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BMS-663068 Tris
Catalog No. A15026 -
Fosamprenavir Calcium Salt
Catalog No. A15089 HIV protease 抑制剂Fosamprenavir Calcium Salt 是抗逆转录病毒蛋白酶抑制剂amprenavir的磷酸酯前药，与母体分子相比具有更高的溶解度，并有可能减轻当前给药方案中的药丸负担；GW433908G是前药的钙盐。 了解更多 -
Tipranavir
Catalog No. A15262 HIV protease 抑制剂Tipranavir是一种非肽类HIV蛋白酶抑制剂（NPPI），可抑制HIV-1蛋白酶的酶促活性和二聚作用，对多种抗PI的HIV-1分离株具有有效的活性。 了解更多 -
Enfuvirtide Acetate(T-20)
Catalog No. A15825 -
Trovirdine
Catalog No. A13199 HIV-1 RT 抑制剂Trovirdine当使用杂聚合引物/模板（寡DNA/核糖体RNA）和dGTP作为底物时，trovirdine抑制HIV-1 RT的IC50为7 nM。 了解更多 -
Nelfinavir
Catalog No. A11504 HIV-1 protease 抑制剂Nelfinavir是一种有效的口服生物可利用的人类免疫缺陷病毒HIV-1蛋白酶抑制剂(Ki=2 nM ),广泛用于与HIV逆转录酶抑制剂联合治疗HIV感染。 了解更多 -
(±)-BI-D
Catalog No. A16024 -
GSK2838232
Catalog No. A15965 -
Darunavir
Catalog No. A20829 -
Teneligliptin hydrobromide
Catalog No. A15258 DPP-4 抑制剂Teneligliptin hydrobromide是一种新颖，有效且持久的二肽基肽酶-4抑制剂。在体外竞争性抑制人血浆，大鼠血浆和人重组DPP-4，IC50值约为1 nM。 了解更多 -
DPPI 1c hydrochloride
Catalog No. A15298 DPP-4 抑制剂DPPI 1c hydrochloride是一种双氰基吡咯烷化合物，可作为CD26（DPP 4）的缓慢结合和定点活性抑制剂，IC50 = 106 nM，对DPP II，DPP III，DPP VIII，DPP IX，FAP几乎没有活性，甚至浓度高达30μM的APP。 了解更多 -
PK 44 phosphate
Catalog No. A15309 -
NVP DPP 728 dihydrochloride
Catalog No. A15320 DPP-4 抑制剂NVP DPP 728 dihydrochloride是一种有效的活性二肽基肽酶(DPP)-IV抑制剂，Ki和IC50值分别为11 nM和14 nM。 了解更多 -
Teneligliptin
Catalog No. A15505 -
1G244
Catalog No. A18709 -
Talabostat
Catalog No. A14079 DPP-IV inhibitorTalabostat (Val-boroPro; PT100) is an orally active and nonselective dipeptidyl peptidase IV (DPP-IV) inhibitor (IC50 < 4 nM; Ki = 0.18 nM) and the first clinical inhibitor of fibroblast activation protein (FAP) (IC50 = 560 nM). 了解更多 -
Saxagliptin hydrate
Catalog No. A16694 DPP4 inhibitorSaxagliptin H2O(BMS477118 H2O) is a selective and reversible DPP4 inhibitor with IC50 of 26 nM and Ki of 1.3 nM. 了解更多 -
Gemigliptin
Catalog No. A21285 DPP4 inhibitorGemigliptin is a highly selective dipeptidyl peptidase 4 (DPP4) inhibitor with a KD of 7.25 nM. 了解更多 -
Teneligliptin hydrobromide hydrate
Catalog No. A21465 DPP-4 inhibitorTeneligliptin hydrobromide hydrate is a potent chemotype prolylthiazolidine-based DPP-4 inhibitor, which competitively inhibits human plasma, rat plasma, and human recombinant DPP-4 in vitro, with IC50s of approximately 1 nM. 了解更多 -
Diprotin A TFA
Catalog No. A21475 DPP IV inhibitorDiprotin A (TFA) is an inhibitor of dipeptidyl peptidase IV (DPP-IV). 了解更多 -
Gosogliptin
Catalog No. A21566 DPP-IV inhibitorGosogliptin is a potent and selective inhibitor of dipeptidyl peptidase-IV (DPP-IV). 了解更多 -
Dutogliptin
Catalog No. A21573 DPP4 inhibitorDutogliptin (PHX-1149 free base) is an orally available, potent, and selective dipeptidyl peptidase-4 (DPP4) inhibitor for the treatment of type 2 diabetes mellitus. 了解更多 -
Vildagliptin dihydrate
Catalog No. A21898 DPP4 inhibitorVildagliptin (LAF237 dihydrate;NVP-LAF 237 dihydrate) is a dipeptidyl peptidase 4 (DPP4) inhibitor that delays the degradation of glucagon-like peptide-1 (GLP-1). 了解更多 -
Saxagliptin (BMS-477118)
Catalog No. A11109 DPP-4 抑制剂Saxagliptin (BMS-477118)是一种新型二肽基肽酶4（DPP-4）抑制剂，IC50为50 nM。 了解更多 -
Sitagliptin phosphate monohydrate
Catalog No. A10848 DDP-4 抑制剂Sitagliptin phosphate monohydrate是二肽基肽酶-4（DPP-4）类的抗糖尿病（抗高血糖）药物。 DPP-4酶的抑制作用被认为会增加胰高血糖素样肽1（GLP-1），从而抑制胰高血糖素释放，刺激胰岛素释放并降低血糖。 了解更多 -
Linagliptin (BI-1356)
Catalog No. A11224 DPP-4 抑制剂Linagliptin (BI-1356)是DPP-4抑制剂，是一种降解肠降血糖素激素胰高血糖素样肽1（GLP-1）和葡萄糖依赖性促胰岛素多肽（GIP）的酶。 了解更多 -
Vildagliptin
Catalog No. A12528 -
Alogliptin Benzoate
Catalog No. A13311 -
Trelagliptin Succinate (SYR-472)
Catalog No. A13312 DPP-4 抑制剂Trelagliptin Succinate (SYR-472)是一种长效的二肽基肽酶4（DPP-4）抑制剂，正在开发用于治疗2型糖尿病（T2D）。 了解更多 -
Sitagliptin
Catalog No. A14377 -
Alogliptin
Catalog No. A13571 -
Anagliptin
Catalog No. A13529 -
UAMC 00039 dihydrochloride
Catalog No. A16047 DPP-II 抑制剂UAMC 00039 dihydrochloride是二肽基肽酶II（DPP-II）的有效抑制剂（IC50 = 0.48 nM）。展示了DPP-II对DPP-9，DPP-8和DPP-IV的选择性（IC50值分别为78.6、142和165μM）。 了解更多 -
Talabostat mesylate
Catalog No. A14080 -
Balicatib
Catalog No. A12020 -
MG-101
Catalog No. A14220 -
PD 151746
Catalog No. A14245 -
Calpain Inhibitor II, ALLM
Catalog No. A14911 Calpain 抑制剂Calpain Inhibitor II, ALLM是钙蛋白酶I，钙蛋白酶II，组织蛋白酶L和组织蛋白酶B的细胞可渗透抑制剂，Ki值分别为120 nM，230 nM，0.6 nM和100 nM。 了解更多 -
Acetyl-Calpastatin (184-210) (human)
Catalog No. A15290 Selective calpain 抑制剂Acetyl-Calpastatin (184-210) (human)选择性钙蛋白酶抑制剂。强烈抑制钙蛋白酶I（Ki = 0.2 nM）和II，但不抑制木瓜蛋白酶，胰蛋白酶和组织蛋白酶L（Ki = 6 uM）。增加淀粉样β蛋白（Aβ）42，Aβ40和Aβ42比率的分泌。 了解更多 -
Calpeptin
Catalog No. A15295 -
Cathepsin Inhibitor 1
Catalog No. A11466 Cathepsin 抑制剂Cathepsin Inhibitor 1抑制剂1 是一种Cathepsin (L, L2, S, K, B)的抑制剂，pIC50分别为7.9、6.7、6.0、5.5和5.2。 了解更多 -
Cysteine Protease inhibitor
Catalog No. A21048 cysteine protease inhibitorCysteine Protease inhibitor is an inhibitor of cysteine protease. 了解更多 -
Odanacatib (MK-0822)
Catalog No. A11265
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