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Histone Acetyltransferase Inhibitor II
Catalog No. A12331 cell permeable p300 inhibitorHistone Acetyltransferase Inhibitor II is a potent and cell permeable p300 inhibitor, with an IC50 of 5 ?M; Histone Acetyltransferase Inhibitor II can be used in cancer research. 了解更多 -
(-)-Epigallocatechin gallate
Catalog No. A10005 Antioxidant, antiangiogenic, antitumor agent(-)-Epigallocatechin gallate是一种从绿茶中分离出来的强效抗氧化剂多酚类黄酮。 了解更多 -
Decitabine
Catalog No. A10292 DNA Methyltransferase 抑制剂Decitabine是一种次甲基化剂，它通过抑制DNA甲基转移酶来使DNA次甲基化。 了解更多 -
Azacitidine(Vidaza)
Catalog No. A10105 DNMT 抑制剂Azacitidine (Vidaza)是DNA和RNA中使用的胞嘧啶核苷的化学类似物，主要用于治疗骨髓增生异常综合症（MDS）。 了解更多 -
SGI-110 (Guadecitabine)
Catalog No. A12744 -
SGI 1027
Catalog No. A14120 -
Procainamide HCl
Catalog No. A14240 -
RG108
Catalog No. A13054 -
O6-Benzylguanine
Catalog No. A13706 -
Nanaomycin A
Catalog No. A13477 -
Lomeguatrib
Catalog No. A12785 -
6-Methyl-5-azacytidine
Catalog No. A13391 -
O6BTG-octylglucoside
Catalog No. A11432 MGMT inhibitorO6BTG-octylglucoside is a potent O6-methylguanine-DNAmethyl-transferase (MGMT) inhibitor, with IC50s of 32 nM in vitro (cell extracts) and 10 nM in HeLa S3 cells. 了解更多 -
OG-L002
Catalog No. A13246 -
Tranylcypromine hydrochloride
Catalog No. A13358 LSD1/BHC110 & MAO 抑制剂Tranylcypromine hydrochloride是一种非选择性的MAO-A/B抑制剂。 了解更多 -
GSK2879552
Catalog No. A15547 -
SP2509 (HCI-2509)
Catalog No. A14443 LSD1 抑制剂SP2509 (HCI-2509)是一种新型组蛋白脱甲基酶LSD1（KDM1A）拮抗剂，IC50为13 nM。对MAO-A和MAO-B没有抑制作用。 了解更多 -
ORY-1001 (RG-6016)
Catalog No. A15893 LSD1 抑制剂ORY-1001 (RG-6016)是一种活性的选择性赖氨酸脱甲基酶LSD1/KDM1A抑制剂，IC50 <20 nM，对相关FAD依赖性氨氧化酶具有高选择性。 了解更多 -
CPI 455
Catalog No. A16178 -
2,4-Pyridinedicarboxylic Acid
Catalog No. A16372 KDM 抑制剂2,4-Pyridinedicarboxylic Acid是针对JMJD2A（KDM4A），KDM4C，KDM4E（IC50、1.4μM），KDM5B（IC50、3μM），KDM6A和 其他的2-氧合酶。 了解更多 -
CBB1007
Catalog No. A16374 -
GSK467
Catalog No. A18807 KDM5B (JARID1B or PLU1) inhibitorGSK467 is a potent and selective inhibitor of KDM5 (also known as JARID1) with a Ki of 10 nM, shows 180-fold selectivity for KDM4C and no measurable inhibitory effects toward KDM6 or other Jumonji family members. GSK467 exploits unique binding modes. 了解更多 -
T-3775440 hydrochloride
Catalog No. A18340 LSD1 inhibitorT-3775440 (hydrochloride) is an irreversible lysine-specific histone demethylase (LSD1) inhibitor with an IC50 value of 2.1 nM. 了解更多 -
QC6352
Catalog No. A19477 -
NCGC00244536
Catalog No. A13025 -
Toxoflavin
Catalog No. A12174 KDM4A inhibitorToxoflavin (Xanthothricin) is an antagonist of transcription factor 4 (TCF4)/β-catenin complex, also acts as an inhibitor of KDM4A, with antitumor activity. 了解更多 -
ORY-1001(trans)
Catalog No. A21622 KDM1A/LSD1 inhibitorORY-1001 trans is a selective irreversible lysine (K)-specific demethylase 1A (KDM1A/LSD1) inhibitor. 了解更多 -
GSK-LSD1 dihydrochloride
Catalog No. A21815 LSD1 inhibitorGSK-LSD1 dihydrochloride is a potent, selective and irreversible lysine specific demethylase 1 (LSD1) inhibitor with an IC50 of 16 nM. 了解更多 -
C646
Catalog No. A12815 -
GSK2801
Catalog No. A14015 -
GSK1324726A (I-BET726)
Catalog No. A14133 BET 抑制剂GSK1324726A (I-BET726)是一种新型、高效、选择性的BET蛋白小分子抑制剂，对BRD2（IC50 = 41 nM）、BRD3（IC50 = 31 nM）和BRD4（IC50 = 22 nM）具有高度的亲和力。 了解更多 -
GSK 525768A
Catalog No. A14134 GSK 525768A是GSK 525762A的对映体化合物，GSK 525762A是一种有效的小分子抑制剂，可破坏溴多糖BET家族（Brd2、Brd3和Brd4）的功能；GSK 525768A对BET没有活性。 了解更多
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