“Lurasidone HCl”的搜索结果

产品 51 到 100 共 112个

每页
页面:
  1. 1
  2. 2
  3. 3

设置降序顺序
  1. Adiphenine HCl

    Catalog No. A11716
    Quick View
    AChR抑制剂
    Adiphenine Hydrochloride是烟碱受体抑制剂,IC50为15μM,用作解痉药物。 了解更多
  2. Bay 65-1942 HCl

    Catalog No. A11338
    Quick View
    IKKβ kinase 抑制剂
    Bay 65-1942 HCl是选择性靶向IKKβ激酶活性的ATP竞争性抑制剂。 了解更多
  3. Dorzolamide HCL

    Catalog No. A10333
    Quick View
    carbonic anhydrase 抑制剂
    Dorzolamide HCl是一种碳酸酐酶抑制剂。它是一种抗青光眼剂,以滴眼剂的形式局部使用。盐酸度尔佐胺用于降低开角型青光眼和高眼压患者的眼内压升高。 了解更多
  4. Fasudil HCl (HA-1077)

    Catalog No. A10381
    Quick View
    ROCK 抑制剂
    Fasudil HCl (HA-1077)是一种环状核苷酸依赖性蛋白激酶抑制剂和Rho相关激酶抑制剂(IC50 = 10.7μM)。 了解更多
  5. BMS-1166 hydrochloride

    Catalog No. A21481
    Quick View
    PD-1/PD-L1 interaction inhibitor
    BMS-1166 hydrochloride is a potent PD-1/PD-L1 interaction inhibitor with an IC50 of 1.4 nM. BMS-1166 antagonizes the inhibitory effect of PD-1/PD-L1 immune checkpoint on T cell activation. 了解更多
  6. CSRM617 Hydrochloride

    Catalog No. A18438
    Quick View
    OC2 inhibitor
    CSRM617 Hydrochloride is an inhibitor of the transcription factor ONECUT2 (OC2), thereby suppressing metastasis in mice. 了解更多
  7. Molindone hydrochloride

    Catalog No. A17647
    Quick View
    MAO inhibitor
    Molindone HCl is a D2 dopamine receptor antagonist. It also acts as a MAO inhibitor. 了解更多
  8. Proadifen HCl

    Catalog No. A17386
    Quick View
    Cytochrome P450 inhibitor
    Proadifen hydrochloride is a Cytochrome P450 inhibitor (IC50 = 19μM). 了解更多
  9. T-3775440 hydrochloride

    Catalog No. A18340
    Quick View
    LSD1 inhibitor
    T-3775440 (hydrochloride) is an irreversible lysine-specific histone demethylase (LSD1) inhibitor with an IC50 value of 2.1 nM. 了解更多
  10. Tacrine HCl Hydrate

    Catalog No. A16970
    Quick View
    AChE and BChE 抑制剂
    Tacrine hydrochloride hydrate是乙酰(AChE)和丁酰胆碱酯酶(BChE)的抑制剂,IC50分别为31 nM和25.6 nM。 了解更多
  11. Pazopanib HCl (GW786034)

    Catalog No. A10699
    Quick View
    VEGFR/PDGFR/FGFR 抑制剂
    Pazopanib HCl (GW786034)是VEGFR-1,VEGFR-2,VEGFR-3,PDGFR-a/β和c-kit的有效且选择性的多靶点酪氨酸激酶抑制剂,可阻止肿瘤生长并抑制血管生成。 了解更多
  12. Irinotecan HCl Trihydrate (Campto)

    Catalog No. A10479
    Quick View
    Topoisomerase 抑制剂
    Irinotecan (CPT 11)是喜树碱家族的一种化合物,是参与细胞DNA复制和转录的拓扑异构酶1的抑制剂。 了解更多
  13. Lexibulin dihydrochloride

    Catalog No. A21774
    Quick View
    tubulin polymerisation inhibitor
    Lexibulin 2Hcl (CYT-997 2Hcl) is a potent tubulin polymerisation inhibitor with IC50 of 10-100 nM in cancer cell lines; with potent cytotoxic and vascular disrupting activity in vitro and in vivo. 了解更多
  14. Azacosterol

    Catalog No. A13295
    Quick View
    24-DHCR 抑制剂
    Azacosterol可作为24-脱氢胆固醇还原酶(24-DHCR)的抑制剂,可防止去甾醇形成胆固醇。 了解更多
  15. K-7174 2HCl

    Catalog No. A15446
    Quick View
    Cell adhesion 抑制剂
    K-7174 dihydrochloride是一种新型的细胞粘附抑制剂;抑制由IL-1beta或TNF-alpha诱导的血管细胞粘附分子1(VCAM-1)的表达。 了解更多
  16. KX2-391 2HCl

    Catalog No. A11471
    Quick View
    Src 抑制剂
    Tirbanibulin dihydrochloride是首个靶向Src肽底物位点的临床Src抑制剂(拟肽类),在癌细胞系中GI50为9-60 nM。 了解更多
  17. AT7867 2HCl

    Catalog No. A15006
    Quick View
    Akt 抑制剂
    AT7867 dihydrochloride是一种有效的ATP竞争性Akt1/2/3和p70S6K/PKA抑制剂,IC50分别为32 nM/17 nM/47 nM和85 nM/20 nM,在AGC激酶家族之外几乎没有活性。 了解更多
  18. RN-1 2HCl

    Catalog No. A14344
    Quick View
    MAO 抑制剂
    RN-1 2HCl对LSD1的选择性优于单胺氧化酶(MAO)-A和MAO-B(在辣根过氧化物酶偶联测定中,IC50值分别为70 nM,0.51和2.79 μM)。 了解更多
  19. Glycyl-H 1152 2HCl

    Catalog No. A13659
    Quick View
    ROCK 抑制剂
    Glycyl-H 1152 2HCl是一种选择性有效的ROCK抑制剂(ROCKII,Aurora A,CAMKII,PKG,PKA和PKC的IC50值分别为0.0118、2.35、2.57、3.26,> 10和> 10 uM。) 了解更多
  20. Dorsomorphin 2HCl

    Catalog No. A13720
    Quick View
    BMP 抑制剂
    Dorsomorphin 2HCl (BML-275)是BMP信号传导的选择性小分子抑制剂,可促进胚胎干细胞的心肌发生。Dorsomorphin通过抑制骨形态发生蛋白信号转导逆转乳腺癌起始细胞的间质表型。 了解更多
  21. Puromycin 2HCl

    Catalog No. A14268
    Quick View
    protein synthesis 抑制剂
    Puromycin 2HCl是一种氨基核苷抗生素,可作为蛋白质合成抑制剂。 了解更多
  22. TAS 103 2HCl

    Catalog No. A14141
    Quick View
    topoisomerase I/II 抑制剂
    TAS 103 2HCl,也称为BMS-247615,是一种喹啉衍生物,在鼠和人肿瘤模型中显示出抗肿瘤活性。 了解更多
  23. GBR-12935 2HCl

    Catalog No. A11937
    Quick View
    DAT and SLC6A2 抑制剂
    GBR-12935 dihydrochloride是一种有效的选择性多巴胺再摄取抑制剂。 了解更多
  24. H 89 2HCl

    Catalog No. A11935
    Quick View
    PKA 抑制剂
    H 89 dihydrochloride是一种可渗透细胞的,选择性的,可逆的,具有ATP竞争性的有效蛋白激酶抑制剂。 了解更多
  25. BMS-790052 2HCl

    Catalog No. A11336
    Quick View
    NS5A 抑制剂
    BMS-790052 2HCl是一种NS5A抑制剂,用于治疗丙型肝炎病毒(HCV)感染。 了解更多
  26. Vanoxerine 2HCl (GBR-12909)

    Catalog No. A10725
    Quick View
    dopamine re-uptake 抑制剂
    Vanoxerine 2HCl (GBR-12909)是哌嗪衍生物,是一种有效的、选择性的多巴胺摄取(dopamine uptake)抑制剂。 了解更多
  27. Vatalanib (PTK787) 2HCl

    Catalog No. A10967
    Quick View
    VEGFR 抑制剂
    Vatalanib (PTK787) 2HCl是一种小分子蛋白激酶抑制剂,可抑制抑制所有已知VEGF受体以及血小板衍生的生长因子受体β和c-kit的血管生成,但对VEGFR-2的选择性最高。 了解更多
  28. Y-27632 2HCl

    Catalog No. A11001
    Quick View
    ROCK 抑制剂
    Y-27632是一种Rho相关的线圈激酶(ROCK)抑制剂,可提高人类胚胎干细胞(hESCs)的克隆效率。比对其他激酶包括PKC,cAMP依赖性蛋白激酶,MLCK和PAK的作用强200多倍。 了解更多
  29. MK-2206 2HCl

    Catalog No. A10003
    Quick View
    AKT 抑制剂
    MK-2206 2HCl是Akt1/2/3的高选择性抑制剂,IC50分别为8 nM/12 nM/65 nM。 了解更多
  30. Nefazodone hydrochloride

    Catalog No. A17622
    Quick View
    5-HT2 receptors inhibitor
    Nefazodone HCl is an inhibitor of 5-HT2 receptors, SERT, NET, and hERG K+ channels used to treat mood disorders. It decreases immobility time in the forced swim test. 了解更多
  31. Tacrine HCl

    Catalog No. A17374
    Quick View
    AChE & butyrylcholinesterase inhibitor
    Tacrine is a derivative of aminoacridine that functions as an inhibitor of both acetylcholinesterase (AChE) and butyrylcholinesterase (IC50s = 31 and 26.5 nM, respectively). 了解更多
  32. IPI-504 (Retaspimycin HCl)

    Catalog No. A11269
    Hsp90 抑制剂
    IPI-504 (Retaspimycin HCl)是新型的,有效的热休克蛋白90(Hsp90)抑制剂。 了解更多
  33. Nepicastat HCl

    Catalog No. A11172
    Quick View
    DBH 抑制剂
    Nepicastat HCl是多巴胺β-羟化酶的抑制剂,该酶催化多巴胺向去甲肾上腺素的转化。 了解更多
  34. Benazepril HCl

    Catalog No. A10123
    Quick View
    RAAS 抑制剂
    Benazepril hydrochloride是一种非肽血管紧张素转化酶(ACE)抑制剂。降低自发性高血压大鼠的血压和心肌肥大。 了解更多
  35. PD153035 (HCl salt)

    Catalog No. A10702
    Quick View
    EGFR 抑制剂
    PD153035 (HCl salt)是EGFR酪氨酸激酶活性的极其有效和特异的抑制剂。 了解更多
  36. Piperidolate hydrochloride

    Catalog No. A18144
    Quick View
    antimuscarinic
    Piperidolate hydrochloride is an antimuscarinic, Also a potential inhibitor of human glutathione transferase P1-1. 了解更多
  37. Promazine hydrochloride

    Catalog No. A17638
    Quick View
    D2DR inhibitor
    Promazine Hydrochloride is a phenothiazine compound and D2DR inhibitor. Promazine Hydrochloride has been employed in studies investigating dopamine-stimulated glycosylation of brain proteins in vitro. It has actions similar to chlorpromazine but with less antipsychotic activity. 了解更多
  38. AX-024 hydrochloride

    Catalog No. A18332
    Quick View
    TNF receptor inhibitor
    AX-024 is an orally available inhibitor of the TCR-Nck interaction that selectively inhibits TCR-triggered T cell activation (IC50 value 1 nM). Inhibiting an immediate TCR signal has promise for treating a broad spectrum of human T cell-mediated autoimmune and inflammatory diseases. 了解更多
  39. Pargyline hydrochloride

    Catalog No. A17288
    Quick View
    MAO inhibitor
    Pargyline hydrochloride is an irreversible inhibitor of monoamine oxidase (MAO) that is used clinically to treat moderate hypertension. 了解更多
  40. Pitofenone Hydrochloride

    Catalog No. A17053
    Quick View
    Antispasmodic Agent
    Pitofenone Hydrochloride是抗痉化合物。它是乙酰胆碱酯酶活性的有效抑制剂。 了解更多
  41. ASTX-660

    Catalog No. A16996
    Quick View
    XIAP 抑制剂
    ASTX660是X染色体连锁的凋亡蛋白抑制剂(XIAP)和细胞IAP 1(cIAP1)的口服生物利用型非拟肽拮抗剂,具有潜在的抗肿瘤和促凋亡活性。1799328-86-1 (free base) 1799328-50-9 (HCl) 1799328-90-7 (mesylate) 1799328-88-3 (sulfate) 了解更多
  42. AN3365

    Catalog No. A16329
    Quick View
    leucyl-tRNA synthetase 抑制剂
    AN3365是一种有效的,选择性的亮氨酰tRNA合成酶抑制剂。 了解更多
  43. TGR-1202 hydrochloride (Umbralisib HCl)

    Catalog No. A16278
    Quick View
    PI3Kδ 抑制剂
    TGR-1202 hydrochloride是一种口服的下一代PI3Kδ抑制剂,在基于酶和细胞的测定中抑制PI3Kδ活性,IC50和EC50值分别为22.2和24.3 nM。 了解更多
  44. BI 1467335 (PXS 4728A)

    Catalog No. A16082
    Quick View
    SSAO/VAP-1 抑制剂
    BI 1467335 (PXS 4728A)是一种非常有效和高度选择性的化合物,正在开发中,用于治疗心脏代谢疾病,例如肝脏相关疾病非酒精性脂肪性肝炎(NASH)。 了解更多
  45. MRT68921

    Catalog No. A15880
    Quick View
    Autophagy ULK1/2 抑制剂
    MRT68921是一种有效的双重自噬激酶ULK1/2抑制剂,IC50分别为2.9 nM和1.1 nM。 了解更多
  46. Asenapine HCl

    Catalog No. A15002
    Quick View
    adrenergic receptor/5-HT receptor 抑制剂
    Asenapine hydrochloride抑制肾上腺素能受体(α1,α2A,α2B,α2C)的Ki为0.25-1.2 nM,还抑制5-HT受体(1A,1B,2A,2B,2C,5A,6、7),Ki为0.03- 4.0 nM。 了解更多
  47. Vandetanib HCl

    Catalog No. A15271
    Quick View
    VEGFR 抑制剂
    Vandetanib hydrochloride是一种有效的VEGFR2抑制剂,IC50为40 nM。 了解更多
  48. TG 100801 HCl

    Catalog No. A15261
    Quick View
    VEGFr2 抑制剂
    TG 100801 HCl是TG 100572(HY-10184)的前药,TG 100572是一种多靶点激酶抑制剂,可抑制选择性生长因子受体酪氨酸激酶和Src家族激酶,IC50值为2/7/2/1/0.5 nM或VEGFR1/VEGFR2/FGFR1/Src/Fyn kianse分别。 了解更多
  49. TG 100572 HCl

    Catalog No. A15260
    Quick View
    VEGFR2/Src kinase 抑制剂
    TG 100572 HCl是一种多靶点激酶抑制剂,可抑制选择性生长因子受体酪氨酸激酶和Src家族激酶,分别对VEGFR1/VEGFR2/FGFR1/Src/Fyn kianse的IC50值为2/7/2/1/0.5 nM。 了解更多
  50. SB-505124 HCl

    Catalog No. A15232
    Quick View
    TGF-β Receptors 抑制剂
    SB-505124 Hydrochloride是激活素受体样激酶(ALKS)的抑制剂。 了解更多

产品 51 到 100 共 112个

每页
页面:
  1. 1
  2. 2
  3. 3

设置降序顺序
Rewards