 抑制剂
    AIM-100是Ack1的小分子抑制剂,IC50为24 nM。 了解更多
  21. RG108

    Catalog No. A13054
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    DNA methyltransferase 抑制剂
    RG108是DNA甲基转移酶的非核苷抑制剂,IC50为115 nM。 了解更多
  22. WIKI4

    Catalog No. A14283
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    Tankyrase 抑制剂
    WIKI4是一种新型的Tankyrase抑制剂,对TNKS2的IC50为15 nM。 了解更多
  23. Nexturastat A

    Catalog No. A14032
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    HDAC6 抑制剂
    Nexturastat A是一种芳基脲衍生物,可作为组蛋白脱乙酰基酶6(HDAC6)的有效且高度选择性的抑制剂(IC50 = 5.02+/-0.60 nM)。 了解更多
  24. Resminostat

    Catalog No. A12556
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    HDAC 抑制剂
    Resminostat,也称为RAS2410,是一种有效的I和II类组蛋白脱乙酰基酶(HDAC)抑制剂。它结合并抑制HDAC,从而导致高度乙酰化的组蛋白的积累。选择性的抑制HDAC1/3/6,IC50为42.5 nM/50.1 nM/71.8 nM,作用于HDAC8效果弱,IC50为877 nM。 了解更多
  25. JW 55

    Catalog No. A13731
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    TNKS1/2 抑制剂
    JW 55是端锚聚合酶1和2(TNKS1/2)的PARP域的抑制剂。 了解更多
  26. Decitabine

    Catalog No. A10292
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    DNA Methyltransferase 抑制剂
    Decitabine是一种次甲基化剂,它通过抑制DNA甲基转移酶来使DNA次甲基化。 了解更多
  27. AZD1152-HQPA (Barasertib)

    Catalog No. A10109
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    Aurora Kinase B 抑制剂
    AZD1152-HQPA (Barasertib)是Aurora B的高效抑制剂,Ki值分别为0.36(Aurora B)和1369 nM(Aurora A),与一组其他50种激酶相比具有很高的特异性。 了解更多

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