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Cell Metabolism

产品 1 到 50 共 394个

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  1. RMC-4550
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    RMC-4550

    Catalog No. A18893
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    SHP2 inhibitor
    RMC-4550 is a potent, selective and allosteric inhibitor of SHP2, with an IC50 of 0.583 nM. 了解更多
  2. SHP394
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    SHP394

    Catalog No. A18613
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    SHP2 inhibitor
    SHP394 is an orally efficacious protein tyrosine phosphatase SHP2 inhibitor with an IC50 of 23 nM. 了解更多
  3. SHP2 IN-1
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    SHP2 IN-1

    Catalog No. A19099
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    SHP2 (PTPN11) inhibitor
    SHP2 IN-1 (compound 13) is an allergic inhibitor of SHP2 (PTPN11), with an IC50 of 3 nM. 了解更多
  4. SHP099 hydrochloride
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    SHP099 hydrochloride

    Catalog No. A21762
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    SHP2 inhibitor
    SHP099 hydrochloride is a potent, selective and orally available SHP2 inhibitor with an IC50 of 70 nM. 了解更多
  5. Celgosivir
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    Celgosivir

    Catalog No. A13118
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    alpha-glucosidase I 抑制剂
    Celgosivir是一种用于潜在治疗HCV感染的α-葡萄糖苷酶I抑制剂。 了解更多
  6. Deoxynojirimycin
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    Deoxynojirimycin

    Catalog No. A14383
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    glucosidase I/II 抑制剂
    Deoxynojirimycin是马耳他酶-葡糖淀粉酶（α-葡糖苷酶I和II）抑制剂。它干扰N-连接的糖基化。 了解更多
  7. Voglibose
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    Voglibose

    Catalog No. A14945
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    alpha-glucosidase 抑制剂
    Voglibose是缬氨酰胺的N取代衍生物，对α-葡萄糖苷酶具有出色的抑制活性，并且对高血糖症和由高血糖症引起的各种疾病具有抗药性。 了解更多
  8. ND-646
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    ND-646

    Catalog No. A20079
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    ACC inhibitor
    ND-646 is an orally bioavailable and steric inhibitor of acetyl-CoA carboxylase (ACC) with IC50s of 3.5 nM and 4.1 nM for recombinant hACC1 and hACC2, respectively. 了解更多
  9. TOFA
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    TOFA

    Catalog No. A12276
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    ACCA inhibitor
    TOFA (RMI14514;MDL14514) is an allosteric inhibitor of acetyl-CoA carboxylase-α (ACCA ). 了解更多
  10. Olumacostat glasaretil
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    Olumacostat glasaretil

    Catalog No. A20840
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    ACC inhibitor
    Olumacostat glasaretil is a small molecule inhibitor of acetyl coenzyme A carboxylase (ACC). 了解更多
  11. PF-05175157
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    PF-05175157

    Catalog No. A21460
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    ACC inhibitor
    PF-05175157 is broad spectrum acetyl-CoA carboxylase (ACC) inhibitor with IC50s of 27.0, 33.0, 23.5 and 50.4 nM for ACC1 (human), ACC2 (human), ACC1 (rat), ACC2 (rat), respectively. 了解更多
  12. CP-640186 hydrochloride
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    CP-640186 hydrochloride

    Catalog No. A21808
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    ACC inhibitor
    CP-640186 hydrochloride is a potent and cell-permeable Acetyl-CoA carboxylase (ACC) inhibitor with IC50s of 53 nM and 61 nM for rat liver ACC1 and rat skeletal muscle ACC2 respectively. 了解更多
  13. Firsocostat
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    Firsocostat

    Catalog No. A21000
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    ACC inhibitor
    Firsocostat (ND-630; GS-0976; NDI-010976) is an acetyl-CoA carboxylase (ACC) inhibitor; inhibits human ACC1 and ACC2 with IC50 values of 2.1 and 6.1 nM, respectively. 了解更多
  14. Triapine
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    Triapine

    Catalog No. A14306
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    Ribonucleotide reductase 抑制剂
    Triapine是一种有效的核糖核苷酸还原酶抑制剂，具有抑制DNA合成的广谱抗肿瘤活性。 了解更多
  15. Didox
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    Didox

    Catalog No. A16304
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    ribonucleotide reductase 抑制剂
    Didox是核糖核苷酸还原酶（RR）的强抑制剂，可通过阻止脱氧核糖核苷酸的产生来干扰DNA的合成和修复，并且数十年来已显示出抗肿瘤作用。 了解更多
  16. PFK15
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    PFK15

    Catalog No. A14287
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    PFKFB3 抑制剂
    PFK15是一种有效的选择性6-磷酸果糖-2-激酶（PFKFB3），IC50为20 nM。 了解更多
  17. PFK-158
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    PFK-158

    Catalog No. A14398
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    PFK-2/FBPase 抑制剂
    PFK-158是6-磷酸果糖-2-激酶/果糖-2,6-双磷酸酶（PFK-2/FBPase）同工型3（PFKFB3）的抑制剂，是3-(3-吡啶基)-1-[4-吡啶基]-2-丙烯-1-酮(3PO)，具有潜在的抗肿瘤活性。 了解更多
  18. 3PO
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    3PO

    Catalog No. A15932
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    PFKFB3 抑制剂
    3PO是PFKFB3（6-磷酸果糖-2-激酶/果糖-2,6-双磷酸酶）抑制剂。 了解更多
  19. AZ-33
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    AZ-33

    Catalog No. A13341
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    LDHA 抑制剂
    AZ33是LDHA抑制剂。 了解更多
  20. C75
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    C75

    Catalog No. A14107
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    FASN 抑制剂
    C75是新型有效的脂肪酸合酶抑制剂（FAS），可作为研究代谢紊乱和癌症中脂肪酸合成的工具。 了解更多
  21. C-75 Trans
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    C-75 Trans

    Catalog No. A15331
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    FASN 抑制剂
    C 75是脂肪酸合酶（FAS）的抑制剂，可减少小鼠的食物摄入量和体重。 了解更多
  22. TVB-3166
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    TVB-3166

    Catalog No. A18763
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    FASN inhibitor
    TVB-3166 is an orally-available, reversible, potent, and selective FASN inhibitor, inducing apoptosis, inhibiting anchorage-independent cell growth under lipid-rich conditions, and inhibiting in-vivo xenograft tumor growth. 了解更多
  23. TVB-3664
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    TVB-3664

    Catalog No. A18829
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    FASN inhibitor
    TVB-3664 is an orally available, reversible, potent, selective and highly bioavailable fatty acid synthase (FASN) inhibitor, with IC50 values of 18 nM and 12 nM for human and mouse cell palmitate synthesis, respectively. TVB-3664 significantly reduces tubulin palmitoylation and mRNA expression. 了解更多
  24. FASN-IN-2
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    FASN-IN-2

    Catalog No. A13063
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    FASN inhibitor
    FASN-IN-2 is a Fatty Acid Synthase (FASN) inhibitor extracted from patent WO2012122391A1, compound 152, has an IC50 of 0.052 μM and an EC50 of 0.072 μM. 了解更多
  25. HS80
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    HS80

    Catalog No. A21615
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    FASN inhibitor
    HS-80 is an enantiomer of Fasnall, which is a selective fatty acid synthase (FASN) inhibitor. HS-80 is able to inhibit the incorporation of tritiated acetate into lipids with an IC50 of 7.13 μM. 了解更多
  26. BMS303141
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    BMS303141

    Catalog No. A13807
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    ATP-citrate lyase 抑制剂
    BMS303141是有效的ATP柠檬酸裂解酶（ACL）抑制剂。BMS303141以8μM的IC50抑制HepG2细胞中的脂质合成，并在鼠类高脂血症模型中降低血浆甘油三酸酯。 了解更多
  27. ETC-1002
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    ETC-1002

    Catalog No. A15815
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    ACL 抑制剂 and AMPK 激活剂
    ETC-1002是一种新颖的，一流的可以降低LDL-C的小分子；肝AMP激活的蛋白激酶（AMPK）的激活剂;对肝ATP-柠檬酸裂解酶也具有有效的抑制活性（IC50 = 29 uM）。 了解更多
  28. Carbidopa
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    Carbidopa

    Catalog No. A10181
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    aromatic-L-amino-acid decarboxylase 抑制剂
    Carbidopa是一种芳香族-L-氨基酸脱羧酶抑制剂，这是一种在L-色氨酸生物合成5-羟色胺和L-DOPA生物合成多巴胺（DA）中重要的酶。 了解更多
  29. PX 12
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    PX 12

    Catalog No. A13831
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    Trx-1 抑制剂
    PX 12抑制缺氧诱导的HIF-1a转录活性（IC50 11 nM）和HT29和MCF-7肿瘤细胞的增殖（IC50分别为1.9和0.9 uM）。 了解更多
  30. CCF642
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    CCF642

    Catalog No. A16122
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    PDI 抑制剂
    CCF642是一种具有抗骨髓瘤活性的新型PDI抑制化合物。 了解更多
  31. KPT 335
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    KPT 335

    Catalog No. A16078
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    SINE 抑制剂
    KPT 335是口服可生物利用的核出口选择性抑制剂（SINE）。 了解更多
  32. KPT276
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    KPT276

    Catalog No. A16341
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    SINE/CRM1 抑制剂
    KPT276是KPT-185的类似物，是核出口（SINE）和CRM1的选择性抑制剂。 了解更多
  33. Eltanexor Z-isomer
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    Eltanexor Z-isomer

    Catalog No. A21786
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    CRM1 inhibitor
    Eltanexor Z-isomer (KPT-8602 Z-isomer) is the less active isomer of KPT-8602. KPT-8602 is a potent CRM1 inhibitor. 了解更多
  34. Leptomycin B
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    Leptomycin B

    Catalog No. A20985
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    nuclear export receptor CRM1 inhibitor
    Leptomycin B (CI 940; LMB) is a potent inhibitor of the nuclear export of proteins. Leptomycin B inactivates CRM1/exportin 1 by covalent modification at a cysteine residue. Leptomycin B is a potent antifungal antibiotic blocking the eukaryotic cell cycle. 了解更多
  35. KPT185
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    KPT185

    Catalog No. A12975
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    CRM1 抑制剂
    KPT185是选择性CRM1抑制剂。KPT-185以100 nM至500 nM的IC50显着抑制白血病细胞增殖，并诱导AML细胞系和原发性AML原始细胞的细胞周期停滞和凋亡。 了解更多
  36. Selinexor (KPT-330)
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    Selinexor (KPT-330)

    Catalog No. A12582
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    CRM1 抑制剂
    CRM1（XPO1）介导的核输出的KPT-330抑制剂在T细胞急性淋巴细胞白血病和急性骨髓性白血病的临床前模型中具有选择性的抗白血病活性。 了解更多
  37. Tipifarnib (Zarnestra)
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    Tipifarnib (Zarnestra)

    Catalog No. A10935
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    FTase 抑制剂
    Tipifarnib (Zarnestra)是一种法尼基转移酶抑制剂，可在激酶途径变得过度活跃之前的翻译后修饰步骤中抑制Ras激酶。 了解更多
  38. FTI 277
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    FTI 277

    Catalog No. A12368
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    FTase 抑制剂
    FTI 277是一种抑制法呢基转移酶(FTase)的抑制剂(IC50 = 0.5 nM)。抑制全细胞的 H-Ras 和 K-Ras 加工(IC50值分别为0.1和10 nM)，破坏mapk的组成型H-Ras特异性激活。在人恶性胶质瘤细胞和许多其他肿瘤细胞系中引起显著的抗增殖作用。 了解更多
  39. LB42708
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    LB42708

    Catalog No. A14020
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    FTase 抑制剂
    LB42708是一种有效的，口服活性和选择性的非肽法呢基转移酶抑制剂（FTase抑制剂）。 了解更多
  40. FTI-277 HCl
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    FTI-277 HCl

    Catalog No. A14439
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    FTase 抑制剂
    FTI-277 HCl是法呢基转移酶（FTase）的抑制剂。一种高效的Ras CAAX拟肽药物，可拮抗H-Ras和K-Ras致癌信号。 了解更多
  41. Lonafarnib (SCH66336)
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    Lonafarnib (SCH66336)

    Catalog No. A12328
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    FPTase 抑制剂
    Lonafarnib (SCH66336)是H-ras、K-ras-4B和N-ras的选择性FPTase抑制剂，IC50分别为1.9 nM、5.2 nM和2.8 nM。 了解更多
  42. L-778123 HCl
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    L-778123 HCl

    Catalog No. A15796
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    FPTase 抑制剂
    L-778123 hydrochloride是FPTase和GGPTase-I双重抑制剂,在酶抑制测定中IC50为2 nM和98 nM。 了解更多
  43. A 922500
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    A 922500

    Catalog No. A11199
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    DGAT-1 抑制剂
    922500是一种二酰基甘油酰基转移酶1（DGAT-1）抑制剂（人和小鼠DGAT-1的IC50值分别为7和24 nM）。 了解更多
  44. PF-04620110
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    PF-04620110

    Catalog No. A11526
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    DGAT1 抑制剂
    PF-04620110是一种有效、选择性的，有口服活性的甘油二酯酰基转移酶-1 (DGAT1) 抑制剂，IC50值为 19 nM。 了解更多
  45. ABT-046
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    ABT-046

    Catalog No. A14984
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    DGAT-1 抑制剂
    ABT-046是一种有效的，选择性的，可口服生物利用的二酰基甘油酰基转移酶1（DGAT-1）抑制剂（IC50 = 8 nM）。 了解更多
  46. DGAT-1 inhibitor 2
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    DGAT-1 inhibitor 2

    Catalog No. A15067
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    DGAT-1 抑制剂
    DGAT-1 inhibitor 2 是有效的DGAT-1抑制剂。 了解更多
  47. AZD7687
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    AZD7687

    Catalog No. A15012
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    DGAT1 抑制剂
    AZD7687是一种有效的选择性DGAT1抑制剂，IC50值为80 nM（hDGAT1）。 了解更多
  48. Xanthohumol
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    Xanthohumol

    Catalog No. A15919
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    COX 抑制剂
    Xanthohumol是一种来自啤酒花的烯丙基查尔酮，可抑制COX-1和COX-2活性并显示化学预防作用。 了解更多
  49. AS1842856
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    AS1842856

    Catalog No. A15871
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    Foxo1 抑制剂
    AS1842856是细胞渗透性抑制剂，可阻断Foxo1的转录活性，IC50为33 nM。它可以直接与活性Foxo1结合，但不能与Ser256磷酸化形式结合。 了解更多
  50. PF 429242
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    PF 429242

    Catalog No. A11230
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    SREBP 抑制剂
    PF 429242是固醇调节元件结合蛋白（SREBP）位点1蛋白酶的可逆竞争性抑制剂。 了解更多

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  1. Cytochrome P450 (29)
  2. PPAR (1)
  3. PDE (71)
  4. HSP (42)
  5. Hydroxylases (12)
  6. Factor Xa (16)
  7. MAO (30)
  8. DHFR (6)
  9. Dehydrogenases (19)
  10. Procollagen C-proteinase (1)
  11. Carbonic Anhydrase (12)
  12. FAAH (11)
  13. 15-PGDH (2)
  14. CETP (6)
  15. Ferroptosis (5)
  16. HMG-CoA Reductase (15)
  17. Isocitrate Dehydrogenase (IDH) (14)
  18. IDO (13)
  19. Lipase (9)
  20. Phospholipases (10)
  21. Lipoxygenase (11)
  22. NAMPT (5)
  23. GLUT (3)
  24. Antimetabolite (3)
  25. Lipid Metabolism (1)
  26. SREBP (2)
  27. LDL (1)
  28. Foxo1 (1)
  29. DGAT (6)
  30. Farnesyl Transferase (6)
  31. CRM1 (6)
  32. Thioredoxin (2)
  33. Decarboxylase (1)
  34. ACLY (2)
  35. Fatty acid synthase (FASN) (6)
  36. Lactate dehydrogenase A (LDHA) (1)
  37. PFKFB3 (3)
  38. Ribonucleotide Reductase (2)
  39. Acetyl-CoA Carboxylase (6)
  40. Glucosidase (3)
  41. Phosphatase (4)
靶点
  1. 5-lipoxygenase (1)
  2. Carbonic Anhydrase (6)
  3. Carbonic Anhydrase I (3)
  4. Carbonic Anhydrase II (3)
  5. Carbonic Anhydrase IV (2)
  6. Carbonic Anhydrase IX (2)
  7. CETP (4)
  8. COX (1)
  9. COX-1 (1)
  10. COX-2 (2)
  11. DNMT (1)
  12. FTase (4)
  13. HDAC1 (1)
  14. HMG-CoA Reductase (9)
  15. HSP90 (1)
  16. KDM1A (LSD1) (1)
  17. MAO-A (1)
  18. MAO-B (1)
  19. PDE4 (1)
  20. PDE5 (1)
  21. Src (1)
  22. TNF-α (1)
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