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Proteases

产品 251 到 300 共 319个

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  1. E 2012
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    E 2012

    Catalog No. A11393
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    gamma-secretase modulator
    E 2012是γ-secretase抑制剂。 了解更多
  2. BMS 299897
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    BMS 299897

    Catalog No. A12444
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    γ-secretase 抑制剂
    BMS 299897是一种有效的γ-分泌酶抑制剂（IC50 = 12 nM）。在体外抑制Aβ40和Aβ42的形成（IC50值分别为7.4和7.9 nM），并在体内降低脑，血浆和脑脊髓液中的Aβ。 了解更多
  3. Flurizan
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    Flurizan

    Catalog No. A12433
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    gamma-secretase modulator
    Flurizan是一种非甾体抗炎药（NSAID），可抑制γ-分泌酶的活性。 了解更多
  4. FLI-06
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    FLI-06

    Catalog No. A13815
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    Gamma-secretase 抑制剂
    FLI-06是一种Notch抑制剂和早期分泌途径抑制剂。FLI-06以不同于布雷菲德菌素A和杀真菌剂A的方式破坏高尔基体。 了解更多
  5. LY3039478
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    LY3039478

    Catalog No. A13544
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    Notch 抑制剂
    LY3039478是一种新型小分子Notch抑制剂，在大多数测试的肿瘤细胞系中，IC50约为1nM。 了解更多
  6. LY-900009
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    LY-900009

    Catalog No. A14088
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    Notch 抑制剂
    LY-900009是一种有效的Notch抑制剂，IC50值为0.27 nM。 了解更多
  7. IMR-1
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    IMR-1

    Catalog No. A16152
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    Notch 抑制剂
    IMR-1是一类新型的Notch抑制剂，靶向转录激活，IC50为6 umol/L。 了解更多
  8. IMR-1A
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    IMR-1A

    Catalog No. A16223
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    Notch 抑制剂
    IMR-1A是IMR-1的代谢产物。IMR-1是一类新型的Notch抑制剂，靶向转录激活，IC50为6 umol/L。 了解更多
  9. NGP-555
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    NGP-555

    Catalog No. A17051
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    γ-Secretase Modulator
    NGP-555是一种γ-分泌酶调节剂，具有选择性机制，可减少Abeta 42，同时提高较短的Abeta形式，例如Abeta 37和38。 了解更多
  10. BPN-15606
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    BPN-15606

    Catalog No. A18681
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    γ-secretase modulator
    BPN-15606 is a highly potent, orally active γ-secretase modulator (GSM), attenuates the production of Aβ42 and Aβ40 by SHSY5Y neuroblastoma cells with IC50 values of 7 nM and 17nM, respectively. 了解更多
  11. LY2886721
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    LY2886721

    Catalog No. A10543
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    BACE1 抑制剂
    LY2886721是一种有效的，选择性的，口服活性的β位淀粉样蛋白前体蛋白裂解酶 1 (BACE1) 抑制剂。LY2886721是一种新型强效药物，用于治疗阿尔茨海默病的研究。 了解更多
  12. AZD3839
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    AZD3839

    Catalog No. A12825
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    BACE1 抑制剂
    AZD3839是人类BACE1的有效选择性抑制剂，Ki为26.1 nM。 了解更多
  13. AMG-8718
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    AMG-8718

    Catalog No. A14407
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    BACE1 抑制剂
    AMG-8718是一种有效的BACE1抑制剂。 了解更多
  14. Timosaponin b-II
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    Timosaponin b-II

    Catalog No. A14591
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    BACE1 抑制剂
    Timosaponin B-II是知母草（Liliaceae，根茎）的主要活性成分，对脑缺血性损伤具有保护作用。 了解更多
  15. gamma-secretase modulator 3
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    gamma-secretase modulator 3

    Catalog No. A15090
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    gamma-secretase modulator
    gamma-secretase modulator 3 是γ-分泌酶调节剂。 了解更多
  16. Compound W
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    Compound W

    Catalog No. A15296
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    Gamma-secretase modulator
    Compound W是一种γ-分泌酶抑制剂，已被证明可以降低分泌的Aβ42和Nβ25的水平。 了解更多
  17. JLK 6
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    JLK 6

    Catalog No. A15301
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    γ-secretase 抑制剂
    JLK 6是γ-分泌酶的抑制剂，可选择性抑制APP裂解而不影响其他γ-分泌酶介导的途径。 了解更多
  18. MRK 560
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    MRK 560

    Catalog No. A15304
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    γ-secretase 抑制剂
    MRK 560是一种可用的γ-分泌酶抑制剂，能够显着减少大鼠脑和CSF中的Abeta肽，并证实该大鼠可用于评估γ-分泌酶抑制剂对中枢神经系统Abeta的作用（40）体内水平。 了解更多
  19. PF-03084014
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    PF-03084014

    Catalog No. A11259
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    γ-secretase 抑制剂
    PF-03084014是一种可逆和选择性的γ-分泌酶抑制剂，IC50值为6.2 nM。 了解更多
  20. Flurbiprofen Axetil
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    Flurbiprofen Axetil

    Catalog No. A13662
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    gamma-secretase 抑制剂
    Flurbiprofen Axetil是非甾体抗炎药(NSAID)。 了解更多
  21. L-685458
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    L-685458

    Catalog No. A15899
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    γ-secretase 抑制剂
    L-685458是一种有效的A beta PPγ-分泌酶抑制剂，Ki为17 nM。 了解更多
  22. Begacestat (GSI-953)
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    Begacestat (GSI-953)

    Catalog No. A11258
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    γ-secretase 抑制剂
    Begacestat (GSI-953)是一种新型的选择性淀粉样前体蛋白γ-分泌酶的噻吩磺酰胺抑制剂。 了解更多
  23. gamma-secretase modulator 1
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    gamma-secretase modulator 1

    Catalog No. A11425
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    Gamma-secretase modulator
    gamma-secretase modulator 1是γ-分泌酶调节剂，γ-分泌酶调节剂1可用于阿尔茨海默病。 了解更多
  24. gamma-secretase modulator 2
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    gamma-secretase modulator 2

    Catalog No. A11427
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    Gamma-secretase modulator
    Gamma-secretase modulator 2是γ-secretase调节剂，可用于阿尔兹海默。 了解更多
  25. TC-E 5006
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    TC-E 5006

    Catalog No. A13217
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    Gamma-secretase modulator
    TC-E 5006是一种γ-分泌酶调节剂。在体外（EC50 = 390 nM）和体内降低Aβ42水平。 了解更多
  26. Verubecestat (MK-8931)
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    Verubecestat (MK-8931)

    Catalog No. A16113
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    β-secretase/BACE1 抑制剂
    Verubecestat (MK-8931)是一种有效的选择性β-分泌酶抑制剂，是BACE1蛋白抑制剂或Beta-site APP裂解酶1抑制剂。 了解更多
  27. CHF5074
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    CHF5074

    Catalog No. A16214
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    γ-Secretase modulator
    CHF5074是新型的γ-分泌酶调节剂，可减少Aβ42和Aβ40的分泌，IC50分别为3.6和18.4 uM。 了解更多
  28. Z-Ile-Leu-aldehyde
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    Z-Ile-Leu-aldehyde

    Catalog No. A16215
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    γ-Secretase 抑制剂
    Z-Ile-Leu-aldehyde是一种有效的γ-分泌酶抑制剂；Notch信号抑制剂。 了解更多
  29. BACE1-IN-4
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    BACE1-IN-4

    Catalog No. A18462
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    BACE1 inhibitor
    BACE1-IN-4 is a potent and highly selective BACE1 inhibitor, with an IC50 of 3.8 nM and a Ki of 1.9 nM, more selective at BACE1 over BACE2. Anti-Alzheimer??s disease. 了解更多
  30. PF-06751979
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    PF-06751979

    Catalog No. A20066
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    BACE1 inhibitor
    PF-06751979 is a potent, brain penetrant, β-site amyloid precursor protein cleaving enzyme 1 (BACE1) inhibitor with an IC50 of 7.3 nM in BACE1 binding assay. 了解更多
  31. Umibecestat (CNP520)
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    Umibecestat (CNP520)

    Catalog No. A18987
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    BACE-1 inhibitor
    Umibecestat (CNP520) is a beta-site amyloid precursor protein cleaving enzyme-1 (BACE-1) inhibitor with IC50s of 11 nM and 10 nM for human BACE-1 and mouse BACE-1, respectively. 了解更多
  32. Lanabecestat
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    Lanabecestat

    Catalog No. A12282
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    BACE1 inhibitor
    Lanabecestat (AZD3293) is a potent, highly permeable, orally active and blood-brain barrier penetrating BACE1 inhibitor with a Ki of 0.4 nM. 了解更多
  33. BACE1-IN-1
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    BACE1-IN-1

    Catalog No. A12183
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    BACE1 inhibitor
    BACE1-IN-1 is a potent and highly brain penetrant BACE1 inhibitor with IC50s of 32 and 47 nM for human BACE1 and BACE2, respectively. 了解更多
  34. BMS-906024
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    BMS-906024

    Catalog No. A21172
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    gamma secretase inhibitor
    BMS-906024 is an oral and selective gamma secretase inhibitor (GSI) that is a small molecule Notch inhibitor. 了解更多
  35. Compound E
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    Compound E

    Catalog No. A21292
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    γ-secretase inhibitor
    Compound E is a γ-secretase inhibitor. 了解更多
  36. β-Secretase Inhibitor IV
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    β-Secretase Inhibitor IV

    Catalog No. A21346
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    BACE-1 inhibitor
    β-Secretase Inhibitor IV is a potent, cell-active BACE-1 inhibitor with IC50s of 15.6 and 16.3nM under BACE-1 concentrations of 2 nM and 100 pM, respectively. 了解更多
  37. AZD3839 free base
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    AZD3839 free base

    Catalog No. A21606
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    BACE1 inhibitor
    AZD3839 (free base) is a potent and selective BACE1 inhibitor with IC50 of 23.6 uM, about 14-fold selectivity over BACE2, also a β-secretase enzyme inhibitor. 了解更多
  38. PAC-1
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    PAC-1

    Catalog No. A11090
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    Caspase activator
    PAC-1是procaspase-3的激活剂，可诱导癌细胞凋亡，EC50为2.08μM。 了解更多
  39. Apoptosis Activator 2
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    Apoptosis Activator 2

    Catalog No. A11944
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    Apoptosis Activator
    Apoptosis Activator 2 强烈诱导caspase-3激活，PARP裂解和DNA片段化，导致细胞破坏（依赖Apaf-1），IC50为约4μM，对HMEC，PREC或MCF-10A细胞无效。 了解更多
  40. LY573636 (Tasisulam)
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    LY573636 (Tasisulam)

    Catalog No. A13070
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    Apoptosis inducer
    LY573636 (Tasisulam)是一种有效的抗肿瘤剂，在体外和体内引起多种人实体瘤的生长停滞和凋亡。LY573636诱导的凋亡通过线粒体靶向机制发生。 了解更多
  41. Z-FA-FMK
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    Z-FA-FMK

    Catalog No. A14284
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    Irreversible Cysteine Protease 抑制剂
    Z-FA-FMK是不可逆的半胱氨酸蛋白酶抑制剂。 了解更多
  42. 25-hydroxy Cholesterol
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    25-hydroxy Cholesterol

    Catalog No. A13704
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    25-hydroxy Cholesterol是一种衍生自膳食胆固醇的侧链取代氧固醇，可抑制固醇调节元件结合蛋白（SREBPs）的裂解，从而抑制各种细胞类型中的内源性胆固醇合成。 了解更多
  43. Boc-D-FMK
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    Boc-D-FMK

    Catalog No. A15392
    Caspase 抑制剂
    BOC-D-FMK是Caspase-3的新型抑制剂。 了解更多
  44. Emricasan
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    Emricasan

    Catalog No. A11394
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    Caspase inhibitor
    Emricasan is a first-in-class caspase inhibitor in clinical trials for the treatment of liver diseases. 了解更多
  45. Z-YVAD-FMK
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    Z-YVAD-FMK

    Catalog No. A16317
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    Caspase-1 抑制剂
    Z-YVAD-FMK是有效的细胞渗透性和caspase-1不可逆抑制剂。 了解更多
  46. Z-VAD(OH)-FMK
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    Z-VAD(OH)-FMK

    Catalog No. A16340
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    Caspase 抑制剂
    Z-VAD(OH)-FMK是所有胱天蛋白酶的不可逆三肽抑制剂。 了解更多
  47. Z-FA-FMK
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    Z-FA-FMK

    Catalog No. A16381
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    Cysteine protease 抑制剂
    Z-FA-FMK是半胱氨酸蛋白酶的不可逆抑制剂。 了解更多
  48. MX1013
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    • 最新产品

    MX1013

    Catalog No. A17218
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    pan-caspase inhibitor
    MX1013 is a dipeptide pan-caspase inhibitor that inhibits caspase-1, caspase-3, and caspase-6, 7, 8, and 9. 了解更多
  49. VX-765 (Belnacasan)
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    VX-765 (Belnacasan)

    Catalog No. A10984
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    Caspase-1/4 抑制剂
    VX-765 (Belnacasan)是一种新型的Caspase-1抑制剂，是一种控制两种细胞因子IL-1b和IL-18生成的酶。 了解更多
  50. Z-VAD-FMK
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    Z-VAD-FMK

    Catalog No. A12373
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    Pan Caspase 抑制剂
    Z-VAD-FMK是一种细胞可渗透、不可逆的泛胱天蛋白酶抑制剂。体外抑制肿瘤细胞caspase加工和凋亡诱导(IC50 = 0.0015 - 5.8 mM)。活跃在体内。 了解更多

产品 251 到 300 共 319个

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  1. Caspase (32)
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  3. Proteasome (25)
  4. HCV Protease (50)
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  9. Aminopeptidase (4)
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  12. Tyrosinase (3)
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  15. Elastases (6)
  16. ADAMs (5)
作用机制
  1. Inhibitor (抑制剂) (292)
  2. Agonist (激动剂) (3)
  3. Activator (激活剂) (3)
  4. Modulator (调节剂) (10)
  5. Inducer (诱导剂) (1)
  6. Substrate (底物) (3)
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  1. Caspase-1 (8)
  2. Caspase-10 (4)
  3. Caspase-2 (4)
  4. Caspase-3 (13)
  5. Caspase-4 (6)
  6. Caspase-5 (5)
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  8. Caspase-7 (6)
  9. Caspase-8 (5)
  10. Caspase-9 (8)
  11. Pan-Caspase (3)
  12. Procaspase-3 (1)
  13. procaspase-7 (1)
  14. Procaspase-9 (1)
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