微信关注
China
Total item
Cart Subtotal
￥ 0.00 “Lurasidone HCl”的搜索结果
-
Almorexant HCl
Catalog No. A14286 OX1/OX2 拮抗剂Almorexant HCl是一种活性双重食欲素受体拮抗剂，对OX1和OX2受体3的IC50为6.6 nM和3.4 nM。 了解更多 -
CX-6258 HCl
Catalog No. A14275 Pan-PIM kinase 抑制剂CX-6258 HCl是一种有效的口服泛Pim激酶抑制剂，对Pim1，Pim2和Pim3的IC50为5 nM，25 nM和16 nM。 了解更多 -
NSC-23766 HCl
Catalog No. A13975 Rac GTPase 抑制剂NSC 23766是Rac特异性GEF TrioN和Tiam 1（IC50 = 50 uM）引起的Rac1激活的细胞可渗透性可逆抑制剂。 了解更多 -
PX-478 HCl
Catalog No. A14319 HIF-1alpha 抑制剂PX-478 HCl是HIF-1alpha抑制剂，也是具有潜在抗肿瘤活性小分子。PX-478对已建立的人类肿瘤异种移植物具有出色的活性，可提供具有HIF-1水平正相关的延长的生长延迟的肿瘤消退。PX-478是高度水溶性的分子，具有良好的i.v.，i.p.和p.o.抗肿瘤活性。 了解更多 -
Dexmedetomidine HCl
Catalog No. A11846 alpha2-adrenoceptor 激动剂Dexmedetomidine hydrochloride是美托咪啶的活性异构体，它充当有效的，高度选择性的α2-AR（α2-肾上腺素受体）激动剂。 了解更多 -
Edivoxetine HCl
Catalog No. A13865 -
SBE 13 HCl
Catalog No. A14426 PLK 抑制剂SBE 13 HCl是PLK1的选择性抑制剂，对于PLK1，PLK3和PLK2，IC 50值分别为200pM，875nM和66μM。 了解更多 -
Afuresertib HCl
Catalog No. A13030 AKT 抑制剂?Afuresertib HCl，也称为GSK2110183，是具有潜在抗肿瘤活性的丝氨酸/苏氨酸蛋白激酶Akt（蛋白激酶B）的生物利用抑制剂。它结合并抑制Akt的活性，这可能导致PI3K/Akt信号传导途径的抑制和肿瘤细胞的增殖以及肿瘤细胞凋亡的诱导.PI3K/Akt信号传导途径的激活通常与肿瘤发生有关，PI3K/Akt信号传导失调可能有助于肿瘤对多种抗肿瘤药的耐药性。 了解更多 -
TRV130 HCl (Oliceridine)
Catalog No. A15444 u-opioid receptor 激动剂TRV130 HCl (Oliceridine)是一种新型的μ-opioid 受体（MOR）G蛋白偏向配体。诱导强大的G蛋白信号传导（pEC50 = 8.1），效力和功效与吗啡相似，但β-arrestin募集和受体内在化作用要低得多。 了解更多 -
Pardoprunox HCl (SLV-308)
Catalog No. A11538 Pardoprunox HCl (SLV-308)是一种抗帕金森病药物，是多巴胺受体D2、D3和5-HT1A激动剂，用于治疗帕金森病。 了解更多 -
RAD1901 HCl salt
Catalog No. A15990 SERD/SERMRAD1901 HCl salt是口服的选择性雌激素受体降解剂（SERD）和选择性雌激素受体调节剂（SERM），具有潜在的抗肿瘤活性和类似雌激素的活性。 了解更多 -
APS-2-79 HCl
Catalog No. A16175 KSR/Ras 抑制剂APS-2-79 HCl，稳定KSR（Ras激酶抑制剂）失活状态并拮抗致癌性Ras信号（IC50值为120 nM，对抗KSR2的ATP-生物素探针标记）的小分子。 了解更多 -
A-438079 HCl
Catalog No. A12597 P2X7 receptor 拮抗剂A-438079 HCl是一种竞争性P2X7受体拮抗剂（抑制人重组P2X7细胞系中Ca2+流入的pIC50 = 6.9）。在其他P2受体上没有活性（IC50 > 10 uM）。 了解更多 -
Ruboxistaurin (LY333531 HCl)
Catalog No. A16604 PKCβ1 and PKCβ2 抑制剂LY333531是一种特异性β-蛋白激酶C的抑制剂。竞争性和可逆性抑制PKCβ1和PKCβ2，IC50值分别为4.7和5.9 nM。 了解更多 -
AZD1208 HCl
Catalog No. A16927 -
RS 17053 HCl
Catalog No. A16885 α1A 拮抗剂RS 17053 HCl是α1A受体拮抗剂，对α1A受体具有很高的亲和力（pKi和pA2估计为9.1-9.9），选择性比α1B和α1D亚型高30-100倍（pKi和pA2估计为7.7- 7.8）。 了解更多 -
Desformylflustrabromine HCl
Catalog No. A17103 Desformylflustrabromine HCl是α4β2的正变构调节剂，也是肌肉型nAChR抑制剂。 了解更多 -
Anavex2-73 HCl
Catalog No. A17145 -
-
最新产品
TCS-OX2-29 HCl
Catalog No. A17136 -
-
Procyclidine HCl
Catalog No. A17371 Muscarinic antagonistProcyclidine hydrochloride is a muscarinic antagonist that crosses the blood-brain barrier and is used in the treatment of drug-induced extrapyramidal disorders and in Parkinsonism. 了解更多 -
-
最新产品
SAR-7334 HCl
Catalog No. A17237 TRPC6 inhibitorSAR7334 is a novel, highly potent and bioavailable inhibitor of TRPC6 channels that opens new opportunities for the investigation of TRPC channel function in vivo. SAR7334 inhibited TRPC6, TRPC3 and TRPC7-mediated Ca(2+) influx into cells with IC50 s of 9.5, 282 and 226 nM, whereas TRPC4 and TRPC5-mediated Ca(2+) entry was not affected. 了解更多 -
-
Ractopamine HCl
Catalog No. A17372 beta-Adrenergic agonistRactopamine HCl is a beta-Adrenergic agonist. It acts by being a full agonist at the TAAR1. 了解更多 -
Acecainide HCl
Catalog No. A22660 Class III antiarrhythmic agentAcecainide, also known as N-acetylprocainamide and ASL 601, is the N-acetylated metabolite of procainamide. Acecainide is a Class III antiarrhythmic agent. It can be given either intravenously or orally, and is eliminated primarily by renal excretion. 了解更多 -
MK-212 HCl
Catalog No. A22531 MK 212 hydrochloride is a 5-HT receptor agonist; displays selectivity for 5-HT2C over 5-HT2A (IC50 values are 0.028 and 0.42 μM for human 5-HT2C and 5-HT2A receptors expressed in HEK293 cells respectively). 了解更多 -
AVN-101 HCl
Catalog No. A22498 5-HT7 receptor antagonistAVN-101 is a very potent 5-HT7 receptor antagonist, with slightly lesser potency toward 5-HT6, 5-HT2A, and 5HT-2C receptors. It is a milti-target drug candidate for the treatment of CNS disorders. 了解更多 -
UK-371804 HCl
Catalog No. A22379 uPA inhibitorUK-371804 is a potent and selective urokinase-type plasmogen activator (uPA) inhibitor with excellent enzyme potency (Ki=10 nM) and selectivity profile (4000-fold versus tPA and 2700-fold versus plasmin). 了解更多 -
SEL24-B489 HCl
Catalog No. A22203 -
Prexasertib HCl
Catalog No. A22156 ATP-competitive CHK1 inhibitorPrexasertib (LY2606368) is an ATP-competitive CHK1 inhibitor with a Ki value of 0.9 nmol/L. For CHK2 and RSK, its IC50 values are 8 nM and 9 nM respectively in cell-free assay. 了解更多 -
PD 0332991 HCl (Palbociclib)
Catalog No. A10701 CDK 4/6 抑制剂PD 0332991 HCl (Palbociclib)是一种高度选择性的CDK4/6抑制剂，它对CDK1/2/5，EGFR，FGFR，PDGFR，InsR等没有抑制活性，具有潜在的抗肿瘤活性。 了解更多 -
Gemcitabine HCl (Gemzar)
Catalog No. A10423 DNA/RNA Synthesis 抑制剂Gemcitabine HCl (Gemzar)是一种DNA synthesis抑制剂，作用于PANC1，MIAPaCa2，BxPC3和Capan2细胞，通过在癌细胞dna复制过程中取代核酸的一个组成部分，防止肿瘤生长。 了解更多 -
Flavopiridol HCl
Catalog No. A11045 -
Topotecan HCl (Hycamtin)
Catalog No. A10939 -
ADL5859 HCl
Catalog No. A11072 Opioid Receptor 激动剂ADL5859 HCl是高效的选择性δ阿片受体激动剂，Ki值为0.84 nM，ED50值为20 nM。 了解更多 -
Cerubidine (Daunorubicin HCl, Rubidomycin HCl)
Catalog No. A10194 Topoisomerase 抑制剂Cerubidine (Daunorubicin HCl,Rubidomycin HCl)通过插入和抑制大分子生物合成与DNA相互作用。这抑制了拓扑异构酶II的进程，该酶使DNA中的超螺旋松弛以进行转录。 了解更多 -
GW3965 HCl
Catalog No. A11204 -
Idarubicin HCl
Catalog No. A10465 Topoisomerase 抑制剂Idarubicin HCl是蒽环类抗生素，是一种比柔红霉素具有更高DNA结合能力和更大细胞毒性的抗白血病药物。 了解更多 -
Alfuzosin HCl
Catalog No. A10052 Alfuzosin HCl是用于治疗良性前列腺增生（BPH）的α1受体拮抗剂。 它通过放松前列腺和膀胱颈的肌肉来起作用，使其更容易排尿。 了解更多 -
AT7519 HCl
Catalog No. A11313 -
CGS 21680 HCl Hydrate
Catalog No. A11619 -
Anamorelin HCl
Catalog No. A12345 Anamorelin HCl目前正在开发中，是口服活性的饥饿素受体（ghrelin receptor）激动剂。用于治疗与恶病质/厌食症相关的非小肺癌。 了解更多 -
Nebivolol HCl
Catalog No. A10630 Nebivolol hydrochloride是β1-肾上腺素受体的高度选择性拮抗剂（Ki = 0.88 nM，β2-肾上腺素受体Ki = 48 nM）。 了解更多 -
Adrenalone HCl
Catalog No. A11807 -
Ivabradine HCl (Procoralan)
Catalog No. A11868 Ivabradine Hydrochloride,也称为S-16257，是缓动剂伊伐布雷定的盐酸盐制剂。 了解更多 -
Fexofenadine HCl
Catalog No. A11859 COX 抑制剂/histamine H1 receptor 激动剂Fexofenadine Hydrochloride是一种抗组胺药，可抑制Cox-1，Cox-2，并且是组胺H1受体激动剂，IC50为246 nM。 了解更多
联系我们
United StatesAdooq Bioscience
Toll Free: (866) 930-6790
Fax: +1-323-606-8156
Email: sales@adooq.com
Not your Region? View all Distributors
最近查看过的产品
FILTER BY:
购物选项
- 分类
-
- Epigenetics (11)
- Apoptosis (3)
- PI3K / Akt / mTOR (7)
- Protein Tyrosine Kinases (9)
- Angiogenesis (10)
- MAPK (1)
- JAK / Stat (6)
- Cell Cycle (13)
- DNA Damage (16)
- Cell Metabolism (18)
- Autophagy Signaling (3)
- Immunology & Inflammation (5)
- GPCR / G Protein (99)
- NF-kB/IkB (3)
- TGF-β / Smad (9)
- Neuronal Signaling (20)
- Proteases (3)
- Microbiology (7)
- Stem Cells / Wnt (1)
- Membrane Transporters/Ion Channels (16)
- Endocrinology / Hormones (5)
- Others (31)
- Natural Products (4)
- Ready to Use Solution (64)
- Products On Sale (88)
- Recombinant Proteins (1)
- Monoclonal Antibodies (1)
- COVID-19 Related Products (1)
- 作用机制
-
- Inhibitor (抑制剂) (112)
- Agonist (激动剂) (36)
- Antagonist (拮抗剂) (50)
- Activator (激活剂) (4)
- Modulator (调节剂) (4)
- Blocker (阻断剂) (11)
- Degrader (降解剂) (1)
- Stabilizer (稳定剂) (1)
- 靶点
-
- AKT1 (1)
- AKT2 (1)
- AKT3 (1)
- Aurora A (1)
- Carbonic Anhydrase I (1)
- Carbonic Anhydrase II (1)
- Carbonic Anhydrase IV (1)
- CDK4 (1)
- COX-1 (1)
- COX-2 (1)
- CXCL12 (1)
- CXCR4 (2)
- DNMT (1)
- EGFR (1)
- EZH2 (1)
- FTase (1)
- HDAC6 (1)
- Histamine H1 receptor (1)
- JAK1 (1)
- JAK3 (1)
- KDM1A (LSD1) (1)
- MAO-A (1)
- MAO-B (1)
- p53 (2)
- Pim1 (2)
- Pim2 (2)
- Pim3 (2)
- SIRT1 (1)
ADOOQ 产品质量保证
We promise all products to perform as described.